Page last updated: 2024-09-05

sb 203580 and saracatinib

sb 203580 has been researched along with saracatinib in 4 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(saracatinib)
Trials
(saracatinib)
Recent Studies (post-2010) (saracatinib)
3,48941,13719425157

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)saracatinib (IC50)
Chain A, Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)0.0027
Tyrosine-protein kinase ABL1Homo sapiens (human)0.03
Epidermal growth factor receptorHomo sapiens (human)1.9615
Tyrosine-protein kinase LckHomo sapiens (human)0.004
Tyrosine-protein kinase YesHomo sapiens (human)0.0038
Mast/stem cell growth factor receptor KitHomo sapiens (human)0.2
Proto-oncogene tyrosine-protein kinase SrcHomo sapiens (human)0.0093
Platelet-derived growth factor receptor alphaHomo sapiens (human)10
Cyclin-dependent kinase 2Homo sapiens (human)10
Vascular endothelial growth factor receptor 2Homo sapiens (human)0.0027
Tyrosine-protein kinase CSKHomo sapiens (human)0.84
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinaseHomo sapiens (human)5.209

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (25.00)24.3611
2020's3 (75.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Bharate, SB; Raghuvanshi, R1
Caballero, E; García-Cárceles, J; Gil, C; Martínez, A1
Laufer, S; Pillaiyar, T1

Reviews

2 review(s) available for sb 203580 and saracatinib

ArticleYear
Kinase Inhibitors as Underexplored Antiviral Agents.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Animals; Antiviral Agents; Drug Repositioning; Humans; Protein Kinase Inhibitors; Virus Diseases; Viruses

2022
Kinases as Potential Therapeutic Targets for Anti-coronaviral Therapy.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Antiviral Agents; COVID-19; COVID-19 Drug Treatment; Humans; Protein Kinase Inhibitors; SARS-CoV-2; Signal Transduction; Virus Replication

2022

Other Studies

2 other study(ies) available for sb 203580 and saracatinib

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
Recent Developments in the Use of Kinase Inhibitors for Management of Viral Infections.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Antiviral Agents; COVID-19; COVID-19 Drug Treatment; Drug Approval; Drug Repositioning; High-Throughput Screening Assays; Humans; Protein Kinase Inhibitors; SARS-CoV-2; United States; United States Food and Drug Administration; Virus Diseases

2022