sb 204070a has been researched along with piperidines in 36 studies
Studies (sb 204070a) | Trials (sb 204070a) | Recent Studies (post-2010) (sb 204070a) | Studies (piperidines) | Trials (piperidines) | Recent Studies (post-2010) (piperidines) |
---|---|---|---|---|---|
45 | 0 | 4 | 40,235 | 5,221 | 14,545 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 19 (52.78) | 18.2507 |
2000's | 14 (38.89) | 29.6817 |
2010's | 3 (8.33) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bingham, S; Ellis, ES; Gaster, LM; Joiner, GF; King, FD; Sanger, GJ; Sutton, JM; Wardle, KA; Wyman, PA | 1 |
Bonhaus, DW; Clark, RD; Eglen, RM; Hegde, SS; Johnson, LG; Leung, E | 1 |
Franks, CM; Hardcastle, J; Hardcastle, PT; Sanger, GJ | 1 |
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI | 1 |
Baxter, GS; Ellis, ES; Gaster, LM; Kennett, GA; Sanger, GJ; Wardle, KA | 1 |
Eglen, RM; Hedge, SS; Loeb, M; Moy, TM; Perry, MR | 1 |
Ellis, ES; Gaster, LM; Jennings, AJ; Joiner, GF; King, FD; Mulholland, KR; Rahman, SK; Starr, S; Wardle, KA; Wyman, PA | 1 |
Briejer, MR; Schuurkes, JA | 1 |
Banner, SE; Bywater, D; Gaster, LM; Sanger, GJ; Smith, MI | 1 |
Fernández, AG; Palacios, JM; Silvestre, JS | 1 |
Kadowaki, M; Kontoh, A; Nagakura, Y; Shimomura, K; Tokita, K; Tomoi, M | 1 |
Kaisar, M; Naylor, RJ; Tuladhar, BR | 1 |
Beleta, J; Bernabeu, E; Bou, J; Cortijo, J; Domènech, T; Fernández, AG; Martí-Cabrera, M; Morcillo, EJ; Palacios, JM | 1 |
Hagan, J; Hatcher, JP; Lewis, VA; Reavill, C; Sanger, GJ | 1 |
Ikeda, K; Nagai, N; Takada, A; Takada, Y; Teramoto, Y; Urano, T | 1 |
Kaibara, M; Mameya, S; Takada, K; Takemura, K; Taniyama, K | 1 |
Enjoji, A; Kanematsu, T; Sakurai-Yamashita, Y; Takada, K; Takemura, K; Taniyama, K; Yamashita, K | 1 |
Hamada, Y; Hioki, K; Kaibara, M; Nakane, Y; Sakurai-Yamashita, Y; Takada, K; Taniyama, K; Yamashita, K | 1 |
Akkermans, LM; Briejer, MR; Prins, NH; Schuurkes, JA; Van Bergen, PJ | 1 |
Ito, H; Kiso, T; Miyata, K; Nagakura, Y; Yamaguchi, T | 1 |
Amor, AL; Bandeira, IP; Carvalho, FL; Castro, L; De Castro-E-Silva, E; Ferreira, MG; Fregoneze, JB; Lima, AK; Macêdo, DF; Maldonado, I; Oliveira, IR; Rocha, MA; Santamaria, GF; Souza, FS | 1 |
Bertrand, PP; Bornstein, JC; Furness, JB; Kunze, WA | 1 |
Naylor, RJ; Tuladhar, BR; Womack, MD | 1 |
Bosmans, JP; Briejer, MR; Heylen, L; Jurzak, M; Leysen, JE; Prins, NH; Schuurkes, JA; Van Daele, P | 1 |
Davies, CH; Gill, CH; Hagan, JJ; Soffin, EM | 1 |
Leclere, PG; Lefebvre, RA | 1 |
Ge, L; Naylor, RJ; Tuladhar, BR | 1 |
Barrett, KE; Isenberg, JI; Paulus, P; Sellers, Z; Tuo, BG | 1 |
Karaki, S; Kuwahara, A; Mitsui, R; Ono, S | 2 |
Bindslev, N; Engelmann, BE; Hansen, MB; Larsen, R; Poulsen, SS | 1 |
Barrett, KE; Buret, AG; Chappell, AE; Dong, H; Smith, AJ | 1 |
Amano, T; Ariga, H; Ishida, T; Kimura, T; Matsueda, K; Tajiri, H; Torii, A; Uehara, H; Yamato, S | 1 |
Karaki, S; Kuwahara, A | 1 |
Alagille, D; Barret, O; Caillé, F; Fowles, K; Holden, D; Lee, H; Morley, TJ; Papin, C; Seibyl, JP; Tamagnan, GD; Tavares, AA | 1 |
Kawatani, M; Koyama, Y; Matsumoto-Miyai, K; Shimada, S; Shinzawa, E; Yamada, E; Yoshizumi, M | 1 |
36 other study(ies) available for sb 204070a and piperidines
Article | Year |
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N-[(1-butyl-4-piperidinyl)methyl]-3,4dihydro-2H-[1,3]oxazino[3,2- a]indole10-carboxamide hydrochloride: the first potent and selective 5-HT4 receptor antagonist amide with oral activity.
