sb 203580 has been researched along with pd 169316 in 32 studies
Studies (sb 203580) | Trials (sb 203580) | Recent Studies (post-2010) (sb 203580) | Studies (pd 169316) | Trials (pd 169316) | Recent Studies (post-2010) (pd 169316) |
---|---|---|---|---|---|
3,489 | 4 | 1,137 | 119 | 0 | 40 |
Protein | Taxonomy | sb 203580 (IC50) | pd 169316 (IC50) |
---|---|---|---|
Tyrosinase | Mus musculus (house mouse) | 0.089 | |
Mitogen-activated protein kinase 14 | Homo sapiens (human) | 0.089 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 26 (81.25) | 29.6817 |
2010's | 6 (18.75) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M | 1 |
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A | 1 |
Jung, SH; Manickam, M; Namasivayam, V; Pillaiyar, T | 1 |
Hatakeyama, D; Kawamura, H; Kozawa, O; Matsuno, H; Uematsu, T | 1 |
Kawamura, H; Kozawa, O; Matsuno, H; Uematsu, T | 1 |
Clarkson, ED; Esplen, JE; Freed, CR; Heidenreich, KA; Marotti, J; Meintzer, MK; Rao, P; Wang, X; Zawada, WM | 1 |
Inaguma, Y; Ito, H; Iwamoto, I; Kato, K; Lida, K | 1 |
Dutta, S; McGinnis, K; Nath, R; Shivers, B; Wang, KK | 1 |
Bayon, Y; Lopez-Hernandez, FJ; Ortiz, MA; Pfahl, M; Piedrafita, FJ | 1 |
Akamatsu, S; Dohi, S; Hirose, H; Kozawa, O; Matsuno, H; Tanabe, K; Uematsu, T; Yamamoto, T | 1 |
Hatakeyama, D; Kozawa, O; Uematsu, T | 1 |
Arena, S; Benatti, U; Corsaro, A; Damonte, G; Florio, T; Millo, E; Schettini, G; Tagliavini, F; Thellung, S; Villa, V | 1 |
Hatakeyama, D; Ito, H; Kato, K; Kozawa, O; Matsuno, H; Niwa, M; Shibata, T; Tatematsu, N; Uematsu, T | 1 |
Hatakeyama, D; Kato, K; Kozawa, O; Matsuno, H; Niwa, M; Oiso, Y; Tokuda, H; Uematsu, T | 1 |
Akamatsu, S; Hirade, K; Ito, H; Katagiri, Y; Kato, K; Kozawa, O; Matsuno, H; Niwa, M; Oiso, Y; Tanabe, K; Uematsu, T | 1 |
Bodero, AJ; Lees-Miller, SP; Ye, R | 1 |
Hara, A; Hatakeyama, D; Hirade, K; Hotta, K; Ito, H; Kanamori, Y; Katayama, M; Kato, K; Kozawa, O; Matsuno, H; Mori, H; Niwa, M; Uematsu, T | 1 |
Hatakeyama, D; Hirade, K; Ito, H; Kato, K; Kozawa, O; Niwa, M; Tokuda, H; Wang, X | 1 |
Akamatsu, S; Hatakeyama, D; Kozawa, O; Shibata, T; Tanabe, K; Tokuda, H; Yoshida, M | 1 |
Boeuf, H; Duval, D; Kedinger, C; Malaisé, M; Reinhardt, B | 1 |
Harada, A; Ishisaki, A; Kanno, Y; Kozawa, O; Takenaka, M; Tokuda, H | 1 |
Akamatsu, S; Hirade, K; Ishisaki, A; Kato, K; Kozawa, O; Matsuno, H; Nakajima, K; Oiso, Y; Suga, H; Takei, M; Takenaka, M; Tanabe, K; Yoshimi, N | 1 |
Jungnelius, M; Karlsson, OP; Karlsson, R; Nordin, H | 1 |
Hirade, K; Ishisaki, A; Kanno, Y; Katagiri, Y; Kitajima, Y; Kozawa, O; Matsuno, H; Nakajima, K; Shu, E; Suga, H | 1 |
Akamatsu, S; Dohi, S; Kato, K; Kozawa, O; Suga, H; Takai, S; Tanabe, K | 1 |
Askari, N; Avitzour, M; Diskin, R; Engelberg, D; Livnah, O; Raboy, B | 1 |
Bailey, SR; Brooks, AC; Cunningham, FM; Elliott, J; Menzies-Gow, NJ; Wheeler-Jones, C | 2 |
Alcaín, FJ; Ariza, J; Barbarroja, N; González-Aragón, D; Jódar, L; López-Pedrera, C; Villalba, JM | 1 |
