Page last updated: 2024-09-05

sb 203580 and u 73122

sb 203580 has been researched along with u 73122 in 13 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(u 73122)
Trials
(u 73122)
Recent Studies (post-2010) (u 73122)
3,48941,1371,2522236

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)u 73122 (IC50)
Telomerase reverse transcriptaseHomo sapiens (human)0.2

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (7.69)18.2507
2000's11 (84.62)29.6817
2010's1 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kato, K; Kawamura, H; Kozawa, O; Matsui, N; Matsuno, H; Niwa, M; Otsuka, T; Uematsu, T1
Bansal, R; Baron, W; de Vries, H; Hoekstra, D; Metz, B1
Hatakeyama, D; Kawamura, H; Kozawa, O; Matsuno, H; Uematsu, T1
Kato, K; Kozawa, O; Matsuno, H; Niwa, M; Tokuda, H; Uematsu, T1
DiMattina, AJ; Holland, JA; Johnson, DK; O'Donnell, RW; Stone, RI; Ziegler, LM1
Akiyama, N; Hirabayashi, T; Murayama, T; Shimamura, K; Takashiro, Y1
Coleman, JW; Davis, BJ; Flanagan, BF; Gilfillan, AM; Metcalfe, DD1
Kuan, YH; Lin, CN; Lin, RH; Tsao, LT; Wang, JP1
Ferjan, I; Stempelj, M1
Hu, W; Huang, J; Mahavadi, S; Murthy, KS; Sriwai, W1
Calixto, JB; Motta, EM; Rae, GA1
Ashizuka, M; Ito, S; Kubota, Y; Ogata, S; Satoh, S; Shirasuna, K; Takeuchi, H1
Aoki, M; Hirose, E; Ishimaru, Y; Kawata, J; Matsmoto, T; Narahara, S; Ono, T; Sagara, K; Yamaguchi, Y1

Other Studies

13 other study(ies) available for sb 203580 and u 73122

ArticleYear
Endothelin-1 stimulates heat shock protein 27 induction in osteoblasts: involvement of p38 MAP kinase.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: Animals; Antihypertensive Agents; Blotting, Northern; Carcinogens; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Estrenes; Flavonoids; Gene Expression Regulation, Enzymologic; Genistein; Heat-Shock Proteins; Imidazoles; Mice; Mitogen-Activated Protein Kinases; Naphthalenes; Oligopeptides; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phorbol Esters; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Propranolol; Protein Kinase C; Pyridines; Pyrrolidinones; RNA, Messenger; Skull; Staurosporine

1999
PDGF and FGF-2 signaling in oligodendrocyte progenitor cells: regulation of proliferation and differentiation by multiple intracellular signaling pathways.
    Molecular and cellular neurosciences, 2000, Volume: 15, Issue:3

    Topics: Animals; Cell Differentiation; Cell Division; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Estrenes; Fibroblast Growth Factor 2; Flavonoids; Genistein; Imidazoles; Intracellular Signaling Peptides and Proteins; MAP Kinase Signaling System; Membrane Proteins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Myristoylated Alanine-Rich C Kinase Substrate; Nerve Tissue Proteins; Oligodendroglia; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Platelet-Derived Growth Factor; Protein Kinase C; Protein Processing, Post-Translational; Proteins; Pyridines; Pyrrolidinones; Rats; Ribosomal Protein S6 Kinases; Signal Transduction; Sirolimus; Stem Cells

2000
Endothelin-1 induces vascular endothelial growth factor synthesis in osteoblasts: involvement of p38 mitogen-activated protein kinase.
    Cellular signalling, 2000, Volume: 12, Issue:6

    Topics: Animals; Endothelial Growth Factors; Endothelin-1; Enzyme Inhibitors; Estrenes; Flavonoids; Gene Expression Regulation; Imidazoles; Lymphokines; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinases; Naphthalenes; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phorbol Esters; Protein Kinase C; Pyridines; Pyrrolidinones; Receptor, Endothelin A; Receptors, Endothelin; Tetradecanoylphorbol Acetate; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2000
Mechanism of prostaglandin E2-stimulated heat shock protein 27 induction in osteoblast-like MC3T3-E1 cells.
    The Journal of endocrinology, 2002, Volume: 172, Issue:2

    Topics: Analysis of Variance; Animals; Butadienes; Calcium; Calcium Channel Blockers; Cell Line; Chelating Agents; Dinoprostone; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Estrenes; Flavonoids; Gallic Acid; Heat-Shock Proteins; HSP70 Heat-Shock Proteins; Imidazoles; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Molecular Chaperones; Naphthalenes; Neoplasm Proteins; Nitriles; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Pyridines; Pyrrolidinones; Staurosporine; Stimulation, Chemical; Time Factors; Type C Phospholipases

2002
Endothelial NADPH oxidase: mechanism of activation by low-density lipoprotein.
    Endothelium : journal of endothelial cell research, 2003, Volume: 10, Issue:6

    Topics: Arachidonic Acids; Cells, Cultured; Chromones; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Estrenes; Flavonoids; Humans; Imidazoles; Indoles; Lipoproteins, LDL; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Morpholines; NADPH Oxidases; p38 Mitogen-Activated Protein Kinases; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phospholipase C gamma; Phospholipases A; Protein Kinase C; Pyridines; Pyrrolidinones; Reactive Oxygen Species; Signal Transduction; src-Family Kinases; Type C Phospholipases; Umbilical Veins

