Page last updated: 2024-09-05

sb 203580 and wortmannin

sb 203580 has been researched along with wortmannin in 82 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(wortmannin)
Trials
(wortmannin)
Recent Studies (post-2010) (wortmannin)
3,48941,1374,0662726

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)wortmannin (IC50)
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoformHomo sapiens (human)0.0465
Myosin light chain kinase, smooth muscleGallus gallus (chicken)0.26
Metabotropic glutamate receptor 1Rattus norvegicus (Norway rat)0.0085
Phosphatidylinositol 3-kinase regulatory subunit alphaHomo sapiens (human)0.2368
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoformHomo sapiens (human)0.1309
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoformHomo sapiens (human)0.0493
Serine/threonine-protein kinase mTORHomo sapiens (human)0.04
Phosphatidylinositol 4-kinase alphaHomo sapiens (human)0.28
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Homo sapiens (human)0.0492
Serine/threonine-protein kinase PLK1Homo sapiens (human)0.4433
Myosin light chain kinase, smooth muscleHomo sapiens (human)2.3567
Phosphoinositide 3-kinase regulatory subunit 5Homo sapiens (human)0.019
Serine/threonine-protein kinase PLK3Homo sapiens (human)0.1057
Phosphatidylinositol 4-kinase betaHomo sapiens (human)0.44

Research

Studies (82)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (7.32)18.2507
2000's68 (82.93)29.6817
2010's7 (8.54)24.3611
2020's1 (1.22)2.80

Authors

AuthorsStudies
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
McGovern, SL; Shoichet, BK1
Bilter, GK; Dias, J; Huang, Z; Keon, BH; Lamerdin, J; MacDonald, ML; Michnick, SW; Minami, T; Owens, S; Shang, Z; Westwick, JK; Yu, H1
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Henne, WA; Kularatne, SA; Low, PS; Santhapuram, HK; Vaitilingam, B; Venkatesh, C; Wang, K1
Laufer, S; Pillaiyar, T1
Begum, N; Duddy, N; McCarthy, M; Ragolia, L; Rienzie, J1
Bracke, M; Coffer, PJ; Koenderman, L; Lammers, JW1
Coffey, ET; Courtney, MJ1
Benítez, D; Buxadé, M; Casaroli-Marano, RP; Espel, E; Fernández-Troy, N; Pérez-Maldonado, C; Ramírez, M1
Barnes, PJ; Giembycz, MA; Hellewell, PG; Lindsay, MA; Lynch, OT1
Arch, JR; Docherty, K; James, RF; MacFarlane, WM; Tadayyon, M; Wu, H1
Fujita, Y; Hirasawa, N; Ohuchi, K; Sato, Y1
Heads, RJ; Marber, MS; Mockridge, JW1
Fujimoto, M; Fukuyama, H; Kawazoe, Y; Kishimoto, T; Morita, Y; Nagata, S; Naka, T; Nakagawa, R; Narazaki, M1
da Silva Xavier, G; Hooper, S; Rafiq, I; Rutter, GA1
Dickenson, JM; Germack, R1
Alessi, DR; Cuenda, A1
Boos, MD; Chini, CC; Dick, CJ; Leibson, PJ; Schoon, RA1
Lee, J; Mira-Arbibe, L; Ulevitch, RJ1
Chen, CS; Dods, P; Gagnon, A; Roustan-Delatour, N; Sorisky, A1
Anversa, P; Bishopric, NH; Discher, DJ; Kajstura, J; Wasserlauf, BJ; Webster, KA; Yamashita, K1
Cruise, L; Fuller, G; Ho, LK; Morris, BJ; Veitch, K1
Fish, EN; Fujita, S; Grumbach, IM; Lekmine, F; Majchrzak, B; Mayer, IA; Platanias, LC; Ravandi, F; Uddin, S; Verma, A1
Buridi, A; Coxon, PY; Kettritz, R; Klein, JB; Manning, T; McLeish, KR; Rane, MJ1
Hayashi, M; Klip, A; Konrad, D; Ramlal, T; Somwar, R; Sweeney, G; Yaworsky, K1
Chen, KY; Chiu, SL; Hsu, HY; Hua, KF; Wen, MH1
Dobashi, K; Ichimonji, I; Iizuka, K; Ishiwara, M; Ishizuka, T; Kawata, T; Mori, M; Nakazawa, T; Okajima, F; Tsukagoshi, H1
Bae, MA; Pie, JE; Song, BJ1
Docherty, K; Elrick, LJ1
Kobayashi, Y; Kurosaka, K; Watanabe, N1
Barnes, PJ; Giembycz, MA; Lindsay, MA; Lynch, OT1
Brunelleschi, S; Colangelo, D; Gaudino, G; Lavagno, L; Penengo, L; Santoro, C; Viano, I1
Kandolf, R; Küpper, JH; Meyer, RG; Rodemann, HP1
Gosmanov, AR; Thomason, DB1
Betti, M; Canesi, L; Ciacci, C; Citterio, B; Gallo, G; Pruzzo, C; Scarpato, A1
Akasaki, T; Inanami, O; Kuwabara, M; Nagahata, H; Sumimoto, H; Yamamori, T1
Cruciani, V; Mikalsen, SO1
Antonescu, CN; Bilan, PJ; Klip, A; Konrad, D; Liu, Z; Nawaz, Z; Niu, W; Rudich, A; Sweeney, G1
Buresi, MC; Buret, AG; Hollenberg, MD; MacNaughton, WK1
Kito, K; Nishida, Ki1
Kikuta, K; Masamune, A; Sakai, Y; Satoh, A; Satoh, M; Shimosegawa, T1
Eggo, MC; Holder, JC; Kumar, S; Patel, NG; Smith, SA1
Greenberg, DA; Jin, K; Mao, XO; Zhu, Y1
Guan, KL; Inoki, K; Li, Y; Vacratsis, P1
Lai, MZ; Wang, JM; Yang-Yen, HF1
Andriantsitohaina, R; Beretz, A; Chang, SJ; Chataigneau, M; Chataigneau, T; Keravis, T; Oak, MH; Schini-Kerth, VB; Stoclet, JC1
Blanquet, PR; Derer, P; Mariani, J1
Dobashi, K; Ishizuka, T; Masubuchi, K; Mori, M; Nakazawa, T; Shimizu, Y; Utsugi, M1
Christoffersen, T; Guren, TK; Thoresen, GH1
Hebert, C; Nikitakis, NG; Norris, K; Sauk, JJ; Siavash, H; Stewart, J1
Coppens, A; Hooghe-Peters, E; Kooijman, R1
Agrawal, DK; DelCore, MG; Hunter, WJ; Krueger, KD1
Burt, HM; Hampong, M; Higo, TT; Jackson, JK; Pelech, SL; Tudan, C1
Consoli, A; De Caterina, R; Madonna, R; Massaro, M; Pandolfi, A1
Cohen, RA; Hou, X; Jiang, B; Pimentel, DR; Xu, S1
Hori, M; Karaki, H; Ozaki, H; Tasaki, K; Wakabayashi, I1
Chung, TW; Kim, CH; Lee, YC1
Ariga, H; Matsumoto, K; Minamitani, T; Orba, Y; Sato, M; Sawa, H1
Allen, WE; Campbell, M; Sawyer, C; Trimble, ER; Vanhaesebroeck, B1
Aikin, R; Maysinger, D; Rosenberg, L1
Chiou, WF; Tsai, HR; Tsai, WJ; Yang, LM1
Cho, ML; Kim, HY; Kim, KW; Lee, SH; Park, MK; Park, SH; Yoon, CH1
Fujisaki, K; Itoh, Y; Kubota, T; Oishi, R; Yano, T1
Chang, WC; Tseng, JT; Wang, JM1
Iso, T; Kanai, H; Kurabayashi, M; Nagai, R; Ohyama, Y; Sakamoto, H; Sato, H; Sato, M; Tamura, J; Uchiyama, T1
Chang, YC; Hsu, JD; Huang, HP; Wang, CJ; Yang, SF1
Ferjan, I; Stempelj, M1
Blume, N; Friedrichsen, BN; Gram, VK; Lee, YC; Møldrup, A; Neubauer, N; Nielsen, JH; Petersen, JS1
Reimer, RA1
Gómez, R; Gomez-Reino, JJ; Gualillo, O; Lago, F; Lago, R; Otero, M1
Engelbrecht, AM; Louw, L; Toit-Kohn, JL1
Chittrakarn, S; Janchawee, B; Kansenalak, S; Keawpradub, N; Purintrapiban, J; Sawangjaroen, K1
Caimmi, PP; Grossini, E; Mary, DA; Molinari, C; Ribichini, F; Uberti, F; Vacca, G1
Carraro-Lacroix, LR; Girardi, AC; Malnic, G1
Balbo, V; Boccafoschi, F; Burlando, B; Mazzucco, L; Ranzato, E1
Jeon, YT; Kim, SH; Kim, YB; Lee, SC; Song, YS1
Anwer, MS; Schonhoff, CM; Webster, CR1
Chen, DB; Feng, L; Liao, WX; Zheng, J1
Chetkovich, D; Golding, NL; Khurana, S; Lewis, AS; Liu, Z; Rosa, K1
Deng, XL; Li, GR; Su, XL; Wang, Y; Zhao, LM1
Anada, T; Ishiko-Uzuka, R; Nishikawa, R; Suzuki, O1

