Page last updated: 2024-09-05

sb 203580 and riluzole

sb 203580 has been researched along with riluzole in 3 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(riluzole)
Trials
(riluzole)
Recent Studies (post-2010) (riluzole)
3,48941,1371,244153572

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)riluzole (IC50)
Sodium channel protein type 2 subunit alphaRattus norvegicus (Norway rat)4.73
Cytochrome P450 1A2Homo sapiens (human)10
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)1.733
Sodium-dependent noradrenaline transporter Homo sapiens (human)1.733

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Hata, Y; Ichisaka, S; Kaneko, R; Kato, K; Katoh-Semba, R; Kitajima, S; Miyazaki, N; Takahashi, Y; Tsuzuki, M; Yamada, H1
Bertz, J; Gladbach, A; Ittner, AA; Ittner, LM; Suh, LS1

Other Studies

3 other study(ies) available for sb 203580 and riluzole

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013
Activation of p38 mitogen-activated protein kinase is required for in vivo brain-derived neurotrophic factor production in the rat hippocampus.
    Neuroscience, 2009, Sep-29, Volume: 163, Issue:1

    Topics: Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Animals; Anisomycin; Brain-Derived Neurotrophic Factor; Calcium Channel Blockers; Calcium Channels, N-Type; Enzyme Activation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Hippocampus; Imidazoles; Male; Neurons; p38 Mitogen-Activated Protein Kinases; Protein Synthesis Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Riluzole; Up-Regulation

2009
p38 MAP kinase-mediated NMDA receptor-dependent suppression of hippocampal hypersynchronicity in a mouse model of Alzheimer's disease.
    Acta neuropathologica communications, 2014, Oct-21, Volume: 2

    Topics: Alzheimer Disease; Animals; Disease Models, Animal; Dizocilpine Maleate; Electrodes, Implanted; Electroencephalography; Enzyme Inhibitors; Epilepsy; Excitatory Amino Acid Antagonists; Gamma Rhythm; Hippocampus; Imidazoles; Male; Mice, Inbred C57BL; Mice, Transgenic; p38 Mitogen-Activated Protein Kinases; Pyridines; Receptors, N-Methyl-D-Aspartate; Riluzole; Theta Rhythm

2014