Page last updated: 2024-09-05

sb 203580 and thapsigargin

sb 203580 has been researched along with thapsigargin in 8 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(thapsigargin)
Trials
(thapsigargin)
Recent Studies (post-2010) (thapsigargin)
3,48941,1375,2343918

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)thapsigargin (IC50)
Sarcoplasmic/endoplasmic reticulum calcium ATPase 1Oryctolagus cuniculus (rabbit)0.002

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (87.50)29.6817
2010's1 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hirasawa, N; Kobayashi, Y; Murakami, A; Ohuchi, K; Oikawa, S; Shiraishi, M1
Kozawa, O; Tokuda, H; Uematsu, T1
Chen, Q; Donahue, HJ; Jacobs, CR; Reilly, GC; Yellowley, CE; You, J; Zhen, X1
Hirasawa, N; Murakami, A; Ohuchi, K1
Chen, BC; Lin, WW1
Klemm, J; Rådmark, O; Samuelsson, B; Werz, O1
Hori, M; Karaki, H; Ozaki, H; Tasaki, K; Wakabayashi, I1
Chae, HJ; Chae, SW; Kim, DS; Kim, HR; Kim, HT; Kim, JH; Lee, GH; Lim, JM1

Other Studies

8 other study(ies) available for sb 203580 and thapsigargin

ArticleYear
Participation of mitogen-activated protein kinase in thapsigargin- and TPA-induced histamine production in murine macrophage RAW 264.7 cells.
    British journal of pharmacology, 2000, Volume: 129, Issue:3

    Topics: Animals; Blotting, Western; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Enzyme Inhibitors; Flavonoids; Histamine Release; Imidazoles; Macrophages; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetradecanoylphorbol Acetate; Thapsigargin

2000
Basic fibroblast growth factor stimulates vascular endothelial growth factor release in osteoblasts: divergent regulation by p42/p44 mitogen-activated protein kinase and p38 mitogen-activated protein kinase.
    Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 2000, Volume: 15, Issue:12

    Topics: Animals; Calcimycin; Calcium; Endothelial Growth Factors; Enzyme Inhibitors; Fibroblast Growth Factor 2; Flavonoids; Imidazoles; In Vitro Techniques; Ionophores; Lymphokines; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Thapsigargin; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2000
Osteopontin gene regulation by oscillatory fluid flow via intracellular calcium mobilization and activation of mitogen-activated protein kinase in MC3T3-E1 osteoblasts.
    The Journal of biological chemistry, 2001, Apr-20, Volume: 276, Issue:16

    Topics: 3T3 Cells; Animals; Calcium Channel Blockers; Calcium Signaling; Enzyme Inhibitors; Gadolinium; Gene Expression Regulation; Imidazoles; Intracellular Fluid; JNK Mitogen-Activated Protein Kinases; Kinetics; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinases; Models, Biological; Oscillometry; Osteoblasts; Osteopontin; p38 Mitogen-Activated Protein Kinases; Pyridines; RNA, Messenger; Sialoglycoproteins; Stress, Mechanical; Thapsigargin; Transcription, Genetic

2001
Expression of 74-kDa histidine decarboxylase protein in a macrophage-like cell line RAW 264.7 and inhibition by dexamethasone.
    European journal of pharmacology, 2001, Apr-20, Volume: 418, Issue:1-2

    Topics: Animals; Catalysis; Cell Line; Dexamethasone; Enzyme Activation; Enzyme Induction; Flavonoids; Histamine; Histidine Decarboxylase; Imidazoles; Immunoblotting; Macrophages; Mice; Mitogen-Activated Protein Kinases; Pyridines; Thapsigargin

2001
PKC- and ERK-dependent activation of I kappa B kinase by lipopolysaccharide in macrophages: enhancement by P2Y receptor-mediated CaMK activation.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: Animals; Benzylamines; Bridged-Ring Compounds; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Enzyme Activation; Enzyme Inhibitors; Flavonoids; I-kappa B Kinase; I-kappa B Proteins; Imidazoles; Indoles; Lipopolysaccharides; Macrophages; Macrophages, Peritoneal; Mitogen-Activated Protein Kinases; NF-kappa B; Norbornanes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; Receptors, Purinergic P2; Sulfonamides; Thapsigargin; Thiocarbamates; Thiones; Time Factors; Transcription Factor RelA; Uridine Triphosphate

2001
p38 MAP kinase mediates stress-induced leukotriene synthesis in a human B-lymphocyte cell line.
    Journal of leukocyte biology, 2001, Volume: 70, Issue:5

    Topics: Arachidonate 5-Lipoxygenase; Arachidonic Acid; Arsenites; B-Lymphocytes; Calcimycin; Calcium; Cell Line; Cell-Free System; Enzyme Activation; Enzyme Inhibitors; Hydroxyeicosatetraenoic Acids; Hypertonic Solutions; Imidazoles; Interleukin-1; Intracellular Signaling Peptides and Proteins; Ionophores; Leukotrienes; Lipoxygenase Inhibitors; Mitogen-Activated Protein Kinases; Osmotic Pressure; Oxidative Stress; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinases; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Protein Tyrosine Phosphatases; Pyridines; Sodium Compounds; Sorbitol; Subcellular Fractions; Thapsigargin; Transforming Growth Factor beta; Tumor Necrosis Factor-alpha; Vanadates

2001
Mechanism of human urotensin II-induced contraction in rat aorta.
    Journal of pharmacological sciences, 2004, Volume: 94, Issue:4

    Topics: Androstadienes; Animals; Aorta, Thoracic; Butadienes; Calcium; Carbazoles; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Humans; Imidazoles; Indoles; Lanthanum; Male; Maleimides; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Muscle Contraction; Myosin Light Chains; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Potassium Chloride; Protein Kinase C; Pyridines; Rats; Rats, Wistar; Thapsigargin; Urotensins; Verapamil; Wortmannin

2004
p38 Mitogen-activated protein kinase is involved in endoplasmic reticulum stress-induced cell death and autophagy in human gingival fibroblasts.
    Biological & pharmaceutical bulletin, 2010, Volume: 33, Issue:4

    Topics: Autophagy; Brefeldin A; Cell Death; Endoplasmic Reticulum; Endoplasmic Reticulum Chaperone BiP; Enzyme Inhibitors; Fibroblasts; Gingiva; Heat-Shock Proteins; Humans; Imidazoles; Microtubule-Associated Proteins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Synthesis Inhibitors; Pyridines; Thapsigargin; Transcription Factor CHOP; Tunicamycin

2010