Reviews

2 review(s) available for sb 203580 and wortmannin

ArticleYear
Kinases as Potential Therapeutic Targets for Anti-coronaviral Therapy.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Antiviral Agents; COVID-19; COVID-19 Drug Treatment; Humans; Protein Kinase Inhibitors; SARS-CoV-2; Signal Transduction; Virus Replication

2022
Use of kinase inhibitors to dissect signaling pathways.
    Methods in molecular biology (Clifton, N.J.), 2000, Volume: 99

    Topics: Androstadienes; Animals; Chromones; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Maleimides; Morpholines; Protein Kinase Inhibitors; Pyridines; Signal Transduction; Sirolimus; Wortmannin

2000

Other Studies

80 other study(ies) available for sb 203580 and wortmannin

ArticleYear
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Kinase inhibitors: not just for kinases anymore.
    Journal of medicinal chemistry, 2003, Apr-10, Volume: 46, Issue:8

    Topics: beta-Lactamase Inhibitors; beta-Lactamases; Chymotrypsin; Enzyme Inhibitors; Kinetics; Light; Malate Dehydrogenase; Models, Biological; Phosphotransferases; Scattering, Radiation

2003
Identifying off-target effects and hidden phenotypes of drugs in human cells.
    Nature chemical biology, 2006, Volume: 2, Issue:6

    Topics: Bacterial Proteins; Cell Line; Cell Proliferation; Cluster Analysis; Drug Design; Drug Evaluation, Preclinical; Genetics; Humans; Luminescent Proteins; Molecular Structure; Phenotype; Recombinant Fusion Proteins; Signal Transduction; Structure-Activity Relationship

2006
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
Synthesis and biological analysis of prostate-specific membrane antigen-targeted anticancer prodrugs.
    Journal of medicinal chemistry, 2010, Nov-11, Volume: 53, Issue:21

    Topics: Antigens, Surface; Antineoplastic Agents; Cell Line, Tumor; Cell Survival; Drug Screening Assays, Antitumor; Glutamate Carboxypeptidase II; Glutarates; Humans; Ligands; Male; Molecular Targeted Therapy; Prodrugs; Prostatic Neoplasms; Structure-Activity Relationship; Urea

2010
Regulation of mitogen-activated protein kinase phosphatase-1 induction by insulin in vascular smooth muscle cells. Evaluation of the role of the nitric oxide signaling pathway and potential defects in hypertension.
    The Journal of biological chemistry, 1998, Sep-25, Volume: 273, Issue:39

    Topics: Androstadienes; Animals; Cell Cycle Proteins; Cells, Cultured; Cyclic GMP; Dual Specificity Phosphatase 1; Enzyme Inhibitors; Flavonoids; Imidazoles; Immediate-Early Proteins; Insulin; Male; Muscle, Smooth, Vascular; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Phosphatidylinositol 3-Kinases; Phosphoprotein Phosphatases; Protein Phosphatase 1; Protein Tyrosine Phosphatases; Pyridines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; RNA, Messenger; Signal Transduction; Wortmannin

1998
Analysis of signal transduction pathways regulating cytokine-mediated Fc receptor activation on human eosinophils.
    Journal of immunology (Baltimore, Md. : 1950), 1998, Dec-15, Volume: 161, Issue:12

    Topics: Androstadienes; Calcium-Calmodulin-Dependent Protein Kinases; Chromones; Enzyme Activation; Enzyme Inhibitors; Eosinophils; Flavonoids; Humans; Imidazoles; Immunoglobulin A; Immunoglobulin G; Interleukin-4; Interleukin-5; Microspheres; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase Inhibitors; Protein Kinases; Protein Processing, Post-Translational; Pyridines; Receptors, Fc; Receptors, IgG; Rosette Formation; Signal Transduction; Th2 Cells; Wortmannin

1998
The mechanism of Ara-C-induced apoptosis of differentiating cerebellar granule neurons.
    The European journal of neuroscience, 1999, Volume: 11, Issue:3

    Topics: Androstadienes; Animals; Antimetabolites, Antineoplastic; Apoptosis; Benzamides; CDC2 Protein Kinase; CDC2-CDC28 Kinases; Cell Differentiation; Cell Survival; Cerebellum; Cyclin-Dependent Kinase 2; Cyclin-Dependent Kinase 4; Cyclin-Dependent Kinase 5; Cyclin-Dependent Kinases; Cytarabine; Enzyme Inhibitors; Flavonoids; Imatinib Mesylate; Imidazoles; Mitogen-Activated Protein Kinase 12; Mitogen-Activated Protein Kinases; Neurons; Piperazines; Piperidines; Poly (ADP-Ribose) Polymerase-1; Poly(ADP-ribose) Polymerases; Protein Kinases; Protein Serine-Threonine Kinases; Proteins; Proto-Oncogene Proteins; Purines; Pyridines; Pyrimidines; Rats; Roscovitine; Signal Transduction; Stress, Physiological; Wortmannin

1999
Wortmannin inhibits translation of tumor necrosis factor-alpha in superantigen-activated T cells.
    International immunology, 1999, Volume: 11, Issue:9

    Topics: Androstadienes; Bacterial Toxins; CD4-Positive T-Lymphocytes; Chromones; Enterotoxins; Enzyme Inhibitors; Humans; Imidazoles; Immunosuppressive Agents; Morpholines; Phosphatidylinositol 3-Kinases; Pyridines; RNA, Messenger; Superantigens; Transcription, Genetic; Tumor Necrosis Factor-alpha; Wortmannin

1999
'Outside-in' signalling mechanisms underlying CD11b/CD18-mediated NADPH oxidase activation in human adherent blood eosinophils.
    British journal of pharmacology, 1999, Volume: 128, Issue:6

    Topics: Androstadienes; Carbazoles; CD18 Antigens; Cell Adhesion; Cell Count; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Eosinophils; Humans; Imidazoles; Indoles; Isoenzymes; Macrophage-1 Antigen; Maleimides; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Pyrazoles; Pyridines; Pyrimidines; Signal Transduction; src-Family Kinases; Superoxides; Tetradecanoylphorbol Acetate; Wortmannin

1999
Insulin stimulates pancreatic-duodenal homoeobox factor-1 (PDX1) DNA-binding activity and insulin promoter activity in pancreatic beta cells.
    The Biochemical journal, 1999, Dec-15, Volume: 344 Pt 3

