Page last updated: 2024-09-05

sb 203580 and nifedipine

sb 203580 has been researched along with nifedipine in 4 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(nifedipine)
Trials
(nifedipine)
Recent Studies (post-2010) (nifedipine)
3,48941,13716,0242,4961,505

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)nifedipine (IC50)
perilipin-5Homo sapiens (human)7.133
perilipin-1Homo sapiens (human)9.619
1-acylglycerol-3-phosphate O-acyltransferase ABHD5 isoform aHomo sapiens (human)8.376
Voltage-dependent L-type calcium channel subunit alpha-1CCavia porcellus (domestic guinea pig)0.0429
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)0.035
Cytochrome P450 1A2Homo sapiens (human)0.3
Cytochrome P450 3A4Homo sapiens (human)10
Adenosine receptor A3Homo sapiens (human)7.214
Cytochrome P450 2C9 Homo sapiens (human)3.06
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)10
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.214
Voltage-dependent L-type calcium channel subunit alpha-1CRattus norvegicus (Norway rat)0.0385
Potassium voltage-gated channel subfamily A member 5Homo sapiens (human)6.1
3-oxo-5-alpha-steroid 4-dehydrogenase 1 Rattus norvegicus (Norway rat)1.12
Adenosine receptor A1Homo sapiens (human)7.701
3-oxo-5-alpha-steroid 4-dehydrogenase 2Rattus norvegicus (Norway rat)1.12
C-C chemokine receptor type 2Homo sapiens (human)2.191
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.214
Cytochrome P450 2J2Homo sapiens (human)3.06
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)0.4733
Voltage-dependent L-type calcium channel subunit alpha-1CMus musculus (house mouse)1.2
Voltage-dependent L-type calcium channel subunit alpha-1SMus musculus (house mouse)1.2
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)0.035
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)0.0394
Myosin light chain kinase, smooth muscleHomo sapiens (human)2.02
Potassium channel subfamily K member 2 Bos taurus (cattle)8.2
Indoleamine 2,3-dioxygenase 2Mus musculus (house mouse)1.5
Voltage-dependent L-type calcium channel subunit alpha-1DMus musculus (house mouse)1.2
Voltage-dependent L-type calcium channel subunit alpha-1FMus musculus (house mouse)1.2

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's3 (75.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Akiyama-Uchida, Y; Ashizawa, N; Kikuchi, H; Ohtsuru, A; Seto, S; Tsukazaki, T; Yamashita, S; Yano, K1
Liu, S; Sun, C; Wang, L; Yan, J1
Campos-Toimil, M; Cuíñas, A; Elíes, J; Orallo, F1
Choi, NK; Hwang, YC; Jung, JY; Kim, SH; Kim, SM; Kim, WJ; Lim, HS; Woo, SM1

Other Studies

4 other study(ies) available for sb 203580 and nifedipine

ArticleYear
Norepinephrine enhances fibrosis mediated by TGF-beta in cardiac fibroblasts.
    Hypertension (Dallas, Tex. : 1979), 2002, Volume: 40, Issue:2

    Topics: Activating Transcription Factor 2; Animals; Animals, Newborn; Blotting, Western; Cell Division; Collagen Type I; Cyclic AMP Response Element-Binding Protein; Drug Synergism; Female; Fibroblasts; Fibronectins; Fibrosis; Flavonoids; Humans; Imidazoles; Luciferases; Myocardium; Nifedipine; Norepinephrine; Phosphorylation; Plasminogen Activator Inhibitor 1; Pregnancy; Pyridines; Rats; Rats, Sprague-Dawley; Recombinant Fusion Proteins; Transcription Factors; Transforming Growth Factor beta; Transforming Growth Factor beta1; Tumor Cells, Cultured

2002
Calcium ameliorates obesity induced by high-fat diet and its potential correlation with p38 MAPK pathway.
    Molecular biology reports, 2012, Volume: 39, Issue:2

    Topics: Adipogenesis; Animals; Calcium, Dietary; Cholesterol; Diet, High-Fat; Gene Expression Regulation; Imidazoles; Male; MAP Kinase Signaling System; Mice; Nifedipine; Obesity; Pyridines; Real-Time Polymerase Chain Reaction; Triglycerides; Weight Gain

2012
Cyclic AMP relaxation of rat aortic smooth muscle is mediated in part by decrease of depletion of intracellular Ca(2+) stores and inhibition of capacitative calcium entry.
    Vascular pharmacology, 2013, Volume: 58, Issue:1-2

    Topics: Animals; Aorta, Thoracic; Calcium; Colforsin; Cyclic AMP; Imidazoles; Male; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nifedipine; p38 Mitogen-Activated Protein Kinases; Phenylephrine; Phosphodiesterase 4 Inhibitors; Pyridines; Rats; Rats, Inbred WKY; Rolipram; Vasodilation; Vasodilator Agents; Verapamil

2013
Effect of nifedipine on the differentiation of human dental pulp cells cultured with mineral trioxide aggregate.
    Journal of endodontics, 2013, Volume: 39, Issue:6

    Topics: Adult; Aluminum Compounds; Anthracenes; Butadienes; Calcium; Calcium Channel Blockers; Calcium Compounds; Cell Culture Techniques; Cell Differentiation; Cell Proliferation; Cells, Cultured; Culture Media; Dental Pulp; Drug Combinations; Extracellular Matrix Proteins; Extracellular Signal-Regulated MAP Kinases; Humans; Imidazoles; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinases; Nifedipine; Nitriles; Odontoblasts; Oxides; p38 Mitogen-Activated Protein Kinases; Phosphoproteins; Pyridines; Root Canal Filling Materials; Sialoglycoproteins; Silicates; Tooth Calcification

2013