Page last updated: 2024-09-03

sb 204070a and ketanserin

sb 204070a has been researched along with ketanserin in 5 studies

Compound Research Comparison

Studies
(sb 204070a)
Trials
(sb 204070a)
Recent Studies (post-2010)
(sb 204070a)
Studies
(ketanserin)
Trials
(ketanserin)
Recent Studies (post-2010) (ketanserin)
45043,094335283

Protein Interaction Comparison

ProteinTaxonomysb 204070a (IC50)ketanserin (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0021
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.015
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.015
5-hydroxytryptamine receptor 1DHomo sapiens (human)0.265
5-hydroxytryptamine receptor 1BHomo sapiens (human)6.5
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0184
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0027
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0016
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.29
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.015
D(2) dopamine receptorRattus norvegicus (Norway rat)1.8
Synaptic vesicular amine transporterHomo sapiens (human)0.18
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.001

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (40.00)18.2507
2000's3 (60.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI1
Kaibara, M; Mameya, S; Takada, K; Takemura, K; Taniyama, K1
Naylor, RJ; Tuladhar, BR; Womack, MD1
Ge, L; Naylor, RJ; Tuladhar, BR1
Bindslev, N; Engelmann, BE; Hansen, MB; Larsen, R; Poulsen, SS1

Other Studies

5 other study(ies) available for sb 204070a and ketanserin

ArticleYear
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach

1995
Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach.
    Japanese journal of pharmacology, 1999, Volume: 79, Issue:1

    Topics: Animals; Atropine; Dioxanes; Enzyme Inhibitors; Female; Gastric Fundus; Granisetron; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscarinic Antagonists; Muscle Relaxation; Muscle Tonus; Nitroarginine; Piperidines; Pyloric Antrum; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Tetrodotoxin

1999
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
5-HT7 receptors mediate the inhibitory effect of 5-HT on peristalsis in the isolated guinea-pig ileum.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Animals; Dioxanes; Dose-Response Relationship, Drug; Granisetron; Guinea Pigs; Ileum; In Vitro Techniques; Ketanserin; Peristalsis; Phenols; Piperidines; Receptors, Serotonin; Serotonin; Sulfonamides

2003
Functional characterization of serotonin receptor subtypes in human duodenal secretion.
    Basic & clinical pharmacology & toxicology, 2006, Volume: 98, Issue:2

    Topics: Adult; Aged; Bumetanide; Dioxanes; Duodenum; Female; Helicobacter Infections; Helicobacter pylori; Humans; In Vitro Techniques; Intestinal Secretions; Ion Transport; Ketanserin; Male; Middle Aged; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sodium Potassium Chloride Symporter Inhibitors

2006