    Topics: Androstadienes; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Chromones; DNA-Binding Proteins; Glucose; Homeodomain Proteins; Humans; Imidazoles; Insulin; Islets of Langerhans; Mitogen-Activated Protein Kinases; Morpholines; Oligodeoxyribonucleotides; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphorylation; Promoter Regions, Genetic; Pyridines; Trans-Activators; Transfection; Wortmannin

1999
Involvement of a phosphatidylinositol 3-kinase-p38 mitogen activated protein kinase pathway in antigen-induced IL-4 production in mast cells.
    Biochimica et biophysica acta, 2000, Jan-03, Volume: 1456, Issue:1

    Topics: Activating Transcription Factor 2; Androstadienes; Animals; Cell Line; Chromones; Cyclic AMP Response Element-Binding Protein; Dinitrophenols; Enzyme Activation; Flavonoids; Imidazoles; Interleukin-4; Mast Cells; Mitogen-Activated Protein Kinases; Morpholines; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Pyridines; Rats; Serum Albumin; Transcription Factors; Wortmannin

2000
Activation of Akt during simulated ischemia/reperfusion in cardiac myocytes.
    Biochemical and biophysical research communications, 2000, Apr-21, Volume: 270, Issue:3

    Topics: Androstadienes; Animals; Animals, Newborn; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Genistein; Imidazoles; Kinetics; Models, Cardiovascular; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Oncogene Protein v-akt; Phosphatidylinositol 3-Kinases; Phosphorylation; Phosphoserine; Phosphotyrosine; Protein-Tyrosine Kinases; Pyridines; Rats; Retroviridae Proteins, Oncogenic; Wortmannin

2000
Signals transducers and activators of transcription (STAT)-induced STAT inhibitor-1 (SSI-1)/suppressor of cytokine signaling-1 (SOCS-1) suppresses tumor necrosis factor alpha-induced cell death in fibroblasts.
    Proceedings of the National Academy of Sciences of the United States of America, 2000, May-09, Volume: 97, Issue:10

    Topics: Androstadienes; Animals; Carrier Proteins; Caspase 3; Caspase Inhibitors; Caspases; Cell Death; Cell Survival; Cytokines; DNA-Binding Proteins; Embryo, Mammalian; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Imidazoles; Interferon-gamma; Interleukin-1; Kinetics; L Cells; Mice; Mice, Knockout; Pyridines; Recombinant Proteins; Repressor Proteins; Signal Transduction; STAT1 Transcription Factor; Suppressor of Cytokine Signaling 1 Protein; Suppressor of Cytokine Signaling Proteins; Trans-Activators; Transfection; Tumor Necrosis Factor-alpha; Wortmannin

2000
Glucose-stimulated preproinsulin gene expression and nuclear trans-location of pancreatic duodenum homeobox-1 require activation of phosphatidylinositol 3-kinase but not p38 MAPK/SAPK2.
    The Journal of biological chemistry, 2000, May-26, Volume: 275, Issue:21

    Topics: Androstadienes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cell Nucleus; Chromones; Enzyme Activation; Enzyme Inhibitors; Gene Expression Regulation; Glucose; Homeodomain Proteins; Imidazoles; Insulin; Islets of Langerhans; MAP Kinase Kinase 6; Microscopy, Confocal; Mitogen-Activated Protein Kinases; Morpholines; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Proinsulin; Promoter Regions, Genetic; Protein Kinase C; Protein Precursors; Pyridines; Signal Transduction; Trans-Activators; Transfection; Wortmannin

2000
Activation of protein kinase B by the A(1)-adenosine receptor in DDT(1)MF-2 cells.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Adenosine; Androstadienes; Animals; Calcium; Cell Line; Chromones; Cricetinae; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genistein; Imidazoles; Indoles; Insulin; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Morpholines; Pertussis Toxin; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyridines; Receptors, Purinergic P1; Virulence Factors, Bordetella; Wortmannin; Xanthines

2000
Regulation of p38 mitogen-activated protein kinase during NK cell activation.
    European journal of immunology, 2000, Volume: 30, Issue:10

    Topics: Androstadienes; Antibody-Dependent Cell Cytotoxicity; Cytotoxicity, Immunologic; Enzyme Inhibitors; Enzyme Precursors; Flavonoids; Humans; Imidazoles; Indoles; Intracellular Signaling Peptides and Proteins; Killer Cells, Natural; Lymphocyte Activation; Maleimides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Protein-Tyrosine Kinases; Pyridines; Receptors, IgG; src-Family Kinases; Syk Kinase; Wortmannin

2000
TAK1 regulates multiple protein kinase cascades activated by bacterial lipopolysaccharide.
    Journal of leukocyte biology, 2000, Volume: 68, Issue:6

    Topics: Androstadienes; Animals; Apoptosis; Cell Line; Chromones; Cysteine Proteinase Inhibitors; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Humans; Hydrogen Peroxide; Hypertonic Solutions; I-kappa B Kinase; Imidazoles; Inflammation; Insulin-Like Growth Factor I; Interleukin-1; JNK Mitogen-Activated Protein Kinases; Lipopolysaccharides; MAP Kinase Kinase Kinases; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinases; Morpholines; NF-kappa B; Okadaic Acid; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Prostaglandins A; Protein Kinases; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Recombinant Fusion Proteins; Signal Transduction; Stress, Physiological; Transfection; Tumor Cells, Cultured; Wortmannin

2000
Phosphatidylinositol-3,4,5-trisphosphate is required for insulin-like growth factor 1-mediated survival of 3T3-L1 preadipocytes.
    Endocrinology, 2001, Volume: 142, Issue:1

    Topics: 3T3 Cells; Adipocytes; Androstadienes; Animals; Apoptosis; Chromones; Culture Media, Serum-Free; Enzyme Inhibitors; Flavonoids; Imidazoles; In Situ Nick-End Labeling; Insulin-Like Growth Factor I; MAP Kinase Kinase 1; Mice; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Morpholines; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol Phosphates; Phosphoinositide-3 Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyridines; Sirolimus; Wortmannin

2001
Reperfusion-activated Akt kinase prevents apoptosis in transgenic mouse hearts overexpressing insulin-like growth factor-1.
    Circulation research, 2001, Mar-30, Volume: 88, Issue:6

    Topics: Androstadienes; Animals; Apoptosis; DNA Fragmentation; Enzyme Activation; Enzyme Inhibitors; Female; Genotype; Imidazoles; Insulin-Like Growth Factor I; Male; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinases; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; p38 Mitogen-Activated Protein Kinases; Perfusion; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Wortmannin

2001
Activation of p44/p42 MAP kinase in striatal neurons via kainate receptors and PI3 kinase.
    Brain research. Molecular brain research, 2001, Apr-18, Volume: 89, Issue:1-2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Androstadienes; Animals; Corpus Striatum; Dizocilpine Maleate; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Flavonoids; Imidazoles; JNK Mitogen-Activated Protein Kinases; Kainic Acid; MAP Kinase Kinase 4; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; N-Methylaspartate; Neurons; Phosphatidylinositol 3-Kinases; Phosphorylation; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Receptors, N-Methyl-D-Aspartate; Wortmannin

2001
The p38 MAPK pathway mediates the growth inhibitory effects of interferon-alpha in BCR-ABL-expressing cells.
    The Journal of biological chemistry, 2001, Jul-27, Volume: 276, Issue:30

    Topics: Androstadienes; Cell Division; Cell Line; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Enzyme Inhibitors; Fusion Proteins, bcr-abl; Genistein; Humans; Imidazoles; Immunoblotting; Interferon-alpha; Intracellular Signaling Peptides and Proteins; K562 Cells; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Serine-Threonine Kinases; Pyridines; Tyrosine; Wortmannin

