Page last updated: 2024-09-05

sb 203580 and sb 216763

sb 203580 has been researched along with sb 216763 in 5 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(sb 216763)
Trials
(sb 216763)
Recent Studies (post-2010) (sb 216763)
3,48941,1373420225

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)sb 216763 (IC50)
G2/mitotic-specific cyclin-B2Homo sapiens (human)0.55
Cyclin-dependent kinase 1Homo sapiens (human)0.55
G2/mitotic-specific cyclin-B1Homo sapiens (human)0.55
Cyclin-A2Homo sapiens (human)0.269
Cyclin-dependent kinase 2Homo sapiens (human)0.269
Glycogen synthase kinase-3 alphaHomo sapiens (human)0.0477
Glycogen synthase kinase-3 betaHomo sapiens (human)0.0342
Cyclin-A1Homo sapiens (human)0.269
G2/mitotic-specific cyclin-B3Homo sapiens (human)0.55

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (60.00)29.6817
2010's1 (20.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Alessi, DR; Arthur, JS; Bain, J; Cohen, P; Elliott, M; Hastie, CJ; Klevernic, I; McLauchlan, H; Plater, L; Shpiro, N1
Albrecht, W; Ansideri, F; Döring, E; Haun, U; Heider, F; Koch, P; Kudolo, M; Laufer, SA; Pantsar, T; Poso, A; Tesch, R1
Basta-Kaim, A; Budziszewska, B; Jaworska-Feil, L; Kubera, M; Lasoń, W; Leśkiewicz, M; Tetich, M1
Choi, SE; Jang, HJ; Kang, Y; Kim, DJ; Kim, HE; Kim, HJ; Kim, HS; Lee, KW; Shin, HC1
Hao, C; Jiang, Y; Li, J; Ma, N; Xu, Z; Yin, L1

Other Studies

5 other study(ies) available for sb 203580 and sb 216763

ArticleYear
The selectivity of protein kinase inhibitors: a further update.
    The Biochemical journal, 2007, Dec-15, Volume: 408, Issue:3

    Topics: Amino Acid Sequence; Animals; Cell Line; Drug Design; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Recombinant Proteins; Spodoptera

2007
Pyridinylimidazoles as dual glycogen synthase kinase 3β/p38α mitogen-activated protein kinase inhibitors.
    European journal of medicinal chemistry, 2019, Aug-01, Volume: 175

    Topics: Amino Acid Sequence; Carbon-13 Magnetic Resonance Spectroscopy; Glycogen Synthase Kinase 3 beta; Humans; Imidazoles; Inhibitory Concentration 50; Molecular Docking Simulation; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Proton Magnetic Resonance Spectroscopy; Pyridines; Sequence Homology, Amino Acid; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship

2019
Mood stabilizers inhibit glucocorticoid receptor function in LMCAT cells.
    European journal of pharmacology, 2004, Jul-14, Volume: 495, Issue:2-3

    Topics: Amphetamine; Animals; Anthracenes; Antimanic Agents; Blotting, Western; Carbamazepine; Cell Line; Cell Survival; Chloramphenicol O-Acetyltransferase; Corticosterone; Dose-Response Relationship, Drug; Flavonoids; Gene Expression Regulation, Enzymologic; Imidazoles; Indoles; Inositol; Lithium; Maleimides; Protein Kinase C; Protein Kinase C-alpha; Pyridines; Receptors, Glucocorticoid; Tamoxifen; Tetradecanoylphorbol Acetate; Valproic Acid

2004
Involvement of glycogen synthase kinase-3beta in palmitate-induced human umbilical vein endothelial cell apoptosis.
    Journal of vascular research, 2007, Volume: 44, Issue:5

    Topics: Adenoviridae; Anthracenes; Apoptosis; Caspase 3; Cell Cycle; Cells, Cultured; Cytosol; Endothelial Cells; Endothelium, Vascular; Enzyme Activation; Fumonisins; Genetic Vectors; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; Humans; Imidazoles; Indoles; Lithium Chloride; Maleimides; Mitochondria; Palmitates; Phosphorylation; Phosphoserine; Poly(ADP-ribose) Polymerases; Protein Processing, Post-Translational; Pyridines; Thiadiazoles; Transduction, Genetic; Umbilical Veins

2007
Effects of signaling pathway inhibitors on hematopoietic stem cells.
    Molecular medicine reports, 2021, Volume: 23, Issue:1

    Topics: Animals; Cell Differentiation; Cell Self Renewal; Female; Glycogen Synthase Kinase 3 beta; Hematopoietic Stem Cells; Histone Deacetylase Inhibitors; Imidazoles; Indoles; Maleimides; Mice; p38 Mitogen-Activated Protein Kinases; Pyridines; Signal Transduction; TOR Serine-Threonine Kinases

2021