Page last updated: 2024-09-05

sb 203580 and suramin

sb 203580 has been researched along with suramin in 5 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(suramin)
Trials
(suramin)
Recent Studies (post-2010) (suramin)
3,48941,1373,02392431

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)suramin (IC50)
ATP-dependent 6-phosphofructokinaseTrypanosoma brucei brucei3
Tyrosine-protein phosphatase non-receptor type 1Homo sapiens (human)9.76
P2X purinoceptor 2Rattus norvegicus (Norway rat)4
DNA-dependent protein kinase catalytic subunitHomo sapiens (human)1.7
DNA primaseMycobacterium tuberculosis CDC15518.2
RmtAAspergillus nidulans5.9
Reverse transcriptase/RNaseH Human immunodeficiency virus 19.4
NAD-dependent protein deacetylase sirtuin-2Homo sapiens (human)1.15
NAD-dependent protein deacetylase sirtuin-1Homo sapiens (human)1.5667
Protein arginine N-methyltransferase 1Homo sapiens (human)5.33
NAD-dependent protein deacylase sirtuin-5, mitochondrialHomo sapiens (human)2.5

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (20.00)18.2507
2000's4 (80.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
McGovern, SL; Shoichet, BK1
Jaakkola, P; Jalkanen, M; Kauppi, T; Kontusaari, S; Määtä, A1
Huwiler, A; Pfeilschifter, J; van den Bosch, H; Wartmann, M1
Kandolf, R; Küpper, JH; Meyer, RG; Rodemann, HP1
Fang, W; He, C; Heng, W; Li, H; Wu, B; You, J; Zheng, J1

Other Studies

5 other study(ies) available for sb 203580 and suramin

ArticleYear
Kinase inhibitors: not just for kinases anymore.
    Journal of medicinal chemistry, 2003, Apr-10, Volume: 46, Issue:8

    Topics: beta-Lactamase Inhibitors; beta-Lactamases; Chymotrypsin; Enzyme Inhibitors; Kinetics; Light; Malate Dehydrogenase; Models, Biological; Phosphotransferases; Scattering, Radiation

2003
Wound reepithelialization activates a growth factor-responsive enhancer in migrating keratinocytes.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1998, Volume: 12, Issue:11

    Topics: Animals; Anisomycin; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; Cell Line; Cell Movement; Enhancer Elements, Genetic; Enzyme Inhibitors; Epithelium; Fibroblast Growth Factors; Flavonoids; Gene Expression Regulation; Genistein; Imidazoles; In Vitro Techniques; Keratinocytes; Membrane Glycoproteins; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Proteoglycans; Pyridines; Receptors, Growth Factor; Skin Physiological Phenomena; Suramin; Syndecan-1; Syndecans; Transcriptional Activation; Wound Healing

1998
Extracellular nucleotides activate the p38-stress-activated protein kinase cascade in glomerular mesangial cells.
    British journal of pharmacology, 2000, Volume: 129, Issue:3

    Topics: Activating Transcription Factor 2; Adenosine Triphosphate; Animals; Blotting, Western; Calcium-Calmodulin-Dependent Protein Kinases; Cattle; Cyclic AMP Response Element-Binding Protein; Enzyme Activation; Enzyme Inhibitors; Glomerular Mesangium; GTP-Binding Proteins; Imidazoles; Isoenzymes; Mitogen-Activated Protein Kinases; Nucleotides; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Stress, Physiological; Suramin; Transcription Factors; Uridine Triphosphate

2000
Early growth response-1 gene (Egr-1) promoter induction by ionizing radiation in U87 malignant glioma cells in vitro.
    European journal of biochemistry, 2002, Volume: 269, Issue:1

    Topics: Androstadienes; Anisomycin; Blotting, Western; Colforsin; DNA-Binding Proteins; Early Growth Response Protein 1; Epidermal Growth Factor; Flavonoids; Glioma; Humans; Imidazoles; Immediate-Early Proteins; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Pyridines; Suramin; Transcription Factors; Wortmannin

2002
[Activation of p38 and c-Jun NH2-terminal kinase mitogen-activated protein kinases in human prostate carcinoma cell lines with different metastatic potentials].
    Zhonghua bing li xue za zhi = Chinese journal of pathology, 2001, Volume: 30, Issue:3

    Topics: Adenosine Triphosphate; Cell Line, Tumor; Humans; Imidazoles; JNK Mitogen-Activated Protein Kinases; Male; Neoplasm Metastasis; p38 Mitogen-Activated Protein Kinases; Prostatic Neoplasms; Purinergic P2 Receptor Agonists; Pyridines; Signal Transduction; Suramin

2001