2001
Role of extracellular signal-regulated kinase and phosphatidylinositol-3 kinase in chemoattractant and LPS delay of constitutive neutrophil apoptosis.
    Cellular signalling, 2001, Volume: 13, Issue:5

    Topics: Androstadienes; Apoptosis; Chemotaxis, Leukocyte; Chromones; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Leukotriene B4; Lipopolysaccharides; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Morpholines; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Virulence Factors, Bordetella; Wortmannin

2001
The antihyperglycemic drug alpha-lipoic acid stimulates glucose uptake via both GLUT4 translocation and GLUT4 activation: potential role of p38 mitogen-activated protein kinase in GLUT4 activation.
    Diabetes, 2001, Volume: 50, Issue:6

    Topics: 3T3 Cells; Androstadienes; Animals; Arabidopsis Proteins; Biological Transport; Deoxyglucose; Enzyme Inhibitors; Glucose; Glucose Transporter Type 4; Hypoglycemic Agents; Imidazoles; Mice; Mitogen-Activated Protein Kinases; Monosaccharide Transport Proteins; Muscle Fibers, Skeletal; Muscle Proteins; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Plant Proteins; Potassium Channels; Pyridines; Thioctic Acid; Wortmannin

2001
Ligands of macrophage scavenger receptor induce cytokine expression via differential modulation of protein kinase signaling pathways.
    The Journal of biological chemistry, 2001, Aug-03, Volume: 276, Issue:31

    Topics: Androstadienes; Animals; Cell Adhesion Molecules; Cell Line; Chromones; Cytokines; Enzyme Inhibitors; Flavonoids; Fucose; Gene Expression Regulation; Imidazoles; Interleukin-1; JNK Mitogen-Activated Protein Kinases; Kinetics; Ligands; Lipoproteins, LDL; Macrophages; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Models, Biological; Morpholines; Oxidation-Reduction; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Polysaccharides; Pyridines; Receptors, Immunologic; Receptors, Scavenger; Time Factors; Tumor Necrosis Factor-alpha; Wortmannin

2001
Sensitized mast cells migrate toward the antigen: a response regulated by p38 mitogen-activated protein kinase and Rho-associated coiled-coil-forming protein kinase.
    Journal of immunology (Baltimore, Md. : 1950), 2001, Aug-15, Volume: 167, Issue:4

    Topics: Androstadienes; Animals; Cell Movement; Cells, Cultured; Clone Cells; Dinitrophenols; Enzyme Activation; Enzyme Inhibitors; Female; Flavonoids; Haptens; Imidazoles; Immunization; Immunoglobulin E; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 1; Mast Cells; Mice; Mice, Inbred BALB C; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-kit; Pyridines; Receptors, IgE; rho-Associated Kinases; Serum Albumin; Wortmannin

2001
Acetaminophen induces apoptosis of C6 glioma cells by activating the c-Jun NH(2)-terminal protein kinase-related cell death pathway.
    Molecular pharmacology, 2001, Volume: 60, Issue:4

    Topics: Acetaminophen; Acetanilides; Analgesics; Analgesics, Non-Narcotic; Androstadienes; Animals; Apoptosis; bcl-2-Associated X Protein; Caspase 3; Caspases; Cytochrome c Group; Cytochrome P-450 CYP2E1; DNA Fragmentation; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Glioma; Imidazoles; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-bcl-2; Pyridines; Rats; Thiazoles; Time Factors; Tumor Cells, Cultured; Wortmannin

2001
Phosphorylation-dependent nucleocytoplasmic shuttling of pancreatic duodenal homeobox-1.
    Diabetes, 2001, Volume: 50, Issue:10

    Topics: Androstadienes; Arsenites; Biological Transport; Cell Line; Cell Nucleus; Cytoplasm; Enzyme Inhibitors; Glucose; Homeodomain Proteins; Humans; Imidazoles; Immunohistochemistry; Insulin; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphorylation; Pyridines; Sodium Compounds; Trans-Activators; Wortmannin

2001
Production of proinflammatory cytokines by resident tissue macrophages after phagocytosis of apoptotic cells.
    Cellular immunology, 2001, Jul-10, Volume: 211, Issue:1

    Topics: Androstadienes; Animals; Apoptosis; Cell Line; Cells, Cultured; Chemokine CXCL2; Chemokines; Colchicine; Cytokines; Enzyme Inhibitors; Imidazoles; Kupffer Cells; Lipopolysaccharides; Macrophages, Alveolar; Male; Mice; Mice, Inbred C57BL; Phagocytosis; Pyridines; RNA, Messenger; T-Lymphocytes; Thymus Gland; Wortmannin

2001
Pharmacological comparison of LTB(4)-induced NADPH oxidase activation in adherent and non-adherent guinea-pig eosinophils.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Androstadienes; Animals; Antibodies; Carbazoles; CD18 Antigens; Cell Adhesion; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Enzyme Precursors; Eosinophils; Flavonoids; Guinea Pigs; Imidazoles; Indoles; Integrin beta1; Intracellular Signaling Peptides and Proteins; Leukotriene B4; Macrophage-1 Antigen; Male; Maleimides; Mitogen-Activated Protein Kinases; NADPH Oxidases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase C; Protein-Tyrosine Kinases; Pyrazoles; Pyridines; Pyrimidines; Rats; src-Family Kinases; Stilbenes; Syk Kinase; Time Factors; Wortmannin

2001
Macrophage stimulating protein (MSP) evokes superoxide anion production by human macrophages of different origin.
    British journal of pharmacology, 2001, Volume: 134, Issue:6

    Topics: Adult; Androstadienes; Animals; Caenorhabditis elegans Proteins; Carrier Proteins; Flavonoids; Growth Substances; Hepatocyte Growth Factor; Humans; Imidazoles; Insecta; Macrophages; Middle Aged; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Protein Kinase C; Proto-Oncogene Proteins; Pyridines; Receptors, Drug; Respiratory Burst; Signal Transduction; Superoxides; Tetradecanoylphorbol Acetate; Wortmannin

2001
Early growth response-1 gene (Egr-1) promoter induction by ionizing radiation in U87 malignant glioma cells in vitro.
    European journal of biochemistry, 2002, Volume: 269, Issue:1

    Topics: Androstadienes; Anisomycin; Blotting, Western; Colforsin; DNA-Binding Proteins; Early Growth Response Protein 1; Epidermal Growth Factor; Flavonoids; Glioma; Humans; Imidazoles; Immediate-Early Proteins; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Pyridines; Suramin; Transcription Factors; Wortmannin

2002
Insulin and isoproterenol differentially regulate mitogen-activated protein kinase-dependent Na(+)-K(+)-2Cl(-) cotransporter activity in skeletal muscle.
    Diabetes, 2002, Volume: 51, Issue:3

    Topics: Androstadienes; Animals; Chromones; Female; Imidazoles; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; Muscle, Skeletal; p38 Mitogen-Activated Protein Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Potassium; Pyridines; Rats; Rats, Sprague-Dawley; Rubidium Radioisotopes; Sodium-Potassium-Chloride Symporters; Wortmannin

2002
Signaling pathways involved in the physiological response of mussel hemocytes to bacterial challenge: the role of stress-activated p38 MAP kinases.
    Developmental and comparative immunology, 2002, Volume: 26, Issue:4

    Topics: Androstadienes; Animals; Bivalvia; Enzyme Activation; Enzyme Inhibitors; Escherichia coli; Flavonoids; Hemocytes; Imidazoles; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Signal Transduction; Wortmannin

2002
Relationship between p38 mitogen-activated protein kinase and small GTPase Rac for the activation of NADPH oxidase in bovine neutrophils.
    Biochemical and biophysical research communications, 2002, May-24, Volume: 293, Issue:5

