Page last updated: 2024-09-05

sb 203580 and tacrolimus

sb 203580 has been researched along with tacrolimus in 5 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(tacrolimus)
Trials
(tacrolimus)
Recent Studies (post-2010) (tacrolimus)
3,48941,13717,7572,3196,661

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)tacrolimus (IC50)
Bile salt export pumpHomo sapiens (human)7.18
Cytochrome P450 3A4Homo sapiens (human)0.58
Cytochrome P450 3A5Homo sapiens (human)0.385
Serine/threonine-protein kinase mTORHomo sapiens (human)0.0021
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)0.2547
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoformHomo sapiens (human)0.0148
Splicing factor 3B subunit 3Homo sapiens (human)0.0123
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)3.3
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)3.7

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andreka, P; Bishopric, NH; Evans, WH; Haywood, GA; Martin, PE; Turner, MS; Webster, KA; You, L1
Casella, GT; Godfrey, S; Grumbles, RM; Rudinsky, MJ; Thomas, CK; Wood, PM1
Aam, BB; Fonnum, F1
Aarnes, H; Fonnum, F; Mariussen, E; Myhre, O; Reistad, T; Voie, OA1
Berntsen, HF; Bogen, IL; Fonnum, F; Moldes-Anaya, A; Walaas, SI; Wigestrand, MB1

Other Studies

5 other study(ies) available for sb 203580 and tacrolimus

ArticleYear
Reversible connexin 43 dephosphorylation during hypoxia and reoxygenation is linked to cellular ATP levels.
    Circulation research, 2004, Oct-01, Volume: 95, Issue:7

    Topics: Adenosine Triphosphate; Alkaloids; Aminoimidazole Carboxamide; Animals; Antimycin A; Benzophenanthridines; Brefeldin A; Carbazoles; Cell Hypoxia; Cells, Cultured; Connexin 43; Cycloheximide; Deoxyglucose; Flavonoids; Imidazoles; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; Myocardial Contraction; Myocytes, Cardiac; Okadaic Acid; Ouabain; Phenanthridines; Phosphorylation; Potassium Cyanide; Protein Processing, Post-Translational; Pyridines; Pyrroles; Rats; Recombinant Fusion Proteins; Ribonucleotides; Staurosporine; Tacrolimus; Tetradecanoylphorbol Acetate

2004
The immunophilin ligand FK506, but not the P38 kinase inhibitor SB203580, improves function of adult rat muscle reinnervated from transplants of embryonic neurons.
    Neuroscience, 2005, Volume: 130, Issue:3

    Topics: Animals; Axons; Cell Count; Cell Survival; Electromyography; Electrophysiology; Enzyme Inhibitors; Female; Hindlimb; Imidazoles; Immunophilins; Immunosuppressive Agents; Muscle Denervation; Muscle Fibers, Skeletal; Muscle, Skeletal; Myelin Sheath; Neuromuscular Junction; Neurons; p38 Mitogen-Activated Protein Kinases; Pyridines; Rats; Rats, Inbred F344; Sciatic Nerve; Stem Cell Transplantation; Tacrolimus

2005
Carbon black particles increase reactive oxygen species formation in rat alveolar macrophages in vitro.
    Archives of toxicology, 2007, Volume: 81, Issue:6

    Topics: Animals; Butadienes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Macrophages, Alveolar; Male; MAP Kinase Kinase 5; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 7; NADPH Oxidases; Nitriles; Onium Compounds; p38 Mitogen-Activated Protein Kinases; Particulate Matter; Pyridines; Rats; Rats, Inbred WKY; Reactive Oxygen Species; Soot; Tacrolimus

2007
Effects of polychlorinated biphenyls on the neutrophil NADPH oxidase system.
    Toxicology letters, 2009, Jun-22, Volume: 187, Issue:3

    Topics: Anthracenes; Aroclors; Butadienes; Cyclosporine; Environmental Pollutants; Enzyme Activation; Enzyme Inhibitors; Humans; Imidazoles; Luminescent Measurements; NADPH Oxidases; Neutrophil Activation; Neutrophils; Nitriles; Pyridines; Respiratory Burst; Tacrolimus

2009
The fungal neurotoxin penitrem A induces the production of reactive oxygen species in human neutrophils at submicromolar concentrations.
    Toxicology, 2017, 12-01, Volume: 392

    Topics: Anthracenes; Antioxidants; Calcineurin; Cell Line; Cyclosporine; Granulocytes; Humans; Imidazoles; Inhibitory Concentration 50; JNK Mitogen-Activated Protein Kinases; Mycotoxins; Neurotoxins; Neutrophils; p38 Mitogen-Activated Protein Kinases; Pyridines; Reactive Oxygen Species; Tacrolimus; Vitamin E

2017