Page last updated: 2024-09-03

sb 204070a and ritanserin

sb 204070a has been researched along with ritanserin in 5 studies

Compound Research Comparison

Studies
(sb 204070a)
Trials
(sb 204070a)
Recent Studies (post-2010)
(sb 204070a)
Studies
(ritanserin)
Trials
(ritanserin)
Recent Studies (post-2010) (ritanserin)
45047357571

Protein Interaction Comparison

ProteinTaxonomysb 204070a (IC50)ritanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.001
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.047
Diacylglycerol kinase alphaHomo sapiens (human)9
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.047
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0025
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0012
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.047
D(2) dopamine receptorRattus norvegicus (Norway rat)0.012

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's3 (60.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Kaisar, M; Naylor, RJ; Tuladhar, BR1
Beleta, J; Bernabeu, E; Bou, J; Cortijo, J; Domènech, T; Fernández, AG; Martí-Cabrera, M; Morcillo, EJ; Palacios, JM1
Naylor, RJ; Tuladhar, BR; Womack, MD1

Other Studies

5 other study(ies) available for sb 204070a and ritanserin

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Evidence for a 5-HT3 receptor involvement in the facilitation of peristalsis on mucosal application of 5-HT in the guinea pig isolated ileum.
    British journal of pharmacology, 1997, Volume: 122, Issue:6

    Topics: Animals; Dioxanes; Female; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methiothepin; Mucous Membrane; Ondansetron; Peristalsis; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Ritanserin; Serotonin; Serotonin Antagonists

1997
Characterization of 5-HT receptors on human pulmonary artery and vein: functional and binding studies.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Abortifacient Agents, Nonsteroidal; Adult; Aged; Benzamides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Dinoprost; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidines; Pulmonary Artery; Pulmonary Veins; Pyridines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstrictor Agents

1997
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000