    Topics: Androstadienes; Animals; Cattle; Chromones; Cytosol; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Glutathione Transferase; Imidazoles; Immunohistochemistry; Mitogen-Activated Protein Kinases; Morpholines; NADPH Oxidases; Neutrophils; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoproteins; Protein Binding; Protein Structure, Tertiary; Pyridines; rac GTP-Binding Proteins; Recombinant Fusion Proteins; Superoxides; Time Factors; Wortmannin; Zymosan

2002
Mechanisms involved in responses to the poroxisome proliferator WY-14,643 on gap junctional intercellular communication in V79 hamster fibroblasts.
    Toxicology and applied pharmacology, 2002, Jul-01, Volume: 182, Issue:1

    Topics: Acetophenones; Androstadienes; Animals; Benzopyrans; Brefeldin A; Butadienes; Cell Communication; Cells, Cultured; Cricetinae; Cricetulus; Enzyme Inhibitors; Flavonoids; Gap Junctions; Imidazoles; Indoles; Maleimides; Mesocricetus; Mitogen-Activated Protein Kinases; Nitriles; Peroxisome Proliferators; Protein Kinase C; Protein Synthesis Inhibitors; Pyridines; Pyrimidines; Signal Transduction; Sirolimus; Wortmannin

2002
Need for GLUT4 activation to reach maximum effect of insulin-mediated glucose uptake in brown adipocytes isolated from GLUT4myc-expressing mice.
    Diabetes, 2002, Volume: 51, Issue:9

    Topics: Adipocytes; Adipose Tissue, Brown; Androstadienes; Animals; Biological Transport; Cell Membrane; Deoxyglucose; Enzyme Inhibitors; Glucose; Glucose Tolerance Test; Glucose Transporter Type 4; Heterozygote; HIV Protease Inhibitors; Humans; Imidazoles; Indinavir; Insulin; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinases; Monosaccharide Transport Proteins; Muscle Proteins; p38 Mitogen-Activated Protein Kinases; Proto-Oncogene Proteins c-myc; Pyridines; Rats; Sequence Tagged Sites; Wortmannin

2002
Activation of proteinase-activated receptor 1 stimulates epithelial chloride secretion through a unique MAP kinase- and cyclo-oxygenase-dependent pathway.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2002, Volume: 16, Issue:12

    Topics: Androstadienes; Butadienes; Cell Line; Chlorides; Epithelial Cells; Humans; Imidazoles; Indoles; Maleimides; Mitogen-Activated Protein Kinases; Nitriles; Nitrobenzenes; Phospholipases A; Phosphorylation; Prostaglandin-Endoperoxide Synthases; Prostaglandins; Pyrazoles; Pyridines; Pyrimidines; Quinazolines; Receptor, PAR-1; Receptors, Thrombin; Signal Transduction; Sulfonamides; Thrombin; Tyrphostins; Wortmannin

2002
Nonrequirement of continuous stimulation with MCP-1 for cell migration and determination of directional migration by initial stimulation with chemokine.
    Experimental cell research, 2002, Nov-15, Volume: 281, Issue:1

    Topics: Androstadienes; Cell Communication; Cell Movement; Cells, Cultured; Chemokine CCL2; Enzyme Inhibitors; Humans; Imidazoles; Mitogen-Activated Protein Kinases; Monocytes; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Signal Transduction; Wortmannin

2002
Inhibition of p38 mitogen-activated protein kinase blocks activation of rat pancreatic stellate cells.
    The Journal of pharmacology and experimental therapeutics, 2003, Volume: 304, Issue:1

    Topics: Actins; Androstadienes; Animals; Blotting, Northern; Blotting, Western; Cell Division; Cell Nucleus; Cells, Cultured; Chemokine CCL2; Electrophoresis; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Imidazoles; Interleukin-1; Intracellular Signaling Peptides and Proteins; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Pancreas; Phosphorylation; Platelet-Derived Growth Factor; Procollagen; Procollagen-Proline Dioxygenase; Protein Serine-Threonine Kinases; Pyridines; Rats; Wortmannin

2003
Differential regulation of lipogenesis and leptin production by independent signaling pathways and rosiglitazone during human adipocyte differentiation.
    Diabetes, 2003, Volume: 52, Issue:1

    Topics: Adipocytes; Androstadienes; Cell Differentiation; Cell Survival; Cells, Cultured; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Leptin; Lipid Metabolism; Lipids; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Pyridines; Rosiglitazone; Signal Transduction; Sirolimus; Stem Cells; Thiazoles; Thiazolidinediones; Tumor Necrosis Factor-alpha; Wortmannin

2003
Vascular endothelial growth factor promotes proliferation of cortical neuron precursors by regulating E2F expression.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2003, Volume: 17, Issue:2

    Topics: Androstadienes; Animals; Blotting, Western; Bromodeoxyuridine; Cell Cycle Proteins; Cell Division; Cell Nucleus; Cells, Cultured; Cerebral Cortex; Cyclin A; Cyclin D1; Cyclin E; DNA-Binding Proteins; Dose-Response Relationship, Drug; E2F Transcription Factors; E2F1 Transcription Factor; E2F2 Transcription Factor; E2F3 Transcription Factor; Electrophoresis, Polyacrylamide Gel; Endothelial Growth Factors; Flavonoids; Imidazoles; Intercellular Signaling Peptides and Proteins; Lymphokines; Mice; Proliferating Cell Nuclear Antigen; Pyridines; Signal Transduction; Time Factors; Transcription Factors; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Wortmannin

2003
The p38 and MK2 kinase cascade phosphorylates tuberin, the tuberous sclerosis 2 gene product, and enhances its interaction with 14-3-3.
    The Journal of biological chemistry, 2003, Apr-18, Volume: 278, Issue:16

    Topics: 14-3-3 Proteins; Amino Acid Sequence; Androstadienes; Anisomycin; Binding Sites; Culture Media, Serum-Free; Dose-Response Relationship, Drug; Genes, Dominant; Glutathione Transferase; Humans; Imidazoles; Intracellular Signaling Peptides and Proteins; Mass Spectrometry; Mitogen-Activated Protein Kinases; Models, Biological; Molecular Sequence Data; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Plasmids; Precipitin Tests; Protein Binding; Protein Kinases; Protein Serine-Threonine Kinases; Pyridines; Recombinant Fusion Proteins; Repressor Proteins; Sequence Homology, Amino Acid; Serine; Time Factors; Tuberous Sclerosis; Tuberous Sclerosis Complex 2 Protein; Tumor Suppressor Proteins; Tyrosine 3-Monooxygenase; Wortmannin

2003
Interleukin-3 stimulation of mcl-1 gene transcription involves activation of the PU.1 transcription factor through a p38 mitogen-activated protein kinase-dependent pathway.
    Molecular and cellular biology, 2003, Volume: 23, Issue:6

    Topics: Androstadienes; Animals; Cell Line; Cyclic AMP Response Element-Binding Protein; Enzyme Inhibitors; Genes, Immediate-Early; Hematopoietic Stem Cells; Humans; Imidazoles; Interleukin-3; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinases; Mutagenesis, Site-Directed; Myeloid Cell Leukemia Sequence 1 Protein; Neoplasm Proteins; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Promoter Regions, Genetic; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-bcl-2; Pyridines; Recombinant Fusion Proteins; Regulatory Sequences, Nucleic Acid; Trans-Activators; Transcription, Genetic; Wortmannin

2003
Red wine polyphenolic compounds inhibit vascular endothelial growth factor expression in vascular smooth muscle cells by preventing the activation of the p38 mitogen-activated protein kinase pathway.
    Arteriosclerosis, thrombosis, and vascular biology, 2003, Jun-01, Volume: 23, Issue:6

    Topics: Androstadienes; Animals; Antioxidants; Cells, Cultured; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Onium Compounds; p38 Mitogen-Activated Protein Kinases; Phenols; Phosphorylation; Platelet-Derived Growth Factor; Polyphenols; Protein Processing, Post-Translational; Pyridines; Rats; Reactive Oxygen Species; RNA, Messenger; Thrombin; Transforming Growth Factor beta; Transforming Growth Factor beta1; Vascular Endothelial Growth Factor A; Wine; Wortmannin

