Page last updated: 2024-09-05

sb 203580 and thiazoles

sb 203580 has been researched along with thiazoles in 32 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(thiazoles)
Trials
(thiazoles)
Recent Studies (post-2010) (thiazoles)
3,48941,13733,1792,10012,330

Research

Studies (32)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (3.13)18.2507
2000's21 (65.63)29.6817
2010's9 (28.13)24.3611
2020's1 (3.13)2.80

Authors

AuthorsStudies
Baillargeon, J; Cleland, LG; James, MJ; Lee, JC; Pouliot, M1
de Caestecker, MP; Watanabe, H; Yamada, Y1
Bae, MA; Pie, JE; Song, BJ1
Cara, DC; Forster, M; Kaur, J; Kubes, P; McCafferty, DM1
Cao, BZ; Jing, Q; Lei, ZB; Li, XY; Pei, G; Qin, YW; Zhang, Z1
Eggo, MC; Holder, JC; Kumar, S; Patel, NG; Smith, SA1
Kaur, J; Kubes, P; Woodman, RC1
Blaschke, F; Bruemmer, D; Kintscher, U; Law, RE; Unger, T1
Guinea Viniegra, J; Hernández Losa, J; Parada Cobo, C; Ramón y Cajal, S; Sánchez-Arevalo Lobo, VJ; Sánchez-Prieto, R1
Dai, J; Remick, DG; Wang, X; Zeng, X1
Rao, GN; Yellaturu, CR1
Bukhtiyarova, M; Casper, D; Springman, EB1
Gaestel, M; Hannigan, MO; Huang, CK; Kotlyarov, A; Wu, D; Wu, Y1
Anto, RJ; Karunagaran, D; Maliekal, TT1
Bark, H; Choi, CH; Kim, SH1
Beer, D; Gedeck, P; Howe, T; Keller, TH; Press, NJ; Trifilieff, A; Walker, C1
Ramesh, G; Reeves, WB1
Al-Khalili, L; Ehrenborg, E; Kannisto, K; Krämer, DK; Krook, A; Perrini, S; Skogsberg, J; Wallberg-Henriksson, H; Wretenberg, P; Zierath, JR1
Laufer, S; Wagner, G1
Chen, J; Deng, J; Geng, L; Jiang, G; Qian, Y; Wang, X; Xie, H; Yan, S; Zheng, S; Zhou, L1
Cordova, FM; Costa, AP; Leal, RB; Oliveira, CS; Posser, T; Rigon, AP; Rocha, JB; Rossi, FM; Santos, DA; Silva, IG1
Chae, B; Chung, JE; Hwang, SJ; Jo, HH; Kim, EJ; Kim, JH; Kim, MR; Kim, SY; Kwon, DJ; Lew, YO; Lim, YT1
Ahn, SG; Kim, SA; Kwon, SM; Yoon, JH1
Adachi, M; Fort, P; Okawa, K; Tsukita, S; Uji, M; Yamazaki, Y; Yano, T1
Azevedo, R; de Vlieg, J; Kazemier, B; Oubrie, A; Raaijmakers, H; van Zeeland, M1
Dionyssiou, MG; Hashemi, S; Kerr, A; McDermott, JC; Nowacki, NB; Tsushima, RG; Zhao, J1
Chen, X; Duan, L; He, T; Luo, J; Shi, Q; Tang, M; Wang, H; Weng, Y; Wu, R; Yang, X; Ye, L; Zhang, Y; Zhou, L1
Falck, D; Giera, M; Honing, M; Kool, J; Niessen, WM; Rahimi Pirkolachachi, F1
Bussink, J; Grénman, R; Iida, M; Kaanders, JH; Peeters, WJ; Span, PN; Stegeman, H; van der Kogel, AJ; Verheijen, MM; Wheeler, DL1
Lu, BX; Luo, YF; Man, RY; Wang, XF; Zeng, QG; Zeng, Y1
Hein, TW; Kuo, L; Ren, Y; Thengchaisri, N; Tsai, SH; Xu, W; Xu, X1
Cao, H; Zhang, Y1

Reviews

1 review(s) available for sb 203580 and thiazoles

ArticleYear
Small molecular anti-cytokine agents.
    Medicinal research reviews, 2006, Volume: 26, Issue:1