Topics: Administration, Oral; Animals; Dioxanes; Dogs; Guinea Pigs; Indoles; Muscle Contraction; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Structure-Activity Relationship; Sulfonamides | 1995 |
RS 39604: a potent, selective and orally active 5-HT4 receptor antagonist.
Topics: Administration, Oral; Animals; Colon; Dioxanes; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; Indoles; Male; Mice; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Sulfonamides; Time Factors | 1995 |
Do 5-HT4 receptors mediate the intestinal secretory response to 5-HT in rat in-vivo?
Topics: 4-Aminobenzoic Acid; 5-Methoxytryptamine; Animals; Benzamides; Blood Pressure; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Cisapride; Colon; Dioxanes; Dose-Response Relationship, Drug; Heart Rate; Ileum; Indoles; Intestinal Mucosa; Jejunum; Male; para-Aminobenzoates; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tropisetron | 1995 |
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach | 1995 |
The effects of SB 204070, a highly potent and selective 5-HT4 receptor antagonist, on guinea-pig distal colon.
Topics: Animals; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dimethylphenylpiperazinium Iodide; Dioxanes; Guinea Pigs; In Vitro Techniques; Male; Muscle, Smooth; Piperidines; Radioligand Assay; Receptors, Neurotransmitter; Receptors, Serotonin; Serotonin Antagonists | 1994 |
Evidence for the involvement of 5-hydroxytryptamine 4 receptors in 5-hydroxytryptophan-induced diarrhea in mice.
Topics: 5-Hydroxytryptophan; Animals; Atropine; Benserazide; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diarrhea; Dioxanes; Indoles; Male; Mice; Parasympathetic Nervous System; Piperidines; Receptors, Serotonin; Sulfonamides | 1994 |
(1-Butyl-4-piperidinyl)methyl 8-amino-7-chloro-1,4-benzodioxane-5-carboxylate hydrochloride: a highly potent and selective 5-HT4 receptor antagonist derived from metoclopramide.
Topics: Animals; Dioxanes; Guinea Pigs; Metoclopramide; Muscle Contraction; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship | 1993 |
5-HT3 and 5-HT4 receptors and cholinergic and tachykininergic neurotransmission in the guinea-pig proximal colon.
Topics: Animals; Biphenyl Compounds; Colon; Dioxanes; Dose-Response Relationship, Drug; Drug Interactions; Female; Granisetron; Guinea Pigs; In Vitro Techniques; Interneurons; Male; Motor Neurons; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-1; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists | 1996 |
Increased defaecation caused by 5-HT4 receptor activation in the mouse.
Topics: 4-Aminobenzoic Acid; 5-Hydroxytryptophan; Animals; Defecation; Dioxanes; Feces; Male; Mice; para-Aminobenzoates; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Water | 1996 |
Effects of 5-HT4 receptor antagonists on rat behaviour in the elevated plus-maze test.
Topics: Animals; Behavior, Animal; Diazepam; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Indoles; Male; Maze Learning; Piperidines; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Sulfonamides | 1996 |
Combined blockade of 5-HT3- and 5-HT4-serotonin receptors inhibits colonic functions in conscious rats and mice.
Topics: 4-Aminobenzoic Acid; Animals; Colon; Dioxanes; Male; Mice; Ondansetron; para-Aminobenzoates; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists | 1997 |
Evidence for a 5-HT3 receptor involvement in the facilitation of peristalsis on mucosal application of 5-HT in the guinea pig isolated ileum.
Topics: Animals; Dioxanes; Female; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Male; Methiothepin; Mucous Membrane; Ondansetron; Peristalsis; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Ritanserin; Serotonin; Serotonin Antagonists | 1997 |
Characterization of 5-HT receptors on human pulmonary artery and vein: functional and binding studies.
Topics: Abortifacient Agents, Nonsteroidal; Adult; Aged; Benzamides; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Dinoprost; Dioxanes; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidines; Pulmonary Artery; Pulmonary Veins; Pyridines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sumatriptan; Vasoconstrictor Agents | 1997 |
5-HT4 receptor antagonism does not affect motor and reward mechanisms in the rat.
