Page last updated: 2024-09-05

sb 203580 and staurosporine aglycone

sb 203580 has been researched along with staurosporine aglycone in 9 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(staurosporine aglycone)
Trials
(staurosporine aglycone)
Recent Studies (post-2010) (staurosporine aglycone)
3,48941,1377390175

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)staurosporine aglycone (IC50)
B2 bradykinin receptorCavia porcellus (domestic guinea pig)8
Serine/threonine-protein kinase D3Homo sapiens (human)2.45
cAMP-dependent protein kinase catalytic subunit alphaBos taurus (cattle)0.83
Beta-lactamaseEscherichia coli K-128
Protein kinase C gamma typeHomo sapiens (human)2.45
Protein kinase C beta typeHomo sapiens (human)2.45
Zinc finger protein GLI1Homo sapiens (human)1.8
Zinc finger protein GLI2Homo sapiens (human)2.7
Malate dehydrogenaseThermus thermophilus8
Cyclin-dependent kinase 4Homo sapiens (human)0.83
Protein kinase C alpha typeHomo sapiens (human)2.45
Chymotrypsinogen BHomo sapiens (human)10
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)8
G1/S-specific cyclin-D1Homo sapiens (human)0.83
Protein kinase C eta typeHomo sapiens (human)2.45
G1/S-specific cyclin-E1Homo sapiens (human)0.83
Cyclin-dependent kinase 2Homo sapiens (human)0.83
Protein kinase C iota typeHomo sapiens (human)2.45
Tyrosine-protein kinase JAK3Homo sapiens (human)0.061
Mitogen-activated protein kinase kinase kinase 9Homo sapiens (human)0.1083
Protein kinase C epsilon typeHomo sapiens (human)2.45
Mitogen-activated protein kinase kinase kinase 10Homo sapiens (human)0.0935
Protein kinase C theta typeHomo sapiens (human)2.45
Protein kinase C zeta typeHomo sapiens (human)2.45
Protein kinase C delta typeHomo sapiens (human)2.45
Calcium/calmodulin-dependent protein kinase type II subunit betaHomo sapiens (human)0.184
Calcium/calmodulin-dependent protein kinase type II subunit gammaHomo sapiens (human)0.184
Calcium/calmodulin-dependent protein kinase type II subunit deltaHomo sapiens (human)0.184
Serine/threonine-protein kinase D1Homo sapiens (human)2.45
Mitogen-activated protein kinase kinase kinase 11Homo sapiens (human)0.0787
Calcium/calmodulin-dependent protein kinase type II subunit alphaHomo sapiens (human)0.184

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (22.22)18.2507
2000's5 (55.56)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Caivano, M; Cohen, P; Davies, SP; Reddy, H1
McGovern, SL; Shoichet, BK1
Angeles, T; Bartlett, BA; Basma, AN; Dionne, CA; Finn, JP; Glicksman, MA; Knight, E; Maroney, AC; Matsuda, Y; Murphy, CA; Neff, NT; Walton, KM1
Koppal, T; Lukas, TJ; Mirzoeva, S; Petrova, TV; Van Eldik, LJ; Watterson, DM1
Hatanaka, H; Ikeuchi, T; Ishikawa, Y1
Iijima, R; Ishida, A; Kobayashi, A; Maeda, M1
El-Hashim, AZ; Jaffal, SM1
Chang, SL; Fong, YC; Hsu, CJ; Lin, CY; Tang, CH1
Egler, J; Lang, F; Zierle, J1

Other Studies

9 other study(ies) available for sb 203580 and staurosporine aglycone

ArticleYear
Specificity and mechanism of action of some commonly used protein kinase inhibitors.
    The Biochemical journal, 2000, Oct-01, Volume: 351, Issue:Pt 1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Acetophenones; Alkaloids; Amides; Animals; Benzamides; Benzophenanthridines; Benzopyrans; Butadienes; Cell Line; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Isoquinolines; Lithium; Magnesium; Nitriles; Phenanthridines; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Sirolimus; Substrate Specificity; Sulfonamides

2000
Kinase inhibitors: not just for kinases anymore.
    Journal of medicinal chemistry, 2003, Apr-10, Volume: 46, Issue:8

    Topics: beta-Lactamase Inhibitors; beta-Lactamases; Chymotrypsin; Enzyme Inhibitors; Kinetics; Light; Malate Dehydrogenase; Models, Biological; Phosphotransferases; Scattering, Radiation

2003
Motoneuron apoptosis is blocked by CEP-1347 (KT 7515), a novel inhibitor of the JNK signaling pathway.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Jan-01, Volume: 18, Issue:1