2003
Expression of adhesion molecules by sphingosine 1-phosphate and histamine in endothelial cells.
    European journal of pharmacology, 2004, Feb-20, Volume: 486, Issue:2

    Topics: Acetophenones; Benzopyrans; Blotting, Western; Carbazoles; Cell Adhesion Molecules; Cells, Cultured; E-Selectin; Endothelium, Vascular; Estrenes; Histamine; Histamine Agonists; Humans; Imidazoles; Indoles; Intercellular Adhesion Molecule-1; Lysophospholipids; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Pyridines; Pyrrolidinones; RNA, Messenger; Signal Transduction; Sphingosine; Type C Phospholipases; Umbilical Veins; Vascular Cell Adhesion Molecule-1

2004
Nitric oxide inhibits IgE-dependent cytokine production and Fos and Jun activation in mast cells.
    Journal of immunology (Baltimore, Md. : 1950), 2004, Dec-01, Volume: 173, Issue:11

    Topics: Animals; Bone Marrow Cells; Cell Degranulation; Cell Line, Tumor; Cells, Cultured; Cytokines; Estrenes; Imidazoles; Immunoglobulin E; MAP Kinase Signaling System; Mast Cells; Mice; Mice, Inbred BALB C; Nitric Oxide; p38 Mitogen-Activated Protein Kinases; Phospholipase C gamma; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Pyridines; Pyrrolidinones; Rats; RNA, Messenger; Type C Phospholipases

2004
Artocarpol A stimulation of superoxide anion generation in neutrophils involved the activation of PLC, PKC and p38 mitogen-activated PK signaling pathways.
    British journal of pharmacology, 2005, Volume: 145, Issue:4

    Topics: Animals; Butadienes; Calcium; Cell-Free System; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Estrenes; Flavonoids; Heterocyclic Compounds, 4 or More Rings; Imidazoles; Immunoblotting; Indoles; Maleimides; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Pyridines; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Signal Transduction; Superoxides; Tetradecanoylphorbol Acetate; Type C Phospholipases

2005
Signaling pathway in nerve growth factor induced histamine release from rat mast cells.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 2005, Volume: 54, Issue:8

    Topics: Analysis of Variance; Androstadienes; Animals; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Flavonoids; Histamine; Imidazoles; Indoles; Male; Maleimides; Mast Cells; Models, Biological; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Protein Kinase C; Pyridines; Pyrrolidinones; Rats; Rats, Wistar; Signal Transduction; Staurosporine; Tyrosine; Wortmannin

2005
Gi-coupled receptors mediate phosphorylation of CPI-17 and MLC20 via preferential activation of the PI3K/ILK pathway.
    The Biochemical journal, 2006, May-15, Volume: 396, Issue:1

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Animals; Azepines; Calcium; Cells, Cultured; Chromones; Enkephalin, D-Penicillamine (2,5)-; Estrenes; GTP-Binding Protein alpha Subunits, Gi-Go; Imidazoles; Morpholines; Muscle Contraction; Muscle Proteins; Myocytes, Smooth Muscle; Myosin Light Chains; Myosin-Light-Chain Phosphatase; p21-Activated Kinases; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoproteins; Phosphorylation; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-akt; Pyridines; Pyrrolidinones; Rabbits; Receptor, Adenosine A1; Receptor, Muscarinic M2; Receptors, G-Protein-Coupled; Receptors, Opioid, delta; Receptors, Somatostatin; Recombinant Fusion Proteins; RNA, Small Interfering; Signal Transduction; Somatostatin; Transfection

2006
Mechanical hyperalgesia induced by endothelin-1 in rats is mediated via phospholipase C, protein kinase C, and MAP kinases.
    Experimental biology and medicine (Maywood, N.J.), 2006, Volume: 231, Issue:6

    Topics: Animals; Endothelin-1; Enzyme Inhibitors; Estrenes; Hyperalgesia; Imidazoles; Indoles; Injections, Intradermal; Male; Maleimides; p38 Mitogen-Activated Protein Kinases; Protein Kinase C; Pyridines; Pyrrolidinones; Rats; Rats, Wistar; Reaction Time; Signal Transduction; Type C Phospholipases

2006
Ca2+ stimulates COX-2 expression through calcium-sensing receptor in fibroblasts.
    Biochemical and biophysical research communications, 2006, Dec-29, Volume: 351, Issue:4

    Topics: Anthracenes; Bone and Bones; Calcium; Calcium Signaling; Cations, Divalent; Cyclooxygenase 2; Dinoprostone; Estrenes; Fibroblasts; Flavonoids; Humans; Imidazoles; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Pyrrolidinones; Receptors, Calcium-Sensing; RNA, Messenger; Type C Phospholipases

2006
Mechanism of tissue factor production by monocytes stimulated with neutrophil elastase.
    Blood cells, molecules & diseases, 2015, Volume: 54, Issue:2

    Topics: Calcium Channel Blockers; Carbazoles; Enzyme Inhibitors; Estrenes; Flavonoids; Gallic Acid; Gene Expression Regulation; Humans; Imidazoles; Indoles; Leukocyte Elastase; Maleimides; Monocytes; p38 Mitogen-Activated Protein Kinases; Primary Cell Culture; Protein Kinase C; Protein Kinase Inhibitors; Pyridines; Pyrrolidinones; RNA, Messenger; Signal Transduction; Thromboplastin; Type C Phospholipases

2015