de Bittencourt Pasquali, MA; Gasparotto, J; Gelain, DP; Moreira, JC; Pires, AS; Terra, SR; Zeidán-Chuliá, F | 1 |
Damaj, MI; Jayanthi, LD; Mannangatti, P; NarasimhaNaidu, K; Ramamoorthy, S | 1 |
Hamanoue, M; Kobayashi, M; Shigiyama, F; Takamatsu, K | 1 |
1 review(s) available for sb 203580 and pd 169316
Article | Year |
---|---|
Inhibitors of Melanogenesis: An Updated Review.
Topics: alpha-MSH; Biphenyl Compounds; Crystallization; Enzyme Inhibitors; Humans; Melanins; Monophenol Monooxygenase; Peptidomimetics; Radiation, Ionizing; Resveratrol; Signal Transduction; Skin | 2018 |
31 other study(ies) available for sb 203580 and pd 169316
Article | Year |
---|---|
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases | 2007 |
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase | 2013 |
Endothelin-1 induces vascular endothelial growth factor synthesis in osteoblasts: involvement of p38 mitogen-activated protein kinase.
Topics: Animals; Endothelial Growth Factors; Endothelin-1; Enzyme Inhibitors; Estrenes; Flavonoids; Gene Expression Regulation; Imidazoles; Lymphokines; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinases; Naphthalenes; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phorbol Esters; Protein Kinase C; Pyridines; Pyrrolidinones; Receptor, Endothelin A; Receptors, Endothelin; Tetradecanoylphorbol Acetate; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2000 |
p38 MAP kinase is involved in the signalling of sphingosine in osteoblasts: sphingosine inhibits prostaglandin F(2alpha)-induced phosphoinositide hydrolysis.
Topics: Animals; Blotting, Western; Dinoprost; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Hydrolysis; Imidazoles; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositols; Phosphorylation; Pyridines; Signal Transduction; Sodium Fluoride; Sphingosine; Time Factors | 2000 |
Inhibitors of p38 MAP kinase increase the survival of transplanted dopamine neurons.
Topics: Animals; Brain Tissue Transplantation; Cell Survival; Cells, Cultured; Dopamine; Enzyme Inhibitors; Fetus; Graft Survival; Imidazoles; Male; Mitogen-Activated Protein Kinases; Neurons; p38 Mitogen-Activated Protein Kinases; Parkinsonian Disorders; Pyridines; Rats; Rats, Sprague-Dawley; Recovery of Function | 2001 |
Protein kinase inhibitors can suppress stress-induced dissociation of Hsp27.
Topics: Anisomycin; Arsenites; Butadienes; Cadmium Chloride; Carcinogens; Dithiothreitol; Enzyme Inhibitors; Flavonoids; Glioma; Heat-Shock Proteins; Humans; Hydrogen Peroxide; Imidazoles; MAP Kinase Kinase Kinases; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Nitriles; Osmotic Pressure; Oxidants; p38 Mitogen-Activated Protein Kinases; Protein Kinase C; Protein Synthesis Inhibitors; Pyridines; Sodium Compounds; Sorbitol; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured | 2001 |
Inhibition of p38 kinase mimics survival signal-linked protection against apoptosis in rat cerebellar granule neurons.