    Topics: Animals; Apoptosis; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cell Survival; Choline O-Acetyltransferase; COS Cells; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fetus; Gene Expression; Imidazoles; Indole Alkaloids; JNK Mitogen-Activated Protein Kinases; MAP Kinase Kinase 4; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Motor Neurons; Neurites; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Rats; Rats, Sprague-Dawley; Spinal Cord

1998
Screening in a cell-based assay for inhibitors of microglial nitric oxide production reveals calmodulin-regulated protein kinases as potential drug discovery targets.
    Brain research, 1999, Oct-09, Volume: 844, Issue:1-2

    Topics: Amidines; Animals; Benzylamines; Calcium Signaling; Calcium-Calmodulin-Dependent Protein Kinases; Carbazoles; Cell Line; Cell Nucleus; Cyclic AMP Response Element-Binding Protein; Drug Design; Enzyme Inhibitors; Flavonoids; Imidazoles; Indole Alkaloids; Isoquinolines; Lipopolysaccharides; Mice; Microglia; NF-kappa B; Nitric Oxide; Nitric Oxide Synthase; Phosphorylation; Pyridines; Staurosporine; Sulfonamides

1999
Brain-derived neurotrophic factor accelerates nitric oxide donor-induced apoptosis of cultured cortical neurons.
    Journal of neurochemistry, 2000, Volume: 75, Issue:2

    Topics: Animals; Apoptosis; Brain-Derived Neurotrophic Factor; Butadienes; Carbazoles; Cell Nucleus; Cell Survival; Cells, Cultured; Cerebral Cortex; Cycloheximide; Dactinomycin; DNA Fragmentation; Drug Synergism; Embryo, Mammalian; Enzyme Inhibitors; Female; Imidazoles; Immunoglobulin G; Indole Alkaloids; Kinetics; Male; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neurons; Nitric Oxide Donors; Nitriles; Nitroprusside; p38 Mitogen-Activated Protein Kinases; Pyridines; Rats; Rats, Wistar; Receptor, trkB; Signal Transduction

2000
Characterization of cAMP-dependent proteolysis of GATA-6.
    Biochemical and biophysical research communications, 2005, Jul-15, Volume: 332, Issue:4

    Topics: Animals; Base Sequence; Benzylamines; Binding Sites; Bucladesine; Carbazoles; Cell Nucleus; CHO Cells; Cricetinae; Cyclic AMP; DNA-Binding Proteins; Enzyme Inhibitors; Flavonoids; GATA6 Transcription Factor; Humans; Imidazoles; Indole Alkaloids; Isoquinolines; MAP Kinase Kinase Kinase 1; MAP Kinase Signaling System; Molecular Sequence Data; Mutation; Naphthalenes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Plasmids; Prostaglandin D2; Proteasome Endopeptidase Complex; Protein Binding; Pyridines; src-Family Kinases; Sulfonamides; Transcription Factors

2005
Nerve growth factor enhances cough and airway obstruction via TrkA receptor- and TRPV1-dependent mechanisms.
    Thorax, 2009, Volume: 64, Issue:9

    Topics: Airway Obstruction; Animals; Carbazoles; Citric Acid; Cough; Diterpenes; Enzyme Inhibitors; Female; Guinea Pigs; Imidazoles; Indole Alkaloids; Male; Nerve Growth Factors; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Receptor, trkA; TRPV Cation Channels

2009
Apoptosis signal-regulating kinase 1 is involved in brain-derived neurotrophic factor (BDNF)-enhanced cell motility and matrix metalloproteinase 1 expression in human chondrosarcoma cells.
    International journal of molecular sciences, 2013, Jul-25, Volume: 14, Issue:8

    Topics: Anthracenes; Bone Neoplasms; Brain-Derived Neurotrophic Factor; Carbazoles; Cell Line, Tumor; Cell Movement; Chondrosarcoma; Humans; Imidazoles; Indole Alkaloids; JNK Mitogen-Activated Protein Kinases; MAP Kinase Kinase Kinase 5; Matrix Metalloproteinase 1; Neoplasm Invasiveness; Neoplasm Metastasis; p38 Mitogen-Activated Protein Kinases; Prognosis; Protein Kinases; Pyridines; Receptor, trkB; Signal Transduction; Thioredoxins; Up-Regulation

2013
Stimulating Effect of Manumycin A on Suicidal Erythrocyte Death.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2016, Volume: 38, Issue:3

    Topics: Annexin A5; Calcium; Carbazoles; Cell Size; Eryptosis; Erythrocyte Membrane; Erythrocytes; Gene Expression Regulation; Humans; Imidazoles; Indole Alkaloids; p38 Mitogen-Activated Protein Kinases; Phosphatidylserines; Polyenes; Polyunsaturated Alkamides; Protein Kinase C; Pyridines; Reactive Oxygen Species

2016