Page last updated: 2024-09-05

sb 203580 and sb 242235

sb 203580 has been researched along with sb 242235 in 3 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(sb 242235)
Trials
(sb 242235)
Recent Studies (post-2010) (sb 242235)
3,48941,1372218

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)sb 242235 (IC50)
Heat shock protein beta-1Homo sapiens (human)0.16
Protein kinase C beta typeHomo sapiens (human)0.017
Protein kinase C alpha typeHomo sapiens (human)0.083
Mitogen-activated protein kinase 14Homo sapiens (human)0.0572

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barberia, JT; Carty, TJ; Cortina, SR; Csiki, C; Dipesa, AJ; Dombroski, MA; Elliott, NC; Gabel, CA; Jordan, CK; Labasi, JM; Letavic, MA; Martin, WH; McClure, KF; Peese, KM; Stock, IA; Svensson, L; Sweeney, FJ; Yu, CH1
Hajduk, PJ; Johnson, EF; Kifle, L; Merta, PJ; Metz, JT; Soni, NB1
Boyfield, I; Fonfria, E; Humphrey, PP; Michel, AD; Simon, J; Thompson, KM1

Other Studies

3 other study(ies) available for sb 203580 and sb 242235

ArticleYear
Benzimidazolone p38 inhibitors.
    Bioorganic & medicinal chemistry letters, 2004, Feb-23, Volume: 14, Issue:4

    Topics: Benzimidazoles; Enzyme Inhibitors; Imidazoles; Mitogen-Activated Protein Kinase 14; Mitogen-Activated Protein Kinases; Molecular Structure; Pyridines; Structure-Activity Relationship

2004
Navigating the kinome.
    Nature chemical biology, 2011, Volume: 7, Issue:4

    Topics: Drug Design; Pharmacogenetics; Protein Kinases; Proteome; Systems Biology

2011
Species and response dependent differences in the effects of MAPK inhibitors on P2X(7) receptor function.
    British journal of pharmacology, 2006, Volume: 149, Issue:7

    Topics: Adenosine Triphosphate; Animals; Calcium Signaling; Cell Line; Cell Membrane Permeability; Dose-Response Relationship, Drug; Ethidium; Humans; Imidazoles; Indicators and Reagents; Interleukin-1beta; Membrane Potentials; Mice; Mitogen-Activated Protein Kinases; Monocytes; Protein Kinase Inhibitors; Pyridines; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Recombinant Fusion Proteins; Species Specificity; Transfection

2006