Topics: Animals; Apoptosis; Blotting, Western; Caspase 3; Caspase Inhibitors; Caspases; Cell Survival; Cells, Cultured; Cerebellum; Dose-Response Relationship, Drug; Fluorescence; Imidazoles; Inhibitory Concentration 50; Microscopy, Phase-Contrast; Mitogen-Activated Protein Kinases; Neurons; p38 Mitogen-Activated Protein Kinases; Potassium; Potassium Deficiency; Pyridines; Rats; Signal Transduction | 2001 |
Retinoid-related molecules induce cytochrome c release and apoptosis through activation of c-Jun NH(2)-terminal kinase/p38 mitogen-activated protein kinases.
Topics: Apoptosis; Caspases; Cytochrome c Group; Enzyme Activation; Enzyme Inhibitors; Humans; Imidazoles; Isoenzymes; JNK Mitogen-Activated Protein Kinases; Jurkat Cells; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Pyridines; Retinoids | 2001 |
1,25-dihydroxyvitamin D3 stimulates vascular endothelial growth factor release in aortic smooth muscle cells: role of p38 mitogen-activated protein kinase.
Topics: 24,25-Dihydroxyvitamin D 3; Animals; Aorta; Calcitriol; Cells, Cultured; Drug Interactions; Endothelial Growth Factors; Imidazoles; Lymphokines; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Rats; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2002 |
Divergent regulation by p44/p42 MAP kinase and p38 MAP kinase of bone morphogenetic protein-4-stimulated osteocalcin synthesis in osteoblasts.
Topics: Bone Morphogenetic Protein 4; Bone Morphogenetic Proteins; Butadienes; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Imidazoles; JNK Mitogen-Activated Protein Kinases; Kinetics; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nitriles; Osteoblasts; Osteocalcin; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines | 2002 |
p38 MAP kinase mediates the cell death induced by PrP106-126 in the SH-SY5Y neuroblastoma cells.
Topics: Amino Acid Chloromethyl Ketones; Apoptosis; Caspase 3; Caspases; Cysteine Proteinase Inhibitors; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; Mitogen-Activated Protein Kinases; Neuroblastoma; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptide Fragments; Prion Diseases; Prions; Pyridines; Tumor Cells, Cultured | 2002 |
Upregulation by retinoic acid of transforming growth factor-beta-stimulated heat shock protein 27 induction in osteoblasts: involvement of mitogen-activated protein kinases.
Topics: Animals; Blotting, Northern; Cell Line; Enzyme Activation; Flavonoids; Heat-Shock Proteins; Imidazoles; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; RNA, Messenger; Signal Transduction; Transforming Growth Factor beta; Tretinoin; Up-Regulation | 2002 |
Specific induction of heat shock protein 27 by glucocorticoid in osteoblasts.
Topics: Animals; Cell Line; Cells, Cultured; Dexamethasone; Heat-Shock Proteins; HSP70 Heat-Shock Proteins; HSP90 Heat-Shock Proteins; Imidazoles; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinases; Osteoblasts; Phosphorylation; Pyridines; RNA, Messenger | 2002 |
Thrombin stimulates dissociation and induction of HSP27 via p38 MAPK in vascular smooth muscle cells.
Topics: Animals; Aorta; Blotting, Northern; Cells, Cultured; Enzyme Inhibitors; Heat-Shock Proteins; Hemostatics; HSP27 Heat-Shock Proteins; HSP70 Heat-Shock Proteins; Imidazoles; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Muscle, Smooth, Vascular; Neoplasm Proteins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Rats; RNA, Messenger; Thrombin | 2002 |
UV-light induces p38 MAPK-dependent phosphorylation of Bcl10.
Topics: Adaptor Proteins, Signal Transducing; B-Cell CLL-Lymphoma 10 Protein; Carrier Proteins; Cell Line; Dose-Response Relationship, Radiation; Enzyme Inhibitors; HeLa Cells; Humans; Imidazoles; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Tumor Cells, Cultured; Ultraviolet Rays | 2003 |
Involvement of p38 mitogen-activated protein kinase in heat shock protein 27 induction in human neutrophils.