    Topics: ADAM Proteins; ADAM17 Protein; Animals; Caspase Inhibitors; Cytochrome P-450 Enzyme Inhibitors; Cytokines; Humans; Hydroxamic Acids; Imidazoles; Matrix Metalloproteinase Inhibitors; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Pyridazines; Pyridines; Pyrimidines; Quinazolines; Structure-Activity Relationship; Succinates; Thiazoles; Tumor Necrosis Factor-alpha; Urea

2006

Other Studies

31 other study(ies) available for sb 203580 and thiazoles

ArticleYear
Inhibition of prostaglandin endoperoxide synthase-2 expression in stimulated human monocytes by inhibitors of p38 mitogen-activated protein kinase.
    Journal of immunology (Baltimore, Md. : 1950), 1997, May-15, Volume: 158, Issue:10

    Topics: Arachidonate 5-Lipoxygenase; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Humans; Imidazoles; Interleukin-1; Mitogen-Activated Protein Kinases; Monocytes; p38 Mitogen-Activated Protein Kinases; Phospholipases A; Phospholipases A2; Pyridines; RNA, Messenger; Thiazoles

1997
Transcriptional cross-talk between Smad, ERK1/2, and p38 mitogen-activated protein kinase pathways regulates transforming growth factor-beta-induced aggrecan gene expression in chondrogenic ATDC5 cells.
    The Journal of biological chemistry, 2001, Apr-27, Volume: 276, Issue:17

    Topics: Aggrecans; Animals; Butadienes; Cell Differentiation; Cell Line; Cell Nucleus; Chondrocytes; Cycloheximide; DNA-Binding Proteins; Dose-Response Relationship, Drug; Enzyme Activation; Extracellular Matrix Proteins; Gene Expression Regulation, Enzymologic; Genes, Dominant; Imidazoles; Immunoblotting; Lectins, C-Type; Luciferases; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Synthesis Inhibitors; Proteoglycans; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Smad Proteins; Thiazoles; Time Factors; Trans-Activators; Transcription, Genetic; Transfection; Transforming Growth Factor beta

2001
Acetaminophen induces apoptosis of C6 glioma cells by activating the c-Jun NH(2)-terminal protein kinase-related cell death pathway.
    Molecular pharmacology, 2001, Volume: 60, Issue:4

    Topics: Acetaminophen; Acetanilides; Analgesics; Analgesics, Non-Narcotic; Androstadienes; Animals; Apoptosis; bcl-2-Associated X Protein; Caspase 3; Caspases; Cytochrome c Group; Cytochrome P-450 CYP2E1; DNA Fragmentation; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Glioma; Imidazoles; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-bcl-2; Pyridines; Rats; Thiazoles; Time Factors; Tumor Cells, Cultured; Wortmannin

2001
Role of p38 mitogen-activated protein kinase in chemokine-induced emigration and chemotaxis in vivo.
    Journal of immunology (Baltimore, Md. : 1950), 2001, Dec-01, Volume: 167, Issue:11

    Topics: Animals; Cell Adhesion; Chemokine CXCL1; Chemokines; Chemokines, CXC; Chemotaxis, Leukocyte; Cytokines; Enzyme Inhibitors; Imidazoles; Infusions, Intravenous; Injections, Intravenous; Keratinocytes; Male; Mice; Mice, Inbred C57BL; Microscopy, Video; Mitogen-Activated Protein Kinases; Muscle, Skeletal; Neutrophil Infiltration; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Thiazoles

2001
OxLDL upregulates CXCR2 expression in monocytes via scavenger receptors and activation of p38 mitogen-activated protein kinase.
    Cardiovascular research, 2002, Feb-01, Volume: 53, Issue:2

    Topics: Cell Adhesion; Chemotaxis, Leukocyte; Coculture Techniques; Dextran Sulfate; Endothelium, Vascular; Enzyme Activation; Flow Cytometry; Humans; Imidazoles; Interleukin-8; Lipoproteins, LDL; Membrane Proteins; Mitogen-Activated Protein Kinases; Monocytes; p38 Mitogen-Activated Protein Kinases; Poly I; Pyridines; Receptors, Immunologic; Receptors, Interleukin-8B; Receptors, Lipoprotein; Receptors, Scavenger; RNA, Messenger; Scavenger Receptors, Class B; Thiazoles; U937 Cells

