Page last updated: 2024-09-03

sb 204070a and sdz 205-557

sb 204070a has been researched along with sdz 205-557 in 6 studies

Compound Research Comparison

Studies
(sb 204070a)
Trials
(sb 204070a)
Recent Studies (post-2010)
(sb 204070a)
Studies
(sdz 205-557)
Trials
(sdz 205-557)
Recent Studies (post-2010) (sdz 205-557)
45045609
10025609

Protein Interaction Comparison

ProteinTaxonomysb 204070a (IC50)sdz 205-557 (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.2512
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.2512

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (83.33)18.2507
2000's1 (16.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Franks, CM; Hardcastle, J; Hardcastle, PT; Sanger, GJ1
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI1
Banner, SE; Bywater, D; Gaster, LM; Sanger, GJ; Smith, MI1
Kadowaki, M; Kontoh, A; Nagakura, Y; Shimomura, K; Tokita, K; Tomoi, M1
Ellis, ES; Gaster, LM; Jennings, AJ; Joiner, GF; King, FD; Mulholland, KR; Rahman, SK; Starr, S; Wardle, KA; Wyman, PA1
Boulouard, M; Bureau, R; Butt-Gueulle, S; Dauphin, F; Daveu, C; Duchatelle, P; Dumuis, A; Lelong-Boulouard, V; LemaƮtre, S; Lepailleur, A; Lezoualc'h, F; Pfeiffer, B; Rault, S1

Other Studies

6 other study(ies) available for sb 204070a and sdz 205-557

ArticleYear
Do 5-HT4 receptors mediate the intestinal secretory response to 5-HT in rat in-vivo?
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; 5-Methoxytryptamine; Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Colon; Dioxanes; Dose-Response Relationship, Drug; Heart Rate; Ileum; Indoles; Intestinal Mucosa; Jejunum; Male; para-Aminobenzoates; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron

1995
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach

1995
Increased defaecation caused by 5-HT4 receptor activation in the mouse.
    European journal of pharmacology, 1996, Jul-18, Volume: 308, Issue:2

    Topics: 4-Aminobenzoic Acid; 5-Hydroxytryptophan; Animals; Defecation; Dioxanes; Feces; Male; Mice; para-Aminobenzoates; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Water

1996
Combined blockade of 5-HT3- and 5-HT4-serotonin receptors inhibits colonic functions in conscious rats and mice.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:1

    Topics: 4-Aminobenzoic Acid; Animals; Colon; Dioxanes; Male; Mice; Ondansetron; para-Aminobenzoates; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists

1997
(1-Butyl-4-piperidinyl)methyl 8-amino-7-chloro-1,4-benzodioxane-5-carboxylate hydrochloride: a highly potent and selective 5-HT4 receptor antagonist derived from metoclopramide.
    Journal of medicinal chemistry, 1993, Dec-10, Volume: 36, Issue:25

    Topics: Animals; Dioxanes; Guinea Pigs; Metoclopramide; Muscle Contraction; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1993
Novel antagonists of serotonin-4 receptors: synthesis and biological evaluation of pyrrolothienopyrazines.
    Bioorganic & medicinal chemistry, 2009, Mar-15, Volume: 17, Issue:6

    Topics: Animals; Chlorocebus aethiops; COS Cells; Humans; Indoles; Models, Molecular; Molecular Structure; Pyrazines; Radioligand Assay; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists; Sulfonamides

2009