Page last updated: 2024-09-03

sb 204070a and atropine

sb 204070a has been researched along with atropine in 9 studies

Compound Research Comparison

Studies
(sb 204070a)
Trials
(sb 204070a)
Recent Studies (post-2010)
(sb 204070a)
Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010) (atropine)
450426,7111,2591,697

Protein Interaction Comparison

ProteinTaxonomysb 204070a (IC50)atropine (IC50)
cystic fibrosis transmembrane conductance regulatorHomo sapiens (human)21.41
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.012
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.0067
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.0007
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.0009
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.0015
Muscarinic acetylcholine receptor M3Homo sapiens (human)0.0021
Alpha-1D adrenergic receptorHomo sapiens (human)1.354
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.012

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (33.33)18.2507
2000's5 (55.56)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI1
Eglen, RM; Hedge, SS; Loeb, M; Moy, TM; Perry, MR1
Kaibara, M; Mameya, S; Takada, K; Takemura, K; Taniyama, K1
Naylor, RJ; Tuladhar, BR; Womack, MD1
Leclere, PG; Lefebvre, RA1
Karaki, S; Kuwahara, A; Mitsui, R; Ono, S2
Amano, T; Ariga, H; Ishida, T; Kimura, T; Matsueda, K; Tajiri, H; Torii, A; Uehara, H; Yamato, S1
Karaki, S; Kuwahara, A1

Other Studies

9 other study(ies) available for sb 204070a and atropine

ArticleYear
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach

1995
Evidence for the involvement of 5-hydroxytryptamine 4 receptors in 5-hydroxytryptophan-induced diarrhea in mice.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:2

    Topics: 5-Hydroxytryptophan; Animals; Atropine; Benserazide; Benzimidazoles; Bridged Bicyclo Compounds; Bridged Bicyclo Compounds, Heterocyclic; Diarrhea; Dioxanes; Indoles; Male; Mice; Parasympathetic Nervous System; Piperidines; Receptors, Serotonin; Sulfonamides

1994
Regional and functional differences of 5-hydroxytryptamine-receptor subtypes in guinea pig stomach.
    Japanese journal of pharmacology, 1999, Volume: 79, Issue:1

    Topics: Animals; Atropine; Dioxanes; Enzyme Inhibitors; Female; Gastric Fundus; Granisetron; Guinea Pigs; In Vitro Techniques; Ketanserin; Male; Methysergide; Muscarinic Antagonists; Muscle Relaxation; Muscle Tonus; Nitroarginine; Piperidines; Pyloric Antrum; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach; Tetrodotoxin

1999
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
Presynaptic modulation of cholinergic neurotransmission in the human proximal stomach.
    British journal of pharmacology, 2002, Volume: 135, Issue:1

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adult; Aged; Aged, 80 and over; Atropine; Benzofurans; Brimonidine Tartrate; Dioxanes; Enzyme Inhibitors; Evoked Potentials; Female; Gastric Fundus; Gastrointestinal Agents; Humans; Male; Middle Aged; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroprusside; Piperidines; Quinoxalines; Receptors, Cholinergic; Receptors, Muscarinic; Receptors, Presynaptic; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Receptors, Vasoactive Intestinal Peptide; Serotonin Antagonists; Stomach; Synaptic Transmission; Vasoactive Intestinal Peptide; Yohimbine

2002
Neural and non-neural mediation of propionate-induced contractile responses in the rat distal colon.
    Neurogastroenterology and motility, 2005, Volume: 17, Issue:4

    Topics: Acetates; Anesthetics, Local; Animals; Atropine; Butyrates; Colon; Cyclooxygenase Inhibitors; Dioxanes; Dose-Response Relationship, Drug; Enteric Nervous System; Fatty Acids, Volatile; Intestinal Mucosa; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Piperidines; Piroxicam; Propionates; Rats; Receptors, Serotonin; Serotonin Antagonists

2005
Muscarinic and 5-HT4 receptors participate in the regulation of the frequency of spontaneous contractions of the longitudinal muscle in rat distal colon.
    Biomedical research (Tokyo, Japan), 2005, Volume: 26, Issue:4

    Topics: Animals; Atropine; Colon; Dioxanes; Gastrointestinal Motility; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists

2005
Urocortin I is present in the enteric nervous system and exerts an excitatory effect via cholinergic and serotonergic pathways in the rat colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2007, Volume: 293, Issue:4

    Topics: Animals; Atropine; Colon; Corticotropin-Releasing Hormone; Dioxanes; Electric Stimulation; Enteric Nervous System; Gastrointestinal Motility; Hexamethonium; Immunohistochemistry; Male; NG-Nitroarginine Methyl Ester; Ondansetron; Peptide Fragments; Piperidines; Pyrimidines; Pyrroles; Rats; Receptors, Corticotropin-Releasing Hormone; Serotonin 5-HT3 Receptor Antagonists; Serotonin 5-HT4 Receptor Antagonists; Tetrodotoxin; Urocortins

2007
Propionate-induced epithelial K(+) and Cl(-)/HCO3(-) secretion and free fatty acid receptor 2 (FFA2, GPR43) expression in the guinea pig distal colon.
    Pflugers Archiv : European journal of physiology, 2011, Volume: 461, Issue:1

    Topics: Animals; Atropine; Bicarbonates; Bumetanide; Capsaicin; Chlorides; Colon; Dioxanes; Enteroendocrine Cells; Fatty Acids, Nonesterified; Granisetron; Guinea Pigs; Hexamethonium; Intestinal Mucosa; Male; omega-Conotoxin GVIA; Piperidines; Potassium; Propionates; Pyridoxal Phosphate; Receptors, G-Protein-Coupled; Serous Membrane; Suramin; Tetrodotoxin

2011