Page last updated: 2024-09-05

sb 203580 and r 59949

sb 203580 has been researched along with r 59949 in 3 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(r 59949)
Trials
(r 59949)
Recent Studies (post-2010) (r 59949)
3,48941,13755021

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)r 59949 (IC50)
TPA: protein transporter TIM10Saccharomyces cerevisiae S288C12.7
TPA: protein transporter TIM23Saccharomyces cerevisiae S288C5.44
Diacylglycerol kinase alphaHomo sapiens (human)0.3

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A1
Goto, K; Hozumi, Y; Nakano, T; Wakabayashi, I1

Other Studies

3 other study(ies) available for sb 203580 and r 59949

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
    The Biochemical journal, 2013, Apr-15, Volume: 451, Issue:2

    Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase

2013
Involvement of diacylglycerol kinase γ in modulation of iNOS synthesis in Golgi apparatus of vascular endothelial cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 2012, Volume: 385, Issue:8

    Topics: Animals; Aorta, Thoracic; Blotting, Western; Brefeldin A; Diacylglycerol Kinase; Endothelial Cells; Enzyme Inhibitors; Golgi Apparatus; Imidazoles; Immunohistochemistry; Interleukin-1beta; Isoenzymes; Male; Nitric Oxide Synthase Type II; Nocodazole; Piperidines; Protein Synthesis Inhibitors; Pyridines; Quinazolinones; Rats; Rats, Wistar; Real-Time Polymerase Chain Reaction; RNA, Messenger

2012