2003
A calcium/calmodulin kinase pathway connects brain-derived neurotrophic factor to the cyclic AMP-responsive transcription factor in the rat hippocampus.
    Neuroscience, 2003, Volume: 118, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Androstadienes; Animals; Antibodies; Benzophenanthridines; Benzopyrans; Blotting, Western; Brain-Derived Neurotrophic Factor; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Calmodulin; Carbazoles; Cell Nucleus; Chromones; Cyclic AMP Response Element-Binding Protein; Cytosol; Enzyme Inhibitors; Flavonoids; Hippocampus; Imidazoles; Immunohistochemistry; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Male; Morpholines; Naphthalenes; Phenanthridines; Phosphorylation; Precipitin Tests; Protein Serine-Threonine Kinases; Pyridines; Pyrroles; Rats; Signal Transduction; Time Factors; Tyrphostins; Wortmannin

2003
C-Jun-NH2-terminal kinase mediates expression of connective tissue growth factor induced by transforming growth factor-beta1 in human lung fibroblasts.
    American journal of respiratory cell and molecular biology, 2003, Volume: 28, Issue:6

    Topics: Androstadienes; Anthracenes; Cells, Cultured; Chromones; Connective Tissue Growth Factor; DNA-Binding Proteins; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Gene Expression Regulation; Humans; Imidazoles; Immediate-Early Proteins; Intercellular Signaling Peptides and Proteins; JNK Mitogen-Activated Protein Kinases; Lung; Mitogen-Activated Protein Kinase 8; Mitogen-Activated Protein Kinase 9; Mitogen-Activated Protein Kinases; Morpholines; Oligonucleotides, Antisense; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Pyridines; RNA, Messenger; Smad2 Protein; Trans-Activators; Transforming Growth Factor beta; Transforming Growth Factor beta1; Wortmannin

2003
Role of ERK, p38 and PI3-kinase in EGF receptor-mediated mitogenic signalling in cultured rat hepatocytes: requirement for sustained ERK activation.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2003, Volume: 13, Issue:4

    Topics: Androstadienes; Animals; Cells, Cultured; Chromones; Enzyme Activation; Enzyme Inhibitors; ErbB Receptors; Imidazoles; Male; Mitogen-Activated Protein Kinases; Mitogens; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Rats; Rats, Wistar; Signal Transduction; Wortmannin

2003
Phenotypic switching of VEGF and collagen XVIII during hypoxia in head and neck squamous carcinoma cells.
    Oral oncology, 2003, Volume: 39, Issue:8

    Topics: Acetylcysteine; Androstadienes; Antimutagenic Agents; Biomarkers; Cell Hypoxia; Cell Line, Tumor; Cobalt; Collagen Type XVIII; Enzyme Inhibitors; Head and Neck Neoplasms; Heat-Shock Proteins; HSP47 Heat-Shock Proteins; Humans; Imidazoles; MAP Kinase Signaling System; Neovascularization, Pathologic; Phosphatidylinositol 3-Kinases; Phosphodiesterase Inhibitors; Phosphoinositide-3 Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Vascular Endothelial Growth Factor A; Wortmannin

2003
IGF-I stimulates IL-8 production in the promyelocytic cell line HL-60 through activation of extracellular signal-regulated protein kinase.
    Cellular signalling, 2003, Volume: 15, Issue:12

    Topics: Androstadienes; Anthracenes; Apoptosis; Butadienes; Cell Survival; Chromones; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation, Leukemic; HL-60 Cells; Humans; Hydrogen Peroxide; Imidazoles; Insulin-Like Growth Factor I; Interleukin-8; JNK Mitogen-Activated Protein Kinases; Kinetics; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; Nitriles; Oxazoles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Receptor, IGF Type 1; RNA, Messenger; Wortmannin

2003
Calphostin C as a rapid and strong inducer of apoptosis in human coronary artery smooth muscle cells.
    International immunopharmacology, 2003, Volume: 3, Issue:13-14

    Topics: Androstadienes; Animals; Apoptosis; Cells, Cultured; Chromones; Coronary Vessels; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Enzyme-Linked Immunosorbent Assay; Flavonoids; Humans; Imidazoles; In Situ Nick-End Labeling; Insulin-Like Growth Factor I; Microscopy, Electron, Scanning; Microscopy, Video; Mitogen-Activated Protein Kinases; Morpholines; Muscle, Smooth, Vascular; Naphthalenes; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Signal Transduction; Staurosporine; Time Factors; Wortmannin

2003
Calcium pyrophosphate dihydrate crystal associated induction of neutrophil activation and repression of TNF-alpha-induced apoptosis is mediated by the p38 MAP kinase.
    Cellular signalling, 2004, Volume: 16, Issue:2

    Topics: Androstadienes; Apoptosis; Calcium Pyrophosphate; Caspase 3; Caspases; Cell Degranulation; Crystallization; DNA Fragmentation; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Mitogen-Activated Protein Kinases; Muramidase; Neutrophil Activation; Neutrophils; p38 Mitogen-Activated Protein Kinases; Peroxidase; Pyridines; Superoxides; Tumor Necrosis Factor-alpha; Wortmannin

2004
Insulin enhances vascular cell adhesion molecule-1 expression in human cultured endothelial cells through a pro-atherogenic pathway mediated by p38 mitogen-activated protein-kinase.
    Diabetologia, 2004, Volume: 47, Issue:3

    Topics: Androstadienes; Arteriosclerosis; Cells, Cultured; Endothelium, Vascular; Enzyme Inhibitors; Gene Expression Regulation; Humans; Imidazoles; Insulin; Intercellular Adhesion Molecule-1; MAP Kinase Signaling System; p38 Mitogen-Activated Protein Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Signal Transduction; Umbilical Veins; Wortmannin

2004
Angiotensin II differentially regulates interleukin-1-beta-inducible NO synthase (iNOS) and vascular cell adhesion molecule-1 (VCAM-1) expression: role of p38 MAPK.
    The Journal of biological chemistry, 2004, May-07, Volume: 279, Issue:19

    Topics: Adenoviridae; Androstadienes; Angiotensin II; Animals; Blotting, Western; Cells, Cultured; Cyclooxygenase 2; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; Imidazoles; Inflammation; Interleukin-1; Isoenzymes; Microscopy, Fluorescence; Mitogen-Activated Protein Kinases; Models, Biological; NF-kappa B; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphorylation; Prostaglandin-Endoperoxide Synthases; Pyridines; Rats; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Time Factors; Vascular Cell Adhesion Molecule-1; Wortmannin

2004
Mechanism of human urotensin II-induced contraction in rat aorta.
    Journal of pharmacological sciences, 2004, Volume: 94, Issue:4

    Topics: Androstadienes; Animals; Aorta, Thoracic; Butadienes; Calcium; Carbazoles; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Humans; Imidazoles; Indoles; Lanthanum; Male; Maleimides; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Muscle Contraction; Myosin Light Chains; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Potassium Chloride; Protein Kinase C; Pyridines; Rats; Rats, Wistar; Thapsigargin; Urotensins; Verapamil; Wortmannin

2004
Hepatitis B viral HBx induces matrix metalloproteinase-9 gene expression through activation of ERK and PI-3K/AKT pathways: involvement of invasive potential.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2004, Volume: 18, Issue:10

    Topics: Androstadienes; Butadienes; Cell Line; Enzyme Inhibitors; Gene Expression Regulation, Viral; Hepatitis B virus; Hepatocytes; Humans; Imidazoles; MAP Kinase Signaling System; Matrix Metalloproteinase 2; Matrix Metalloproteinase 9; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Neoplasm Invasiveness; NF-kappa B; Nitriles; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Recombinant Fusion Proteins; Signal Transduction; Trans-Activators; Transcription, Genetic; Transfection; Viral Regulatory and Accessory Proteins; Wortmannin

