sb 203580 has been researched along with piperidines in 24 studies
Studies (sb 203580) | Trials (sb 203580) | Recent Studies (post-2010) (sb 203580) | Studies (piperidines) | Trials (piperidines) | Recent Studies (post-2010) (piperidines) |
---|---|---|---|---|---|
3,489 | 4 | 1,137 | 40,235 | 5,221 | 14,545 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (12.50) | 18.2507 |
2000's | 9 (37.50) | 29.6817 |
2010's | 12 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Coffey, ET; Courtney, MJ | 1 |
Ishida, T; Kawai, M; Kawashima, S; Namiki, M; Rikitake, Y; Sakoda, T; Ueyama, T; Yokoyama, M | 1 |
Kato, K; Kawamura, H; Kozawa, O; Matsui, N; Matsuno, H; Niwa, M; Otsuka, T; Uematsu, T | 1 |
Buhl, T; Di Padova, FE; Feifel, R; Gram, H; Hiestand, P; Manning, U; Revesz, L; Zimmerlin, AG | 1 |
Brune, K; Hinz, B; Pahl, A; Ramer, R | 1 |
Balla, A; Csermely, P; Dénes, L; Hargitai, J; Jednákovits, A; Krajcsi, P; Pénzes, Z; Tálosi, L | 1 |
Bouchard, JF; Lagneux, C; Lamontagne, D; Lépicier, P | 1 |
Alger, BE; Mason, SE; Reich, CG | 1 |
Han, H; Long, H; Wang, H; Wang, J; Wang, Z; Xu, D; Zhang, Y | 1 |
Akamatsu, S; Hirade, K; Ishisaki, A; Kanno, Y; Kato, K; Kozawa, O; Matsuno, H; Nakajima, K; Oiso, Y; Shu, E; Suga, H; Takai, S; Tanabe, K | 1 |
Farge, D; Mauviel, A; Michel, L; Tacheau, C; Verrecchia, F | 1 |
Calderone, A; Dupuis, J; Préfontaine, A | 1 |
Fortes, B; Hurley, DJ; Linden, J; Moore, JN; Sun, WC; Thompson, R; Vandenplas, ML | 1 |
Giacobbe, E; Leoncini, G; Signorello, MG | 1 |
Chen, YL; Chen, ZC; Lv, Y; Shen, X; Zhao, G | 1 |
Forman, SP; Katzenberg, G; Ohanian, J; Ohanian, V | 1 |
Goto, K; Hozumi, Y; Nakano, T; Wakabayashi, I | 1 |
Li, M; She, T; Shi, C; Wang, B; Yu, L | 1 |
Cheng, M; Li, M; Meng, W; She, T; Shi, C; Wang, B; Yu, L | 1 |
E, LL; Liang, L; Liu, H; Liu, N; Wang, DS; Yu, J; Zhou, W | 1 |
Chay, KO; Joo, YE; Jung, YD; Khoi, PN; Kim, KK; Lian, S; Xia, Y; Yoon, HJ | 1 |
Chen, G; Deng, L; Song, F; Zhang, L; Zhao, H; Zhu, H | 1 |
Lin, R; Si, L; Yang, R; Yang, S | 1 |
Bay-Jensen, AC; Hägglund, P; Karsdal, MA; Kayed, A; Kjelgaard-Petersen, CF; Mobasheri, A; Sharma, N; Thudium, CS | 1 |
24 other study(ies) available for sb 203580 and piperidines
Article | Year |
---|---|
The mechanism of Ara-C-induced apoptosis of differentiating cerebellar granule neurons.
Topics: Androstadienes; Animals; Antimetabolites, Antineoplastic; Apoptosis; Benzamides; CDC2 Protein Kinase; CDC2-CDC28 Kinases; Cell Differentiation; Cell Survival; Cerebellum; Cyclin-Dependent Kinase 2; Cyclin-Dependent Kinase 4; Cyclin-Dependent Kinase 5; Cyclin-Dependent Kinases; Cytarabine; Enzyme Inhibitors; Flavonoids; Imatinib Mesylate; Imidazoles; Mitogen-Activated Protein Kinase 12; Mitogen-Activated Protein Kinases; Neurons; Piperazines; Piperidines; Poly (ADP-Ribose) Polymerase-1; Poly(ADP-ribose) Polymerases; Protein Kinases; Protein Serine-Threonine Kinases; Proteins; Proto-Oncogene Proteins; Purines; Pyridines; Pyrimidines; Rats; Roscovitine; Signal Transduction; Stress, Physiological; Wortmannin | 1999 |
Endothelin-1 activates p38 mitogen-activated protein kinase via endothelin-A receptor in rat myocardial cells.