Topics: Apoptosis; Calcium-Calmodulin-Dependent Protein Kinases; Cycloheximide; Dactinomycin; Dose-Response Relationship, Drug; Enzyme Induction; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Heat-Shock Proteins; Humans; Imidazoles; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neutrophils; Nucleic Acid Synthesis Inhibitors; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase C; Protein Synthesis Inhibitors; Pyridines; Pyrrolidines; RNA, Messenger; Thiocarbamates; Time Factors; Tumor Necrosis Factor-alpha | 2003 |
Mechanism of simvastatin on induction of heat shock protein in osteoblasts.
Topics: 3T3 Cells; Animals; Cycloheximide; Dose-Response Relationship, Drug; Enzyme Inhibitors; Heat-Shock Proteins; Imidazoles; Lovastatin; Mice; Mitogen-Activated Protein Kinases; Osteoblasts; Osteogenesis; p38 Mitogen-Activated Protein Kinases; Pyridines; Reproducibility of Results; RNA, Messenger; Sensitivity and Specificity; Simvastatin | 2003 |
Involvement of MAP kinases in TGF-beta-stimulated vascular endothelial growth factor synthesis in osteoblasts.
Topics: 3T3 Cells; Angiogenesis Inducing Agents; Animals; Butadienes; Dose-Response Relationship, Drug; Drug Synergism; Endothelial Growth Factors; Flavonoids; Imidazoles; Intercellular Signaling Peptides and Proteins; Lymphokines; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nitriles; Osteoblasts; Pyridines; Transforming Growth Factor beta; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors | 2003 |
A p38 inhibitor allows to dissociate differentiation and apoptotic processes triggered upon LIF withdrawal in mouse embryonic stem cells.
Topics: Animals; Apoptosis; Blotting, Western; Caspases; Cell Differentiation; Cell Survival; Cells, Cultured; Clone Cells; Culture Media; Enzyme Activation; Enzyme Inhibitors; Flow Cytometry; Gene Expression Profiling; Gene Expression Regulation; Green Fluorescent Proteins; Imidazoles; Interleukin-6; Leukemia Inhibitory Factor; Luminescent Proteins; Mice; Mitogen-Activated Protein Kinases; Models, Biological; Proto-Oncogene Proteins c-bcl-2; Pyridines; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; Stem Cells | 2004 |
Interleukin (IL)-17 enhances tumor necrosis factor-alpha-stimulated IL-6 synthesis via p38 mitogen-activated protein kinase in osteoblasts.
Topics: Animals; Anisomycin; Cell Line; Dose-Response Relationship, Drug; Imidazoles; Interleukin-17; Interleukin-6; Lysophospholipids; Mice; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Sphingosine; Tumor Necrosis Factor-alpha | 2004 |
Vasopressin phosphorylates HSP27 in aortic smooth muscle cells.
Topics: Animals; Aorta; Arginine Vasopressin; Heat-Shock Proteins; Imidazoles; Muscle, Smooth, Vascular; Phosphorylation; Pyridines; Rats; Rats, Wistar | 2004 |
Kinetic studies of small molecule interactions with protein kinases using biosensor technology.
Topics: Binding Sites; Biosensing Techniques; Buffers; Enzymes, Immobilized; Imidazoles; Kinetics; Protein Kinase Inhibitors; Protein Kinases; Pyridines; Pyrimidines; Substrate Specificity; Surface Plasmon Resonance | 2005 |
Akt regulates thrombin-induced HSP27 phosphorylation in aortic smooth muscle cells: function at a point downstream from p38 MAP kinase.