2004
Induction of matrix metalloproteinase-2 by tenascin-X deficiency is mediated through the c-Jun N-terminal kinase and protein tyrosine kinase phosphorylation pathway.
    Experimental cell research, 2004, Jul-15, Volume: 297, Issue:2

    Topics: Androstadienes; Animals; Animals, Newborn; Anthracenes; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Flavonoids; Genistein; Imidazoles; Male; Matrix Metalloproteinase 2; Mice; Mice, Knockout; Phosphorylation; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-jun; Pyridines; Skin; Tenascin; Wortmannin

2004
Glucose-potentiated chemotaxis in human vascular smooth muscle is dependent on cross-talk between the PI3K and MAPK signaling pathways.
    Circulation research, 2004, Aug-20, Volume: 95, Issue:4

    Topics: Alkyl and Aryl Transferases; Androstadienes; Anthracenes; Antibodies, Monoclonal; Cells, Cultured; Chemotaxis; Chromones; Class I Phosphatidylinositol 3-Kinases; Farnesyltranstransferase; Flavonoids; Glucose; Humans; Imidazoles; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Lovastatin; MAP Kinase Kinase 4; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Morpholines; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Polyisoprenyl Phosphates; Protein Kinases; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; ras Proteins; Sesquiterpenes; Sirolimus; TOR Serine-Threonine Kinases; Wortmannin

2004
Cross-talk between phosphatidylinositol 3-kinase/AKT and c-jun NH2-terminal kinase mediates survival of isolated human islets.
    Endocrinology, 2004, Volume: 145, Issue:10

    Topics: Androstadienes; Anthracenes; Apoptosis; Cell Death; Culture Techniques; Cytokines; Cytoprotection; Enzyme Activation; Enzyme Inhibitors; Humans; Imidazoles; Insulin-Like Growth Factor I; Islets of Langerhans; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Tissue Survival; Wortmannin

2004
Andrographolide acts through inhibition of ERK1/2 and Akt phosphorylation to suppress chemotactic migration.
    European journal of pharmacology, 2004, Sep-13, Volume: 498, Issue:1-3

    Topics: Androstadienes; Animals; Anthracenes; Cell Line; Cell Movement; Cell Survival; Chemokine CCL4; Chemotaxis; Chromones; Complement C5a; Diterpenes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Imidazoles; JNK Mitogen-Activated Protein Kinases; Macrophage Inflammatory Proteins; MAP Kinase Kinase 1; MAP Kinase Kinase 2; MAP Kinase Kinase 4; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Morpholines; p38 Mitogen-Activated Protein Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Wortmannin

2004
Increased interleukin-17 production via a phosphoinositide 3-kinase/Akt and nuclear factor kappaB-dependent pathway in patients with rheumatoid arthritis.
    Arthritis research & therapy, 2005, Volume: 7, Issue:1

    Topics: Adult; Aged; Androstadienes; Antibodies, Monoclonal; Arthritis, Rheumatoid; CD28 Antigens; CD3 Complex; CD4-Positive T-Lymphocytes; Chemokines; Chromones; Cytokines; Female; Flavonoids; Gene Expression Regulation; Humans; Imidazoles; Interleukin-17; Leukocytes, Mononuclear; Lymphocyte Activation; Male; Middle Aged; Morpholines; NF-kappa B; Osteoarthritis; Phosphatidylinositol 3-Kinases; Phytohemagglutinins; Proto-Oncogene Proteins c-akt; Pyridines; Pyrrolidines; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Thiocarbamates; Wortmannin

2005
Fenofibrate induces apoptotic injury in cultured human hepatocytes by inhibiting phosphorylation of Akt.
    Apoptosis : an international journal on programmed cell death, 2005, Volume: 10, Issue:2

    Topics: Androstadienes; Annexin A5; Apoptosis; Caspases; Cell Line; Cell Membrane; Cell Nucleus; Cell Survival; DNA; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Fenofibrate; Hepatocytes; Humans; Hydroxyeicosatetraenoic Acids; Hypolipidemic Agents; Imidazoles; In Situ Nick-End Labeling; Insulin; Microscopy, Fluorescence; Phosphatidylinositol 3-Kinases; Phosphatidylserines; Phosphorylation; PPAR alpha; Propidium; Protein Transport; Proto-Oncogene Proteins c-bcl-2; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Wortmannin

2005
Induction of human NF-IL6beta by epidermal growth factor is mediated through the p38 signaling pathway and cAMP response element-binding protein activation in A431 cells.
    Molecular biology of the cell, 2005, Volume: 16, Issue:7

    Topics: Amino Acid Motifs; Androstadienes; Blotting, Western; CCAAT-Enhancer-Binding Protein-delta; Cell Line, Tumor; Cell Nucleus; Chromatin Immunoprecipitation; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Enzyme Inhibitors; Epidermal Growth Factor; Genes, Reporter; Humans; Imidazoles; Inflammation; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Plasmids; Promoter Regions, Genetic; Protein Binding; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Sp1 Transcription Factor; Time Factors; Transfection; Wortmannin

2005
Mitochondrial reactive oxygen species and c-Src play a critical role in hypoxic response in vascular smooth muscle cells.
    Cardiovascular research, 2005, Sep-01, Volume: 67, Issue:4

    Topics: Androstadienes; Animals; Blotting, Northern; Catalase; Cell Hypoxia; Cell Line; Flavonoids; Hydrogen Peroxide; Hypoxia-Inducible Factor 1, alpha Subunit; Imidazoles; Immunoblotting; Microscopy, Fluorescence; Mitochondria; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Naphthalenes; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Plasminogen Activator Inhibitor 1; Protein Kinase Inhibitors; Proto-Oncogene Proteins pp60(c-src); Pyrazoles; Pyridines; Pyrimidines; Rabbits; RNA, Messenger; Rotenone; Wortmannin

2005
Hibiscus anthocyanins rich extract-induced apoptotic cell death in human promyelocytic leukemia cells.
    Toxicology and applied pharmacology, 2005, Jun-15, Volume: 205, Issue:3

    Topics: Androstadienes; Anthocyanins; Anthracenes; Apoptosis; BH3 Interacting Domain Death Agonist Protein; Carrier Proteins; Caspases; Cell Survival; Cytochromes c; DNA, Mitochondrial; Dose-Response Relationship, Drug; Fas Ligand Protein; Flavonoids; Flowers; Hibiscus; HL-60 Cells; Humans; Imidazoles; Membrane Glycoproteins; p38 Mitogen-Activated Protein Kinases; Plant Extracts; Proto-Oncogene Proteins c-jun; Pyridines; RNA, Messenger; Time Factors; Wortmannin

2005
Signaling pathway in nerve growth factor induced histamine release from rat mast cells.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2005, Volume: 54, Issue:8

    Topics: Analysis of Variance; Androstadienes; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Flavonoids; Histamine; Imidazoles; Indoles; Male; Maleimides; Mast Cells; Models, Biological; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Protein Kinase C; Pyridines; Pyrrolidinones; Rats; Rats, Wistar; Signal Transduction; Staurosporine; Tyrosine; Wortmannin

2005
Stimulation of pancreatic beta-cell replication by incretins involves transcriptional induction of cyclin D1 via multiple signalling pathways.
    The Journal of endocrinology, 2006, Volume: 188, Issue:3

    Topics: Adenylyl Cyclases; Androstadienes; Animals; Animals, Newborn; Cell Line; Cell Proliferation; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclin D1; Enzyme Activation; Flavonoids; Gastric Inhibitory Polypeptide; Glucagon-Like Peptide 1; Human Growth Hormone; Imidazoles; Insulin-Secreting Cells; Isoquinolines; Liraglutide; Mitogen-Activated Protein Kinase Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Rats; Signal Transduction; Stimulation, Chemical; Sulfonamides; Transcription, Genetic; Transduction, Genetic; Wortmannin

