Page last updated: 2024-09-05

sb 203580 and tetrodotoxin

sb 203580 has been researched along with tetrodotoxin in 5 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(tetrodotoxin)
Trials
(tetrodotoxin)
Recent Studies (post-2010) (tetrodotoxin)
3,48941,13712,992111,477

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)tetrodotoxin (IC50)
Sodium channel protein type 9 subunit alphaHomo sapiens (human)0.0186

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Choe, ES; McGinty, JF1
Dib-Hajj, SD; Hudmon, A; Rush, AM; Waxman, SG; Wittmack, EK1
Kwan, YW; Ngai, SM; Seto, SW1
Amaya, F; Bean, BP; Binshtok, AM; Brenner, GJ; Ji, RR; Samad, TA; Shi, L; Vardeh, D; Wang, H; Woolf, CJ; Zimmermann, K1
Kanai, T; Maruta, T; Miyazaki, S; Nemoto, T; Satoh, S; Wada, A; Yanagita, T; Yoshikawa, N1

Other Studies

5 other study(ies) available for sb 203580 and tetrodotoxin

ArticleYear
N-Methyl-D-aspartate receptors and p38 mitogen-activated protein kinase are required for cAMP-dependent cyclase response element binding protein and Elk-1 phosphorylation in the striatum.
    Neuroscience, 2000, Volume: 101, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cyclic AMP Response Element-Binding Protein; Dizocilpine Maleate; DNA-Binding Proteins; Enzyme Inhibitors; ets-Domain Protein Elk-1; Flavonoids; Imidazoles; Male; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Neostriatum; Neurons; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-fos; Pyridines; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Sodium Channels; Tetrodotoxin; Thionucleotides; Transcription Factors

2000
Voltage-gated sodium channel Nav1.6 is modulated by p38 mitogen-activated protein kinase.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jul-13, Volume: 25, Issue:28

    Topics: Amino Acid Substitution; Animals; Anisomycin; Brain Chemistry; Cell Line; Enzyme Activation; Humans; Imidazoles; Ion Transport; Kidney; Male; Mice; Mutagenesis, Site-Directed; NAV1.6 Voltage-Gated Sodium Channel; Nerve Tissue Proteins; Neurons; p38 Mitogen-Activated Protein Kinases; Patch-Clamp Techniques; Phosphorylation; Phosphoserine; Protein Interaction Mapping; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Purkinje Cells; Pyridines; Rats; Rats, Sprague-Dawley; Recombinant Fusion Proteins; Sodium; Sodium Channels; Tetrodotoxin; Transfection

2005
Modulatory effect of interleukin-1beta on rat isolated basilar artery contraction.
    European journal of pharmacology, 2006, Feb-15, Volume: 531, Issue:1-3

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Antagonists; Animals; Basilar Artery; Calcium-Calmodulin-Dependent Protein Kinases; Cyclohexenes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Imidazoles; In Vitro Techniques; Interleukin-1; Male; Monoterpenes; Phenylephrine; Prazosin; Protoporphyrins; Pyridines; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Vasoconstriction; Vasoconstrictor Agents

2006
Nociceptors are interleukin-1beta sensors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Dec-24, Volume: 28, Issue:52

    Topics: Action Potentials; Animals; Biophysics; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ganglia, Spinal; Imidazoles; Interleukin-1beta; Intermediate Filament Proteins; Male; Membrane Glycoproteins; Nerve Fibers, Unmyelinated; Nerve Tissue Proteins; Nociceptors; p38 Mitogen-Activated Protein Kinases; Patch-Clamp Techniques; Peripherins; Physical Stimulation; Pyridines; Rats; Rats, Sprague-Dawley; Sensory Receptor Cells; Sodium Channel Blockers; Tetrodotoxin; Time Factors

2008
Nav1.7-Ca2+ influx-induced increased phosphorylations of extracellular signal-regulated kinase (ERK) and p38 attenuate tau phosphorylation via glycogen synthase kinase-3beta: priming of Nav1.7 gating by ERK and p38.
    European journal of pharmacology, 2010, Aug-25, Volume: 640, Issue:1-3

    Topics: Animals; Calcium; Carbazoles; Cattle; Dose-Response Relationship, Drug; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Growth Cones; Humans; Imidazoles; Ion Channel Gating; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Nicotine; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C-alpha; Pyridines; Receptors, Nicotinic; Sodium Channels; tau Proteins; Tetrodotoxin; Time Factors; Veratridine

2010