Topics: Animals; Blotting, Western; Cardiomegaly; Cells, Cultured; Dose-Response Relationship, Drug; Endothelin-1; Enzyme Activation; Enzyme Inhibitors; Imidazoles; Leucine; Mitogen-Activated Protein Kinases; Myocardium; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phosphorylation; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptors, Endothelin; Sarcomeres | 1999 |
Endothelin-1 stimulates heat shock protein 27 induction in osteoblasts: involvement of p38 MAP kinase.
Topics: Animals; Antihypertensive Agents; Blotting, Northern; Carcinogens; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Estrenes; Flavonoids; Gene Expression Regulation, Enzymologic; Genistein; Heat-Shock Proteins; Imidazoles; Mice; Mitogen-Activated Protein Kinases; Naphthalenes; Oligopeptides; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phorbol Esters; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Propranolol; Protein Kinase C; Pyridines; Pyrrolidinones; RNA, Messenger; Skull; Staurosporine | 1999 |
SAR of 4-hydroxypiperidine and hydroxyalkyl substituted heterocycles as novel p38 map kinase inhibitors.
Topics: Animals; Enzyme Inhibitors; Heterocyclic Compounds; Humans; Imidazoles; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Piperidines; Pyridines; Rats; Structure-Activity Relationship | 2000 |
R(+)-methanandamide induces cyclooxygenase-2 expression in human neuroglioma cells via a non-cannabinoid receptor-mediated mechanism.
Topics: Analgesics, Non-Narcotic; Arachidonic Acids; Blotting, Western; Brain Neoplasms; Cannabinoid Receptor Modulators; Cell Line; Central Nervous System; Cyclooxygenase 2; Dinoprostone; Dose-Response Relationship, Drug; Dronabinol; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Glioma; Humans; Imidazoles; Interleukin-1; Isoenzymes; Membrane Proteins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Pertussis Toxin; Phosphorylation; Piperidines; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Pyridines; Receptors, Cannabinoid; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Tumor Cells, Cultured; Virulence Factors, Bordetella | 2001 |
Pharmacologically activated migration of aortic endothelial cells is mediated through p38 SAPK.
Topics: Animals; Aorta; Blotting, Western; Cattle; Cell Movement; Endothelial Growth Factors; Endothelium; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Mitogen-Activated Protein Kinases; Oxazines; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Piperidines; Pyridines | 2002 |
Endocannabinoids protect the rat isolated heart against ischaemia.
Topics: Amides; Animals; Arachidonic Acids; Biomarkers; Blotting, Western; Camphanes; Cannabinoid Receptor Modulators; Endocannabinoids; Ethanolamines; Glycerides; Heart; Imidazoles; L-Lactate Dehydrogenase; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Myocardial Infarction; Myocardial Ischemia; Myocardial Reperfusion Injury; p38 Mitogen-Activated Protein Kinases; Palmitic Acids; Piperidines; Protein Kinase C; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Rimonabant; Signal Transduction | 2003 |
Novel form of LTD induced by transient, partial inhibition of the Na,K-pump in rat hippocampal CA1 cells.
Topics: Animals; Drug Interactions; Electric Stimulation; Electrophysiology; Enzyme Inhibitors; Evoked Potentials; Hippocampus; Imidazoles; In Vitro Techniques; Indoles; Long-Term Synaptic Depression; Male; Maleimides; Neural Inhibition; Neurons; Ouabain; Peptides; Piperidines; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Sodium-Potassium-Exchanging ATPase; Time Factors | 2004 |
HERG K channel conductance promotes H2O2-induced apoptosis in HEK293 cells: cellular mechanisms.