2002
Differential regulation of lipogenesis and leptin production by independent signaling pathways and rosiglitazone during human adipocyte differentiation.
    Diabetes, 2003, Volume: 52, Issue:1

    Topics: Adipocytes; Androstadienes; Cell Differentiation; Cell Survival; Cells, Cultured; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Leptin; Lipid Metabolism; Lipids; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Pyridines; Rosiglitazone; Signal Transduction; Sirolimus; Stem Cells; Thiazoles; Thiazolidinediones; Tumor Necrosis Factor-alpha; Wortmannin

2003
P38 MAPK: critical molecule in thrombin-induced NF-kappa B-dependent leukocyte recruitment.
    American journal of physiology. Heart and circulatory physiology, 2003, Volume: 284, Issue:4

    Topics: Adenosine Triphosphate; Binding Sites; Binding, Competitive; Cell Adhesion; Cells, Cultured; E-Selectin; Endothelium, Vascular; Enzyme Activation; Enzyme Inhibitors; Humans; Imidazoles; Leukocytes; Mitogen-Activated Protein Kinases; NF-kappa B; P-Selectin; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Thiazoles; Thrombin; Umbilical Veins

2003
p38 MAP kinase negatively regulates angiotensin II-mediated effects on cell cycle molecules in human coronary smooth muscle cells.
    Biochemical and biophysical research communications, 2003, Jun-06, Volume: 305, Issue:3

    Topics: Angiotensin II; Cell Cycle; Cells, Cultured; Cyclin D1; DNA; Enzyme Inhibitors; Humans; Imidazoles; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Myocardium; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Retinoblastoma Protein; Thiazoles

2003
Role of the p38 MAPK pathway in cisplatin-based therapy.
    Oncogene, 2003, Jun-26, Volume: 22, Issue:26

    Topics: Animals; Antineoplastic Agents; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cell Survival; Cisplatin; COS Cells; Cross-Linking Reagents; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Resistance, Neoplasm; Enzyme Activation; Enzyme Inhibitors; HeLa Cells; Humans; Imidazoles; Kinetics; MAP Kinase Kinase 3; MAP Kinase Kinase 6; Mitogen-Activated Protein Kinase 12; Mitogen-Activated Protein Kinase 13; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phenotype; Phosphorylation; Plasmids; Platinum Compounds; Precipitin Tests; Protein Isoforms; Protein-Tyrosine Kinases; Pyridines; Signal Transduction; Thiazoles; Transfection; Tumor Cells, Cultured

2003
Homocysteine mediated expression and secretion of monocyte chemoattractant protein-1 and interleukin-8 in human monocytes.
    Circulation research, 2003, Aug-22, Volume: 93, Issue:4

    Topics: Antioxidants; Cells, Cultured; Chemokine CCL2; Chromans; Dimethyl Sulfoxide; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Genistein; Homocysteine; Humans; Imidazoles; Indoles; Interleukin-8; Monocytes; Naphthalenes; Onium Compounds; Pyridines; Pyrrolidines; Reactive Oxygen Species; RNA, Messenger; Sulfonamides; Thiazoles; Thiazolidinediones; Thiocarbamates; Time Factors; Troglitazone; Tyrphostins

2003
A requirement for calcium-independent phospholipase A2 in thrombin-induced arachidonic acid release and growth in vascular smooth muscle cells.
    The Journal of biological chemistry, 2003, Oct-31, Volume: 278, Issue:44

    Topics: Animals; Arachidonic Acid; Blotting, Western; Coloring Agents; DNA; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Inhibitors; Group VI Phospholipases A2; Imidazoles; Male; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Naphthalenes; Oleic Acid; Oligonucleotides, Antisense; p38 Mitogen-Activated Protein Kinases; Phospholipases A; Phospholipases A2; Pyridines; Pyrones; Rats; Rats, Sprague-Dawley; Signal Transduction; Tetrazolium Salts; Thiazoles; Thrombin; Time Factors

2003
A Biacore biosensor method for detailed kinetic binding analysis of small molecule inhibitors of p38alpha mitogen-activated protein kinase.
    Analytical biochemistry, 2004, Feb-01, Volume: 325, Issue:1

    Topics: Animals; Escherichia coli; Imidazoles; Kinetics; Mice; Mitogen-Activated Protein Kinases; Molecular Structure; Phosphorylation; Protein Binding; Protein Denaturation; Pyridines; Recombinant Proteins; Surface Plasmon Resonance; Thiazoles

