sb 203580 has been researched along with troglitazone in 6 studies
Studies (sb 203580) | Trials (sb 203580) | Recent Studies (post-2010) (sb 203580) | Studies (troglitazone) | Trials (troglitazone) | Recent Studies (post-2010) (troglitazone) |
---|---|---|---|---|---|
3,489 | 4 | 1,137 | 1,857 | 146 | 287 |
Protein | Taxonomy | sb 203580 (IC50) | troglitazone (IC50) |
---|---|---|---|
Bile salt export pump | Rattus norvegicus (Norway rat) | 3.9 | |
Bile salt export pump | Homo sapiens (human) | 5.05 | |
Carbonic anhydrase 2 | Homo sapiens (human) | 0.97 | |
Adenosine receptor A3 | Homo sapiens (human) | 5.208 | |
Cytochrome P450 2C9 | Homo sapiens (human) | 4 | |
Alpha-1B adrenergic receptor | Rattus norvegicus (Norway rat) | 5.208 | |
Thromboxane-A synthase | Homo sapiens (human) | 2.966 | |
Amine oxidase [flavin-containing] B | Homo sapiens (human) | 2.07 | |
Mitogen-activated protein kinase 1 | Homo sapiens (human) | 1.238 | |
Peroxisome proliferator-activated receptor gamma | Homo sapiens (human) | 1.03 | |
5-hydroxytryptamine receptor 2B | Homo sapiens (human) | 1.312 | |
Alpha-1A adrenergic receptor | Rattus norvegicus (Norway rat) | 5.208 | |
ATP-binding cassette sub-family C member 8 | Homo sapiens (human) | 1.285 | |
ATP-sensitive inward rectifier potassium channel 11 | Homo sapiens (human) | 1.285 | |
Indoleamine 2,3-dioxygenase 2 | Mus musculus (house mouse) | 4.5 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 5 (83.33) | 29.6817 |
2010's | 1 (16.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bilter, GK; Dias, J; Huang, Z; Keon, BH; Lamerdin, J; MacDonald, ML; Michnick, SW; Minami, T; Owens, S; Shang, Z; Westwick, JK; Yu, H | 1 |
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ | 1 |
Dai, J; Remick, DG; Wang, X; Zeng, X | 1 |
Blaschke, F; Bruemmer, D; Herle, AJ; Hsueh, WA; Law, RE; Yin, F | 1 |
Jung, JY; Kim, HT; Kim, YK; Kwon, CH; Park, JY; Yoo, CI | 1 |
Kim, YK; Kwon, CH; Yoon, CS | 1 |
6 other study(ies) available for sb 203580 and troglitazone
Article | Year |
---|---|
Identifying off-target effects and hidden phenotypes of drugs in human cells.
Topics: Bacterial Proteins; Cell Line; Cell Proliferation; Cluster Analysis; Drug Design; Drug Evaluation, Preclinical; Genetics; Humans; Luminescent Proteins; Molecular Structure; Phenotype; Recombinant Fusion Proteins; Signal Transduction; Structure-Activity Relationship | 2006 |
Identification of potent Yes1 kinase inhibitors using a library screening approach.
Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship | 2013 |
Homocysteine mediated expression and secretion of monocyte chemoattractant protein-1 and interleukin-8 in human monocytes.
Topics: Antioxidants; Cells, Cultured; Chemokine CCL2; Chromans; Dimethyl Sulfoxide; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Genistein; Homocysteine; Humans; Imidazoles; Indoles; Interleukin-8; Monocytes; Naphthalenes; Onium Compounds; Pyridines; Pyrrolidines; Reactive Oxygen Species; RNA, Messenger; Sulfonamides; Thiazoles; Thiazolidinediones; Thiocarbamates; Time Factors; Troglitazone; Tyrphostins | 2003 |
Signaling pathways involved in induction of GADD45 gene expression and apoptosis by troglitazone in human MCF-7 breast carcinoma cells.
Topics: Antineoplastic Agents; Apoptosis; Breast Neoplasms; Carcinoma; Cell Cycle; Chromans; Enzyme Inhibitors; Female; Flavonoids; GADD45 Proteins; Gene Expression Regulation, Neoplastic; Humans; Imidazoles; Intracellular Signaling Peptides and Proteins; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Proteins; Pyridines; RNA, Small Interfering; Signal Transduction; Thiazolidinediones; Troglitazone; Tumor Cells, Cultured | 2004 |
Role of mitogen-activated protein kinase (MAPK) in troglitazone-induced osteoblastic cell death.
Topics: 3T3 Cells; Anilides; Animals; Apoptosis; Blotting, Western; Butadienes; Caspase 3; Caspase Inhibitors; Cell Survival; Chromans; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Flow Cytometry; Hypoglycemic Agents; Imidazoles; MAP Kinase Kinase 1; MAP Kinase Signaling System; Membrane Potential, Mitochondrial; Mice; Mitogen-Activated Protein Kinases; Nitriles; Osteoblasts; PPAR gamma; Pyridines; Reactive Oxygen Species; Thiazolidinediones; Troglitazone | 2007 |
Ciglitazone induces caspase-independent apoptosis via p38-dependent AIF nuclear translocation in renal epithelial cells.
Topics: Active Transport, Cell Nucleus; Animals; Apoptosis; Apoptosis Inducing Factor; Blotting, Western; Cell Line; Cell Nucleus; Cell Survival; Chromans; Clofibric Acid; Dose-Response Relationship, Drug; Epithelial Cells; Fibric Acids; Flow Cytometry; Fluorescent Antibody Technique; G1 Phase; Imidazoles; Kidney Tubules; Membrane Potential, Mitochondrial; Opossums; p38 Mitogen-Activated Protein Kinases; PPAR gamma; Pyridines; Thiazolidinediones; Troglitazone | 2008 |