Topics: Anti-Arrhythmia Agents; Caspase 3; Caspase 9; Caspases; Cell Line; DNA Fragmentation; Enzyme Inhibitors; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Humans; Hydrogen Peroxide; Imidazoles; p38 Mitogen-Activated Protein Kinases; Piperidines; Poly(ADP-ribose) Polymerases; Potassium Channels, Voltage-Gated; Pyridines; Signal Transduction | 2004 |
Possible involvement of phosphatidylinositol 3-kinase/Akt signal pathway in vasopressin-induced HSP27 phosphorylation in aortic smooth muscle A10 cells.
Topics: Animals; Aorta; Blotting, Western; Cell Line; Chromones; Enzyme Inhibitors; Heat-Shock Proteins; HSP27 Heat-Shock Proteins; Imidazoles; MAP Kinase Signaling System; Molecular Chaperones; Morpholines; Muscle, Smooth; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Neoplasm Proteins; Phosphatidylinositol 3-Kinases; Phosphorylation; Piperidines; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Quinolones; Rats; Time Factors; Vasopressins | 2005 |
Involvement of ERK signaling in halofuginone-driven inhibition of fibroblast ability to contract collagen lattices.
Topics: Blotting, Western; Butadienes; Cell Line; Cell Proliferation; Cell Survival; Collagen Type I; Dose-Response Relationship, Drug; Extracellular Matrix; Extracellular Signal-Regulated MAP Kinases; Fibroblasts; Flavonoids; Humans; Imidazoles; MAP Kinase Signaling System; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Piperidines; Protein Synthesis Inhibitors; Pyridines; Quinazolinones; Time Factors | 2007 |
Role of endothelin receptors on basal and endothelin-1-stimulated lung myofibroblast proliferation.
Topics: Animals; Cell Proliferation; Cells, Cultured; Chromones; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Enzyme Inhibitors; Fibroblasts; Imidazoles; Lung; Male; Morpholines; Myoblasts, Smooth Muscle; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phosphoinositide-3 Kinase Inhibitors; Piperidines; Pyridines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B | 2008 |
Differential modulation of lipopolysaccharide-induced expression of inflammatory genes in equine monocytes through activation of adenosine A2A receptors.
Topics: Adenosine A2 Receptor Agonists; Animals; Base Sequence; Bucladesine; Cyclooxygenase 2; Cytokines; DNA Primers; Drug Synergism; Gene Expression; Horses; Imidazoles; In Vitro Techniques; Inflammation Mediators; Interleukin-10; Lipopolysaccharides; Monocytes; Piperidines; Pyridines; Receptor, Adenosine A2A | 2010 |
Activation by 2-arachidonoylglycerol of platelet p38MAPK/cPLA2 pathway.
Topics: Apyrase; Arachidonic Acid; Arachidonic Acids; Blood Platelets; Endocannabinoids; Glycerides; Humans; Imidazoles; In Vitro Techniques; Indomethacin; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Phospholipases A2, Cytosolic; Phosphorylation; Piperidines; Pyrazoles; Pyridines; Reactive Oxygen Species; Rimonabant; Signal Transduction | 2011 |
[Protective effect of remifentanil preconditioning against hepatic ischemia-reperfusion injury in rats: role of p38 mitogen-activated protein kinases].
Topics: Alanine Transaminase; Animals; Aspartate Aminotransferases; Imidazoles; Interleukin-1beta; Ischemia; Ischemic Preconditioning; Liver; Male; MAP Kinase Signaling System; p38 Mitogen-Activated Protein Kinases; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Remifentanil; Reperfusion Injury; Tumor Necrosis Factor-alpha | 2011 |
Endothelin-1 stimulates small artery VCAM-1 expression through p38MAPK-dependent neutral sphingomyelinase.
Topics: Aniline Compounds; Animals; Benzylidene Compounds; Endothelin B Receptor Antagonists; Endothelin-1; HSP27 Heat-Shock Proteins; Imidazoles; Mesenteric Arteries; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Piperidines; Pyridines; Rats; Sphingomyelin Phosphodiesterase; Vascular Cell Adhesion Molecule-1 | 2012 |
Involvement of diacylglycerol kinase γ in modulation of iNOS synthesis in Golgi apparatus of vascular endothelial cells.