2004
A requirement of MAPKAPK2 in the uropod localization of PTEN during FMLP-induced neutrophil chemotaxis.
    Biochemical and biophysical research communications, 2004, Apr-09, Volume: 316, Issue:3

    Topics: Actins; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cell Movement; Cell Surface Extensions; Chemotaxis; Enzyme Inhibitors; Imidazoles; Immunoblotting; Intracellular Signaling Peptides and Proteins; Lipid Metabolism; Mice; Mice, Inbred C57BL; Microscopy, Confocal; Microscopy, Fluorescence; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Phosphatidylinositol 3-Kinases; Phosphatidylinositol Phosphates; Phosphoric Monoester Hydrolases; Phosphorylation; Protein Serine-Threonine Kinases; PTEN Phosphohydrolase; Pyridines; Thiazoles; Thiazolidines; Time Factors; Tumor Suppressor Proteins

2004
Differential activation of Smads in HeLa and SiHa cells that differ in their response to transforming growth factor-beta.
    The Journal of biological chemistry, 2004, Aug-27, Volume: 279, Issue:35

    Topics: Blotting, Western; Cell Cycle; Cell Division; Cell Line, Tumor; Cell Nucleus; Cell Survival; Coloring Agents; DNA; Enzyme Inhibitors; G1 Phase; Genes, Reporter; HeLa Cells; Humans; Imidazoles; JNK Mitogen-Activated Protein Kinases; Luciferases; MAP Kinase Kinase 4; MAP Kinase Signaling System; Microscopy, Fluorescence; Mitogen-Activated Protein Kinase Kinases; Protein Binding; Pyridines; Resting Phase, Cell Cycle; S Phase; Tetrazolium Salts; Thiazoles; Time Factors; Transcription Factor AP-1; Transforming Growth Factor beta

2004
Mercury induces multidrug resistance-associated protein gene through p38 mitogen-activated protein kinase.
    Toxicology letters, 2005, Jan-15, Volume: 155, Issue:1

    Topics: Blotting, Western; Cell Division; Cell Line; Cell Line, Tumor; Cell Survival; Chemokines, CC; Enzyme Inhibitors; Fluorescent Antibody Technique; Humans; Imidazoles; Mercury; p38 Mitogen-Activated Protein Kinases; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA; Tetrazolium Salts; Thiazoles

2005
CGH2466, a combined adenosine receptor antagonist, p38 mitogen-activated protein kinase and phosphodiesterase type 4 inhibitor with potent in vitro and in vivo anti-inflammatory activities.
    British journal of pharmacology, 2005, Volume: 144, Issue:7

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cricetinae; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Dose-Response Relationship, Drug; Female; Humans; Imidazoles; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; p38 Mitogen-Activated Protein Kinases; Phosphodiesterase Inhibitors; Protein Kinase Inhibitors; Purinergic P1 Receptor Antagonists; Pyridines; Receptors, Purinergic P1; Thiazoles

2005
p38 MAP kinase inhibition ameliorates cisplatin nephrotoxicity in mice.
    American journal of physiology. Renal physiology, 2005, Volume: 289, Issue:1

    Topics: Animals; Cell Line; Cisplatin; Enzyme Activation; Enzyme Inhibitors; Free Radical Scavengers; Imidazoles; Kidney Diseases; Male; Mice; Mice, Inbred C57BL; p38 Mitogen-Activated Protein Kinases; Pyridines; Reactive Oxygen Species; Thiazoles; Thiourea; Tumor Necrosis Factor-alpha

2005
Direct activation of glucose transport in primary human myotubes after activation of peroxisome proliferator-activated receptor delta.
    Diabetes, 2005, Volume: 54, Issue:4

    Topics: Adipocytes; Animals; Biological Transport; Cell Line; Cells, Cultured; Fibroblasts; Flavonoids; Gene Expression Regulation; Glucose; Humans; Imidazoles; MAP Kinase Kinase Kinases; Muscle Fibers, Skeletal; Muscle, Skeletal; p38 Mitogen-Activated Protein Kinases; PPAR delta; Pyridines; Thiazoles