Topics: Amphetamine; Animals; Behavior, Animal; Cocaine; Dioxanes; Hyperkinesis; Male; Motor Activity; Nicotine; Piperidines; Rats; Rats, Sprague-Dawley; Self Stimulation; Serotonin Antagonists | 1998 |
Plasma levels of 5-HT and 5-HIAA increased after intestinal ischemia/reperfusion in rats.
Topics: 5-Methoxytryptamine; Animals; Dioxanes; Disease Models, Animal; Hydroxyindoleacetic Acid; Intestines; Isoindoles; Male; Piperazines; Piperidines; Pyrimidines; Rats; Rats, Wistar; Reperfusion Injury; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 1998 |
Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach.
Topics: Animals; Atropine; Dioxanes; Enzyme Inhibitors; Female; Gastric Fundus; Granisetron; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscarinic Antagonists; Muscle Relaxation; Muscle Tonus; Nitroarginine; Piperidines; Pyloric Antrum; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Tetrodotoxin | 1999 |
Ability of mosapride to bind to 5-HT4 receptor in the human stomach.
Topics: Aged; Animals; Benzamides; Binding Sites; Binding, Competitive; Dioxanes; Dose-Response Relationship, Drug; Female; Gastric Mucosa; Gastrointestinal Agents; Guinea Pigs; Humans; Iodine Radioisotopes; Male; Middle Aged; Morpholines; Piperidines; Radioligand Assay; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Stomach | 1999 |
Regional difference in correlation of 5-HT4 receptor distribution with cholinergic transmission in the guinea pig stomach.
Topics: Acetylcholine; Animals; Autoradiography; Binding Sites; Binding, Competitive; Dioxanes; Female; Gastric Fundus; Gastric Mucosa; Guinea Pigs; In Vitro Techniques; Iodine Radioisotopes; Male; Piperidines; Pyloric Antrum; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin Antagonists; Stomach; Synaptic Transmission | 1999 |
Evidence for 5-HT7 receptors mediating relaxation of human colonic circular smooth muscle.
Topics: Colon; Dioxanes; Humans; In Vitro Techniques; Muscle, Smooth; Piperidines; Receptors, Serotonin; Serotonin Antagonists | 1999 |
The role of 5-hydroxytryptamine3 and 5-hydroxytryptamine4 receptors in the regulation of gut motility in the ferret.
Topics: Animals; Benzimidazoles; Dioxanes; Ferrets; Gastrointestinal Motility; Male; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Receptors, Serotonin, 5-HT4; Serotonin Antagonists | 2000 |
Central 5-HT(4) receptors and drinking behavior.
Topics: Animals; Dioxanes; Drinking; Drinking Behavior; Indoles; Injections, Intraventricular; Male; Piperidines; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Sulfonamides; Thirst; Water Deprivation | 2000 |
The terminals of myenteric intrinsic primary afferent neurons of the guinea-pig ileum are excited by 5-hydroxytryptamine acting at 5-hydroxytryptamine-3 receptors.
Topics: 5-Methoxytryptamine; Action Potentials; Animals; Dioxanes; Granisetron; Guinea Pigs; Ileum; Indoles; Myenteric Plexus; Neurons, Afferent; Piperidines; Presynaptic Terminals; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Signal Transduction; Tropisetron | 2000 |
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron | 2000 |
The in vitro pharmacological profile of prucalopride, a novel enterokinetic compound.
Topics: Acetylcholine; Animals; Benzofurans; Binding, Competitive; Carbachol; Cell Line; CHO Cells; Colon; Cricetinae; Dioxanes; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Esophagus; Female; Gallbladder; Gastrointestinal Agents; Granisetron; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Indoles; Indomethacin; Male; Motilin; Muscle Contraction; Piperidines; Rabbits; Rats; Rats, Wistar; Receptors, Cholecystokinin; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Gastrointestinal Hormone; Receptors, Neuropeptide; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sincalide; Stomach; Sulfonamides; Vasodilator Agents | 2001 |
5-HT7 receptors modulate synchronized network activity in rat hippocampus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dioxanes; Extracellular Space; Hippocampus; Male; Membrane Potentials; Microelectrodes; Nerve Net; Piperazines; Piperidines; Potassium Channels, Calcium-Activated; Pyramidal Cells; Pyridines; Rats; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2002 |
Presynaptic modulation of cholinergic neurotransmission in the human proximal stomach.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Adult; Aged; Aged, 80 and over; Atropine; Benzofurans; Brimonidine Tartrate; Dioxanes; Enzyme Inhibitors; Evoked Potentials; Female; Gastric Fundus; Gastrointestinal Agents; Humans; Male; Middle Aged; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroprusside; Piperidines; Quinoxalines; Receptors, Cholinergic; Receptors, Muscarinic; Receptors, Presynaptic; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Receptors, Vasoactive Intestinal Peptide; Serotonin Antagonists; Stomach; Synaptic Transmission; Vasoactive Intestinal Peptide; Yohimbine | 2002 |
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides | 2003 |
5-HT induces duodenal mucosal bicarbonate secretion via cAMP- and Ca2+-dependent signaling pathways and 5-HT4 receptors in mice.