2006
Meat hydrolysate and essential amino acid-induced glucagon-like peptide-1 secretion, in the human NCI-H716 enteroendocrine cell line, is regulated by extracellular signal-regulated kinase1/2 and p38 mitogen-activated protein kinases.
    The Journal of endocrinology, 2006, Volume: 191, Issue:1

    Topics: Amino Acids, Essential; Androstadienes; Blotting, Western; Butadienes; Cell Line; Depression, Chemical; Enterocytes; Enzyme Activation; Glucagon-Like Peptide 1; Humans; Imidazoles; Meat; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Hydrolysates; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Statistics, Nonparametric; Wortmannin

2006
Phosphatidylinositol 3-kinase, MEK-1 and p38 mediate leptin/interferon-gamma synergistic NOS type II induction in chondrocytes.
    Life sciences, 2007, Oct-27, Volume: 81, Issue:19-20

    Topics: Androstadienes; Animals; Blotting, Western; Cell Line; Cells, Cultured; Chondrocytes; Chromones; Enzyme Induction; Enzyme Inhibitors; Enzymes; Flavonoids; Humans; Imidazoles; Interferon-gamma; Leptin; MAP Kinase Kinase 1; Morpholines; Nitric Oxide Synthase Type II; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Wortmannin

2007
Docosahexaenoic acid induces apoptosis in colorectal carcinoma cells by modulating the PI3 kinase and p38 MAPK pathways.
    The Journal of nutritional biochemistry, 2009, Volume: 20, Issue:2

    Topics: Adenocarcinoma; Androstadienes; Apoptosis; Cell Line, Tumor; Cell Survival; Colonic Neoplasms; Docosahexaenoic Acids; Humans; Imidazoles; Kinetics; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Tumor Cells, Cultured; Wortmannin

2009
Study on glucose transport in muscle cells by extracts from Mitragyna speciosa (Korth) and mitragynine.
    Natural product research, 2011, Volume: 25, Issue:15

    Topics: Androstadienes; Animals; Blotting, Western; Cell Line; Enzyme Inhibitors; Glucose; Imidazoles; Insulin; Mitragyna; Muscles; Plant Extracts; Pyridines; Rats; Secologanin Tryptamine Alkaloids; Signal Transduction; Wortmannin

2011
Urocortin II induces nitric oxide production through cAMP and Ca2+ related pathways in endothelial cells.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2009, Volume: 23, Issue:1-3

    Topics: Androstadienes; Animals; Aorta; Blotting, Western; Butadienes; Calcimycin; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Dideoxyadenosine; Endothelial Cells; Imidazoles; Ionophores; Mitogen-Activated Protein Kinase 3; Nitric Oxide; Nitriles; Oncogene Protein v-akt; p38 Mitogen-Activated Protein Kinases; Peptide Fragments; Peptides, Cyclic; Pyridines; Signal Transduction; Swine; Urocortins; Wortmannin

2009
Long-term regulation of vacuolar H(+)-ATPase by angiotensin II in proximal tubule cells.
    Pflugers Archiv : European journal of physiology, 2009, Volume: 458, Issue:5

    Topics: Ammonium Chloride; Androstadienes; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Animals; Buffers; Cell Line, Transformed; Cell Membrane; Cycloheximide; Dactinomycin; Epithelial Cells; Gene Expression; Genistein; Hydrogen-Ion Concentration; Imidazoles; Kidney Tubules, Proximal; Losartan; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Protein Subunits; Protein Transport; Protein-Tyrosine Kinases; Pyridines; Rats; Time Factors; Up-Regulation; Vacuolar Proton-Translocating ATPases; Wortmannin

2009
Scratch wound closure of C2C12 mouse myoblasts is enhanced by human platelet lysate.
    Cell biology international, 2009, Volume: 33, Issue:9

    Topics: Androstadienes; Animals; Blood Platelets; Cell Line; Cell Movement; Chemotaxis; Complex Mixtures; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Humans; Imidazoles; Mice; Myoblasts; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Signal Transduction; Wortmannin; Wound Healing

2009
Genistein inhibits cell growth by modulating various mitogen-activated protein kinases and AKT in cervical cancer cells.
    Annals of the New York Academy of Sciences, 2009, Volume: 1171

    Topics: Androstadienes; Anthracenes; Anticarcinogenic Agents; Blotting, Western; Cell Line, Tumor; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Flavonoids; Genistein; HeLa Cells; Humans; Imidazoles; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Proto-Oncogene Proteins c-akt; Pyridines; Uterine Cervical Neoplasms; Wortmannin

2009
Cyclic AMP stimulates Mrp2 translocation by activating p38{alpha} MAPK in hepatic cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2010, Volume: 298, Issue:5

    Topics: Androstadienes; Animals; Cell Line, Tumor; Cyclic AMP; Hepatocytes; Humans; Imidazoles; MAP Kinase Kinase 6; MAP Kinase Kinase Kinases; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; p38 Mitogen-Activated Protein Kinases; Protein Transport; Pyridines; Rats; Transfection; Wortmannin

2010
Deciphering mechanisms controlling placental artery endothelial cell migration stimulated by vascular endothelial growth factor.
    Endocrinology, 2010, Volume: 151, Issue:7

    Topics: Androstadienes; Animals; Anthracenes; Arteries; Butadienes; Caveolin 1; Cell Movement; Cells, Cultured; CSK Tyrosine-Protein Kinase; Electrophoresis, Polyacrylamide Gel; Endothelial Cells; Enzyme Inhibitors; Female; Focal Adhesion Protein-Tyrosine Kinases; Imidazoles; Immunoprecipitation; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Nitric Oxide Synthase Type III; Nitriles; Nitrogen Oxides; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Placenta; Pregnancy; Protein-Tyrosine Kinases; Pyridines; Pyrimidines; Sheep; Signal Transduction; src-Family Kinases; Vascular Endothelial Growth Factor A; Wortmannin

2010
An essential role for modulation of hyperpolarization-activated current in the development of binaural temporal precision.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Feb-22, Volume: 32, Issue:8

    Topics: Age Factors; Analysis of Variance; Androstadienes; Animals; Biophysical Phenomena; Bucladesine; Colforsin; Cyclic Nucleotide-Gated Cation Channels; Electric Stimulation; Enzyme Inhibitors; Female; Gene Expression Regulation, Developmental; Gerbillinae; Imidazoles; In Vitro Techniques; Ion Channel Gating; Male; Neurons; Olivary Nucleus; Patch-Clamp Techniques; Pyridines; Pyrimidines; Wortmannin

2012
KCa3.1 channels mediate the increase of cell migration and proliferation by advanced glycation endproducts in cultured rat vascular smooth muscle cells.
    Laboratory investigation; a journal of technical methods and pathology, 2013, Volume: 93, Issue:2

    Topics: Analysis of Variance; Androstadienes; Animals; Blotting, Western; Butadienes; Cell Movement; Cell Proliferation; Cells, Cultured; Chromones; Flavonoids; Glycation End Products, Advanced; Imidazoles; Intermediate-Conductance Calcium-Activated Potassium Channels; Morpholines; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nitriles; Patch-Clamp Techniques; Pyridines; Rats; RNA Interference; RNA, Small Interfering; Serum Albumin, Bovine; Signal Transduction; Wortmannin

2013
Osteoblastic differentiation of stromal ST-2 cells from octacalcium phosphate exposure via p38 signaling pathway.
    Dental materials journal, 2014, Volume: 33, Issue:2

    Topics: Alkaline Phosphatase; Androstadienes; Animals; Calcium Phosphates; Cell Differentiation; Cell Line; Cell Proliferation; Flavonoids; Imidazoles; Mice; Molecular Structure; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Pyridines; Signal Transduction; Stromal Cells; Wortmannin

2014