2005
Involvement of p38 mitogen-activated protein kinase pathway in honokiol-induced apoptosis in a human hepatoma cell line (hepG2).
    Liver international : official journal of the International Association for the Study of the Liver, 2008, Volume: 28, Issue:10

    Topics: Apoptosis; Biphenyl Compounds; Blotting, Western; Carcinoma, Hepatocellular; Caspases; Cell Line, Tumor; Cell Proliferation; Flow Cytometry; Humans; Imidazoles; Lignans; p38 Mitogen-Activated Protein Kinases; Pyridines; Signal Transduction; Tetrazolium Salts; Thiazoles

2008
Neurotoxicity of cadmium on immature hippocampus and a neuroprotective role for p38 MAPK.
    Neurotoxicology, 2008, Volume: 29, Issue:4

    Topics: Animals; Animals, Newborn; Cadmium; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Flavonoids; Hippocampus; Imidazoles; In Vitro Techniques; Male; Neurotoxins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Rats; Rats, Wistar; Signal Transduction; Tetrazolium Salts; Thiazoles

2008
Antioxidant effects of equol on bovine aortic endothelial cells.
    Biochemical and biophysical research communications, 2008, Oct-24, Volume: 375, Issue:3

    Topics: Animals; Antioxidants; Aorta; Apoptosis; Cattle; Cytoprotection; Endothelium, Vascular; Equol; Hydrogen Peroxide; Imidazoles; Isoflavones; p38 Mitogen-Activated Protein Kinases; Phytoestrogens; Proto-Oncogene Proteins c-bcl-2; Pyridines; Reactive Oxygen Species; Tetrazolium Salts; Thiazoles

2008
Transforming growth factor beta1-induced heat shock protein 27 activation promotes migration of mouse dental papilla-derived MDPC-23 cells.
    Journal of endodontics, 2010, Volume: 36, Issue:8

    Topics: Animals; Blotting, Western; Cell Count; Cell Line; Cell Movement; Cell Proliferation; Chemotaxis; Coloring Agents; Dental Papilla; Enzyme Inhibitors; HSP27 Heat-Shock Proteins; Imidazoles; Mice; NF-kappa B; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Proto-Oncogene Proteins c-akt; Pyridines; Signal Transduction; Tetrazolium Salts; Thiazoles; Transforming Growth Factor beta1

2010
Tara up-regulates E-cadherin transcription by binding to the Trio RhoGEF and inhibiting Rac signaling.
    The Journal of cell biology, 2011, Apr-18, Volume: 193, Issue:2

    Topics: Adherens Junctions; Animals; Benzimidazoles; Cadherins; Cell Line; Dogs; Epithelial-Mesenchymal Transition; Guanine Nucleotide Exchange Factors; Humans; Imidazoles; Mice; Microfilament Proteins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; rac1 GTP-Binding Protein; Rho Guanine Nucleotide Exchange Factors; Signal Transduction; T-Box Domain Proteins; Thiazoles; Transcription, Genetic; Up-Regulation

2011
X-ray structure of p38α bound to TAK-715: comparison with three classic inhibitors.
    Acta crystallographica. Section D, Biological crystallography, 2012, Volume: 68, Issue:Pt 8

    Topics: Adenosine Triphosphate; Benzamides; Catalytic Domain; Cloning, Molecular; Crystallization; Crystallography, X-Ray; Humans; Imidazoles; Indoles; Ligands; p38 Mitogen-Activated Protein Kinases; Protein Binding; Protein Conformation; Protein Kinase Inhibitors; Pyridazines; Pyridines; Pyrimidines; Structure-Activity Relationship; Thiazoles

2012
Cross-talk between glycogen synthase kinase 3β (GSK3β) and p38MAPK regulates myocyte enhancer factor 2 (MEF2) activity in skeletal and cardiac muscle.
    Journal of molecular and cellular cardiology, 2013, Volume: 54

    Topics: Animals; Cell Line; Enhancer Elements, Genetic; Female; Gene Expression Regulation; Genes, Reporter; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Imidazoles; Luciferases; Male; MEF2 Transcription Factors; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle, Skeletal; Myoblasts; Myoblasts, Skeletal; Myocardium; Myocytes, Cardiac; Myogenic Regulatory Factors; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Primary Cell Culture; Protein Processing, Post-Translational; Pyridines; Signal Transduction; Thiazoles; Transcriptional Activation; Urea