Topics: Animals; Aorta, Thoracic; Blotting, Western; Brefeldin A; Diacylglycerol Kinase; Endothelial Cells; Enzyme Inhibitors; Golgi Apparatus; Imidazoles; Immunohistochemistry; Interleukin-1beta; Isoenzymes; Male; Nitric Oxide Synthase Type II; Nocodazole; Piperidines; Protein Synthesis Inhibitors; Pyridines; Quinazolinones; Rats; Rats, Wistar; Real-Time Polymerase Chain Reaction; RNA, Messenger | 2012 |
[Endothelin-1 stimulates the expression of pacemaker channel I(f) in cardiomyocytes through a p38 MAPK-independent signaling pathway].
Topics: Animals; Animals, Newborn; Cyclic Nucleotide-Gated Cation Channels; Endothelin-1; Imidazoles; Myocytes, Cardiac; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Patch-Clamp Techniques; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Signal Transduction | 2012 |
Endothelin-1 stimulates the expression of L-type Ca2+ channels in neonatal rat cardiomyocytes via the extracellular signal-regulated kinase 1/2 pathway.
Topics: Animals; Animals, Newborn; Anthracenes; Blotting, Western; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Flavonoids; Imidazoles; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocytes, Cardiac; Oligopeptides; Patch-Clamp Techniques; Peptides, Cyclic; Piperidines; Pyridines; Rats; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction | 2013 |
Endothelin-1 stimulates proinflammatory cytokine expression in human periodontal ligament cells via mitogen-activated protein kinase pathway.
Topics: Adult; Anthracenes; Calcium-Calmodulin-Dependent Protein Kinases; Cell Culture Techniques; Cells, Cultured; Cytokines; Dose-Response Relationship, Drug; Endothelin B Receptor Antagonists; Endothelin Receptor Antagonists; Endothelin-1; Female; Flavonoids; Humans; Imidazoles; Interleukin-1beta; Interleukin-6; JNK Mitogen-Activated Protein Kinases; Male; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Periodontal Ligament; Periodontitis; Piperidines; Pyridines; Time Factors; Tumor Necrosis Factor-alpha | 2014 |
Piperine inhibits IL-1β-induced IL-6 expression by suppressing p38 MAPK and STAT3 activation in gastric cancer cells.
Topics: Alkaloids; Benzodioxoles; Blotting, Western; Cell Line, Tumor; Cell Movement; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation, Neoplastic; Humans; Imidazoles; Interleukin-1beta; Interleukin-6; Mutation; Neoplasm Invasiveness; p38 Mitogen-Activated Protein Kinases; Piperidines; Polyunsaturated Alkamides; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA Interference; STAT3 Transcription Factor; Stomach Neoplasms; UDPglucose 4-Epimerase | 2015 |
The role of p38MAPK activation in spinal dorsal horn in remifentanil-induced postoperative hyperalgesia in rats.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Anti-Inflammatory Agents, Non-Steroidal; Disease Models, Animal; Enzyme Activation; Hyperalgesia; Imidazoles; Male; p38 Mitogen-Activated Protein Kinases; Pain Measurement; Pain Threshold; Pain, Postoperative; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Remifentanil; Spinal Cord Dorsal Horn; Time Factors | 2016 |
Piperine functions as a tumor suppressor for human ovarian tumor growth via activation of JNK/p38 MAPK-mediated intrinsic apoptotic pathway.
Topics: Alkaloids; Anthracenes; Apoptosis; Benzodioxoles; Caspase 3; Caspase 9; Caspase Inhibitors; Cell Proliferation; Cell Survival; Female; Humans; Imidazoles; MAP Kinase Kinase 4; Oligopeptides; Ovarian Neoplasms; p38 Mitogen-Activated Protein Kinases; Piperidines; Polyunsaturated Alkamides; Pyridines; Tumor Suppressor Proteins | 2018 |
Tofacitinib and TPCA-1 exert chondroprotective effects on extracellular matrix turnover in bovine articular cartilage ex vivo.
Topics: Amides; Animals; Cartilage, Articular; Cattle; Chondrocytes; Collagen Type II; Extracellular Matrix Proteins; Imidazoles; Osteoarthritis; Oxazines; Piperidines; Proteoglycans; Pyridines; Pyrimidines; Pyrroles; Thiophenes | 2019 |