sb 203580 has been researched along with thiourea in 9 studies
Studies (sb 203580) | Trials (sb 203580) | Recent Studies (post-2010) (sb 203580) | Studies (thiourea) | Trials (thiourea) | Recent Studies (post-2010) (thiourea) |
---|---|---|---|---|---|
3,489 | 4 | 1,137 | 6,959 | 46 | 1,737 |
Protein | Taxonomy | sb 203580 (IC50) | thiourea (IC50) |
---|---|---|---|
Urease | Canavalia ensiformis (jack bean) | 0.56 | |
Serine-protein kinase ATM | Homo sapiens (human) | 0.2 | |
Serine/threonine-protein kinase ATR | Homo sapiens (human) | 0.2 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 5 (55.56) | 29.6817 |
2010's | 4 (44.44) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M | 1 |
Churg, A; Dai, J; Vincent, R; Xie, C | 1 |
Ramesh, G; Reeves, WB | 1 |
Kim, JY; Ro, JY | 1 |
Chen, JD; Gan, HT; Pasricha, PJ | 1 |
Ehrlich, D; Humpel, C; Pirchl, M | 1 |
Chen, F; Chen, R; Chen, Y; Ding, F; Guo, L; Ma, N; Mei, J; Xiao, H; Zhong, H | 1 |
Gao, HW; He, YY; Khan, M; Li, YM; Ma, TH; Yang, JB; Yao, M | 1 |
Deng, WQ; Duan, N; Guo, TT; Huang, LL; Jiang, TT; Liang, XJ; Shu, SS; Tang, X; Wang, Y; Xiang, XH; Zhang, J; Zhu, XL | 1 |
9 other study(ies) available for sb 203580 and thiourea
Article | Year |
---|---|
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases | 2007 |
Air pollution particles produce airway wall remodeling in rat tracheal explants.
Topics: Air Pollution; alpha-Fetoproteins; Animals; Cells, Cultured; Chelating Agents; Collagen; Deferoxamine; DNA, Complementary; Enzyme Inhibitors; Fibrosis; Flavonoids; Gene Expression Regulation; Hydroxyproline; Imidazoles; Iron; Mitogen-Activated Protein Kinases; NF-kappa B; Organ Culture Techniques; Oxidants; p38 Mitogen-Activated Protein Kinases; Peptides; Procollagen; Promoter Regions, Genetic; Pyridines; Rats; Thiourea; Time Factors; Trachea; Transforming Growth Factor beta; Transforming Growth Factor beta1 | 2003 |
p38 MAP kinase inhibition ameliorates cisplatin nephrotoxicity in mice.
Topics: Animals; Cell Line; Cisplatin; Enzyme Activation; Enzyme Inhibitors; Free Radical Scavengers; Imidazoles; Kidney Diseases; Male; Mice; Mice, Inbred C57BL; p38 Mitogen-Activated Protein Kinases; Pyridines; Reactive Oxygen Species; Thiazoles; Thiourea; Tumor Necrosis Factor-alpha | 2005 |
Signal pathway of cytokines produced by reactive oxygen species generated from phorbol myristate acetate-stimulated HMC-1 cells.
Topics: Antioxidants; Free Radical Scavengers; Humans; Imidazoles; Interleukin-8; JNK Mitogen-Activated Protein Kinases; Mast Cells; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Reactive Oxygen Species; RNA, Messenger; Signal Transduction; Tetradecanoylphorbol Acetate; Thiourea; Transcription Factors; Tumor Necrosis Factor-alpha | 2005 |
Blockade of p38 mitogen-activated protein kinase pathway ameliorates delayed intestinal transit in burned rats.
Topics: Animals; Burns; Cyclooxygenase 2 Inhibitors; Disease Models, Animal; Enzyme Inhibitors; Gastrointestinal Transit; Imidazoles; Intestinal Diseases; Male; p38 Mitogen-Activated Protein Kinases; Pyridines; Rats; Rats, Sprague-Dawley; Sulfonamides; Thiourea | 2007 |
Ethanol transiently suppresses choline-acetyltransferase in basal nucleus of Meynert slices.
Topics: Analysis of Variance; Animals; Animals, Newborn; Basal Nucleus of Meynert; Central Nervous System Depressants; Chemokine CXCL2; Choline O-Acetyltransferase; Citrulline; Dose-Response Relationship, Drug; Down-Regulation; Drug Interactions; Enzyme Inhibitors; Ethanol; Imidazoles; In Vitro Techniques; Nerve Growth Factor; Neurons; Pyridines; Rats; Thiourea; Time Factors; Tumor Necrosis Factor-alpha | 2012 |
Phosphorylation of eIF2α suppresses cisplatin-induced A549 cell apoptosis via p38 inhibition.
Topics: Aged; Antineoplastic Agents; Apoptosis; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Cinnamates; Cisplatin; Drug Resistance, Neoplasm; eIF-2 Kinase; Enzyme Activation; Enzyme Inhibitors; Eukaryotic Initiation Factor-2; Female; Humans; Imidazoles; Lung Neoplasms; Male; Middle Aged; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Prognosis; Pyridines; Signal Transduction; Thiourea; Tissue Array Analysis | 2013 |
Tubeimoside-1 induces oxidative stress-mediated apoptosis and G0/G1 phase arrest in human prostate carcinoma cells in vitro.
Topics: Acetylcysteine; Amino Acid Chloromethyl Ketones; Anthracenes; Apoptosis; Caspase 3; Cell Cycle Checkpoints; Cell Line, Tumor; Cell Survival; Cinnamates; Cyclin E; Cyclin-Dependent Kinase 2; Dose-Response Relationship, Drug; Endoplasmic Reticulum Stress; G1 Phase; Humans; Imidazoles; JNK Mitogen-Activated Protein Kinases; Male; MAP Kinase Kinase Kinase 5; Membrane Potential, Mitochondrial; Oxidative Stress; p38 Mitogen-Activated Protein Kinases; Prostatic Neoplasms; Proto-Oncogene Proteins c-bcl-2; Pyridines; Reactive Oxygen Species; Resting Phase, Cell Cycle; Saponins; Thiourea; Triterpenes | 2016 |
[P38 MAPK signaling pathway mediates advanced oxidation protein product-induced epithelial-to-mesenchymal transition in tubular cells].
Topics: Advanced Oxidation Protein Products; Antigens, CD; Cadherins; Cell Line; Cinnamates; Endoplasmic Reticulum Chaperone BiP; Endoplasmic Reticulum Stress; Epithelial-Mesenchymal Transition; Heat-Shock Proteins; Humans; Imidazoles; MAP Kinase Signaling System; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Thiourea; Vimentin | 2016 |