2013
S100A9 promotes the proliferation and invasion of HepG2 hepatocellular carcinoma cells via the activation of the MAPK signaling pathway.
    International journal of oncology, 2013, Volume: 42, Issue:3

    Topics: Animals; Calgranulin B; Carcinoma, Hepatocellular; Cell Line, Tumor; Cell Proliferation; Cell Transformation, Neoplastic; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Female; Flavonoids; Hep G2 Cells; Humans; Imidazoles; Liver Neoplasms; MAP Kinase Signaling System; Mice; Mice, Nude; Mitogen-Activated Protein Kinases; Neoplasm Invasiveness; Neoplasm Transplantation; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Random Allocation; Tetrazolium Salts; Thiazoles; Xenograft Model Antitumor Assays

2013
Comparison of (bio-)transformation methods for the generation of metabolite-like compound libraries of p38α MAP kinase inhibitors using high-resolution screening.
    Journal of pharmaceutical and biomedical analysis, 2014, Volume: 88

    Topics: Bacillus megaterium; Benzamides; Chemistry, Pharmaceutical; Cytochrome P-450 Enzyme System; High-Throughput Screening Assays; Humans; Hydrogen Peroxide; Imidazoles; Indoles; Light; Liver; Microsomes, Liver; Mitogen-Activated Protein Kinase 14; Naphthalenes; Oxygen; Photochemistry; Piperazines; Protein Kinase Inhibitors; Pyrazoles; Pyridines; Recombinant Proteins; Structure-Activity Relationship; Thiazoles

2014
Combining radiotherapy with MEK1/2, STAT5 or STAT6 inhibition reduces survival of head and neck cancer lines.
    Molecular cancer, 2013, Nov-05, Volume: 12, Issue:1

    Topics: Antineoplastic Agents; Butadienes; Carcinoma, Squamous Cell; Cell Line, Tumor; Cell Survival; Chemoradiotherapy; Dasatinib; Drug Screening Assays, Antitumor; Head and Neck Neoplasms; Humans; Imidazoles; Isoxazoles; Leflunomide; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Nitriles; Protein Kinase Inhibitors; Pyridines; Pyrimidines; Radiation Tolerance; STAT5 Transcription Factor; STAT6 Transcription Factor; Thiazoles; Tumor Suppressor Proteins

2013
Induction of GADD45α protects M17 neuroblastoma cells against MPP*.
    IUBMB life, 2014, Volume: 66, Issue:11

    Topics: 1-Methyl-4-phenylpyridinium; Analysis of Variance; Anthracenes; Blotting, Western; Caspase 3; Cell Cycle Proteins; Cell Line, Tumor; Cell Survival; Chromatin Immunoprecipitation; Dose-Response Relationship, Drug; Gene Expression Regulation; Humans; Imidazoles; In Situ Nick-End Labeling; Nuclear Proteins; Parkinson Disease; Pyridines; Real-Time Polymerase Chain Reaction; RNA Interference; Tetrazolium Salts; Thiazoles

2014
Requisite roles of LOX-1, JNK, and arginase in diabetes-induced endothelial vasodilator dysfunction of porcine coronary arterioles.
    Journal of molecular and cellular cardiology, 2019, Volume: 131

    Topics: Animals; Anthracenes; Arginase; Arterioles; Coronary Vessels; Cyclic N-Oxides; Diabetes Mellitus, Experimental; Dioxanes; Imidazoles; In Vitro Techniques; JNK Mitogen-Activated Protein Kinases; Male; Nitric Oxide; Pyridines; Scavenger Receptors, Class E; Serotonin; Spin Labels; Swine; Thiazoles; Vasodilation

2019
Monomeric C-reactive protein affects cell injury and apoptosis through activation of p38 mitogen-activated protein kinase in human coronary artery endothelial cells.
    Bosnian journal of basic medical sciences, 2020, Nov-02, Volume: 20, Issue:4

    Topics: Antigens, CD; Apoptosis; Atherosclerosis; C-Reactive Protein; Cell Adhesion; Cell Adhesion Molecules; Cell Proliferation; Cells, Cultured; Coronary Vessels; Cyclooxygenase 2; Endothelial Cells; Humans; Imidazoles; Inflammation; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; RNA, Small Interfering; Tetrazolium Salts; Thiazoles; Time Factors; Vascular Endothelial Growth Factor A

2020