Topics: Animals; Bicarbonates; Calcium Signaling; Cyclic AMP; Dioxanes; Dose-Response Relationship, Drug; Duodenum; Intestinal Mucosa; Ion Channels; Mice; Piperidines; Receptors, Serotonin, 5-HT4; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Serotonin; Serotonin Receptor Agonists; Signal Transduction; Sulfonamides | 2004 |
Neural and non-neural mediation of propionate-induced contractile responses in the rat distal colon.
Topics: Acetates; Anesthetics, Local; Animals; Atropine; Butyrates; Colon; Cyclooxygenase Inhibitors; Dioxanes; Dose-Response Relationship, Drug; Enteric Nervous System; Fatty Acids, Volatile; Intestinal Mucosa; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Piperidines; Piroxicam; Propionates; Rats; Receptors, Serotonin; Serotonin Antagonists | 2005 |
Muscarinic and 5-HT4 receptors participate in the regulation of the frequency of spontaneous contractions of the longitudinal muscle in rat distal colon.
Topics: Animals; Atropine; Colon; Dioxanes; Gastrointestinal Motility; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists | 2005 |
Functional characterization of serotonin receptor subtypes in human duodenal secretion.
Topics: Adult; Aged; Bumetanide; Dioxanes; Duodenum; Female; Helicobacter Infections; Helicobacter pylori; Humans; In Vitro Techniques; Intestinal Secretions; Ion Transport; Ketanserin; Male; Middle Aged; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium Potassium Chloride Symporter Inhibitors | 2006 |
5-Hydroxytryptamine contributes significantly to a reflex pathway by which the duodenal mucosa protects itself from gastric acid injury.
Topics: Animals; Bicarbonates; Calcium; Dioxanes; Duodenum; Gastric Acid; Intestinal Mucosa; Mice; Piperidines; Reflex; Serotonin; Serotonin Antagonists; Sodium-Calcium Exchanger; Thiourea; Time Factors | 2006 |
Urocortin I is present in the enteric nervous system and exerts an excitatory effect via cholinergic and serotonergic pathways in the rat colon.
Topics: Animals; Atropine; Colon; Corticotropin-Releasing Hormone; Dioxanes; Electric Stimulation; Enteric Nervous System; Gastrointestinal Motility; Hexamethonium; Immunohistochemistry; Male; NG-Nitroarginine Methyl Ester; Ondansetron; Peptide Fragments; Piperidines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Tetrodotoxin; Urocortins | 2007 |
Propionate-induced epithelial K(+) and Cl(-)/HCO3(-) secretion and free fatty acid receptor 2 (FFA2, GPR43) expression in the guinea pig distal colon.
Topics: Animals; Atropine; Bicarbonates; Bumetanide; Capsaicin; Chlorides; Colon; Dioxanes; Enteroendocrine Cells; Fatty Acids, Nonesterified; Granisetron; Guinea Pigs; Hexamethonium; Intestinal Mucosa; Male; omega-Conotoxin GVIA; Piperidines; Potassium; Propionates; Pyridoxal Phosphate; Receptors, G-Protein-Coupled; Serous Membrane; Suramin; Tetrodotoxin | 2011 |
In vivo evaluation of 18F-MNI698: an 18F-labeled radiotracer for imaging of serotonin 4 receptors in brain.
Topics: Animals; Brain; Brain Mapping; Dioxanes; Dose-Response Relationship, Radiation; Female; Fluorine Radioisotopes; Image Processing, Computer-Assisted; Kinetics; Macaca mulatta; Male; Piperidines; Positron-Emission Tomography; Radiopharmaceuticals; Receptors, Serotonin, 5-HT4; Reproducibility of Results; Serotonin Antagonists; Time Factors; Tissue Distribution | 2014 |
Serotonergic regulation of distention-induced ATP release from the urothelium.
Topics: Adenosine Triphosphate; Animals; Citalopram; Dioxanes; Male; Mice; Oxadiazoles; Piperazines; Piperidines; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin, 5-HT4; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Urinary Bladder; Urothelium | 2016 |