Topics: Adenylyl Cyclases; Animals; Aorta; Bucladesine; Cells, Cultured; Colforsin; Cyclic AMP; Heat-Shock Proteins; Imidazoles; Muscle, Smooth, Vascular; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Rats; Thrombin | 2005 |
Midazolam suppresses thrombin-induced heat shock protein 27 phosphorylation through inhibition of p38 mitogen-activated protein kinase in cardiac myocytes.
Topics: Anesthetics, Intravenous; Animals; Heat-Shock Proteins; Imidazoles; JNK Mitogen-Activated Protein Kinases; Mice; Midazolam; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocytes, Cardiac; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Thrombin | 2005 |
Intrinsically active variants of all human p38 isoforms.
Topics: Amino Acid Sequence; Enzyme Inhibitors; Humans; Imidazoles; Kinetics; Models, Molecular; Molecular Sequence Data; Mutation; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Conformation; Protein Isoforms; Pyridines; Substrate Specificity | 2007 |
Endotoxin-induced activation of equine platelets: evidence for direct activation of p38 MAPK pathways and vasoactive mediator production.
Topics: Animals; Blood Platelets; Dose-Response Relationship, Drug; Endotoxemia; Endotoxins; Enzyme Inhibitors; Female; Horse Diseases; Horses; Imidazoles; Leukocytes; Male; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Platelet Activation; Pyridines; Signal Transduction; Thromboxane A2 | 2007 |
Endotoxin-induced activation of equine digital vein endothelial cells: role of p38 MAPK.
Topics: Animals; Cell Adhesion; Cells, Cultured; Endothelial Cells; Enzyme Inhibitors; Epoprostenol; Hoof and Claw; Horses; Imidazoles; Lipopolysaccharides; Neutrophils; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Veins | 2009 |
ES936 stimulates DNA synthesis in HeLa cells independently on NAD(P)H:quinone oxidoreductase 1 inhibition, through a mechanism involving p38 MAPK.
Topics: 3T3 Cells; Ambroxol; Animals; Caco-2 Cells; Cell Cycle; DNA; Enzyme Inhibitors; ErbB Receptors; Free Radical Scavengers; HeLa Cells; Humans; Imidazoles; Indolequinones; Kinetics; Mice; NAD(P)H Dehydrogenase (Quinone); p38 Mitogen-Activated Protein Kinases; Pyridines; Pyruvic Acid; Reactive Oxygen Species; RNA, Small Interfering | 2010 |
Vitamin A (retinol) downregulates the receptor for advanced glycation endproducts (RAGE) by oxidant-dependent activation of p38 MAPK and NF-kB in human lung cancer A549 cells.
Topics: alpha-Tocopherol; Antioxidants; Cell Line, Tumor; Down-Regulation; Humans; Imidazoles; Lung Neoplasms; Mitogen-Activated Protein Kinase 11; Mitogen-Activated Protein Kinase 14; NF-kappa B; Oxidation-Reduction; p38 Mitogen-Activated Protein Kinases; Peptides; Phosphorylation; Pyridines; Receptor for Advanced Glycation End Products; Receptors, Immunologic; RNA Interference; RNA, Small Interfering; Signal Transduction; Transcription Factor RelA; Vitamin A | 2013 |
A Role for p38 Mitogen-activated Protein Kinase-mediated Threonine 30-dependent Norepinephrine Transporter Regulation in Cocaine Sensitization and Conditioned Place Preference.
Topics: Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Psychological; Gene Products, tat; Imidazoles; Male; Mice; Mice, Inbred C57BL; Motor Activity; Norepinephrine Plasma Membrane Transport Proteins; Nucleus Accumbens; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Prefrontal Cortex; Protein Kinase Inhibitors; Pyridines; Synaptosomes; Threonine; Up-Regulation | 2015 |
Cell-permeable p38 MAP kinase protects adult hippocampal neurons from cell death.
Topics: Animals; Cell Death; Cells, Cultured; Hippocampus; Hypoglycemia; Imidazoles; Mice; Neurons; Neuroprotection; p38 Mitogen-Activated Protein Kinases; Pyridines | 2019 |