Page last updated: 2024-09-05

sb 203580 and minocycline

sb 203580 has been researched along with minocycline in 14 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(minocycline)
Trials
(minocycline)
Recent Studies (post-2010) (minocycline)
3,48941,1376,5795022,921

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)minocycline (IC50)
Multidrug transporter MdfAEscherichia coli K-122.6

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (35.71)29.6817
2010's8 (57.14)24.3611
2020's1 (7.14)2.80

Authors

AuthorsStudies
Fiebich, BL; Goldsteins, G; Keinanen, R; Koistinaho, J; Tikka, T1
Bales, KR; Bymaster, FP; Chernet, E; Dodel, RC; Du, Y; Gao, F; Lin, S; Luecke, S; Ma, Z; Nelson, DL; Paul, SM; Perry, KW; Phebus, LA; Triarhou, LC1
Bhat, NR; Guo, G1
Bradesi, S; Mayer, EA; Pothoulakis, C; Steinauer, J; Svensson, CI; Yaksh, TL1
Ito, N; Obata, H; Saito, S1
Chen, FY; Chen, Y; Cui, Y; Li, YY; Liu, XG; Na, XD; Wei, XH; Xin, WJ; Zhang, XQ1
Ahn, DK; Bae, YC; Ju, JS; Kang, YM; Lee, MK; Park, MK; Won, KA1
Lyons, D; Ma, F; Westlund, KN; Zhang, L1
Ho, I; Kotani, J; Mei, XP; Sakuma, Y; Wu, D; Xie, C; Xu, LX1
Chen, C; Meng, QX; Qi, J; Wu, H; Wu, Y; Zhao, TB1
Chen, CH; Chen, NF; Chen, WF; Feng, CW; Huang, SY; Sung, CS; Wen, ZH; Wong, CS1
Domoto, R; Kawabata, A; Nakashima, K; Nishibori, M; Sekiguchi, F; Tsubota, M; Wake, H; Yamanishi, H; Yamasoba, D1
Beggs, S; Moriarty, O; Salter, MW; Sengar, AS; Tu, Y; Walker, SM1
Gao, F; Jia, X; Li, Z; Peng, X; Tian, X; Zhang, A1

Other Studies

14 other study(ies) available for sb 203580 and minocycline

ArticleYear
Minocycline, a tetracycline derivative, is neuroprotective against excitotoxicity by inhibiting activation and proliferation of microglia.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, Apr-15, Volume: 21, Issue:8

    Topics: Animals; Anti-Bacterial Agents; Cell Death; Cell Division; Cell Survival; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acids; Glutamic Acid; Hydro-Lyases; Imidazoles; Kainic Acid; Microglia; Minocycline; Mitogen-Activated Protein Kinases; Neuroprotective Agents; p38 Mitogen-Activated Protein Kinases; Pyridines; Rats; Rats, Wistar; Spinal Cord

2001
Minocycline prevents nigrostriatal dopaminergic neurodegeneration in the MPTP model of Parkinson's disease.
    Proceedings of the National Academy of Sciences of the United States of America, 2001, Dec-04, Volume: 98, Issue:25

    Topics: Animals; Caspase 1; Cells, Cultured; Dopamine; Humans; Imidazoles; Male; Mice; Mice, Inbred C57BL; Minocycline; Mitogen-Activated Protein Kinases; Monoamine Oxidase; MPTP Poisoning; Nerve Degeneration; Neurons; Neuroprotective Agents; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; p38 Mitogen-Activated Protein Kinases; Parkinsonian Disorders; Phosphorylation; Pyridines; Visual Cortex

2001
p38alpha MAP kinase mediates hypoxia-induced motor neuron cell death: a potential target of minocycline's neuroprotective action.
    Neurochemical research, 2007, Volume: 32, Issue:12

    Topics: Anti-Bacterial Agents; Blotting, Western; Cell Death; Cell Hypoxia; Cell Line; Cells, Cultured; Enzyme Inhibitors; Flow Cytometry; Glucose; Humans; Imidazoles; L-Lactate Dehydrogenase; Minocycline; Motor Neurons; Neuroprotective Agents; p38 Mitogen-Activated Protein Kinases; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Small Interfering

2007
Role of spinal microglia in visceral hyperalgesia and NK1R up-regulation in a rat model of chronic stress.
    Gastroenterology, 2009, Volume: 136, Issue:4

    Topics: Animals; Disease Models, Animal; Enzyme Inhibitors; Hyperalgesia; Imidazoles; Male; Microglia; Minocycline; p38 Mitogen-Activated Protein Kinases; Pyridines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Spinal Nerves; Stress, Physiological; Up-Regulation; Viscera; Water Deprivation

2009
Spinal microglial expression and mechanical hypersensitivity in a postoperative pain model: comparison with a neuropathic pain model.
    Anesthesiology, 2009, Volume: 111, Issue:3

    Topics: Animals; Anti-Bacterial Agents; Behavior, Animal; CD11b Antigen; Enzyme Inhibitors; Fluorescent Antibody Technique; Hyperalgesia; Imidazoles; Immunohistochemistry; Male; Microglia; Minocycline; p38 Mitogen-Activated Protein Kinases; Pain; Pain, Postoperative; Peripheral Nervous System Diseases; Pyridines; Rats; Rats, Sprague-Dawley; Spinal Cord; Spinal Nerves

2009
Activation of p38 signaling in the microglia in the nucleus accumbens contributes to the acquisition and maintenance of morphine-induced conditioned place preference.
    Brain, behavior, and immunity, 2012, Volume: 26, Issue:2

    Topics: Animals; Conditioning, Operant; Enzyme Activation; Imidazoles; Male; Microglia; Minocycline; Morphine; Nucleus Accumbens; p38 Mitogen-Activated Protein Kinases; Pyridines; Rats; Rats, Sprague-Dawley; Signal Transduction

2012
Participation of microglial p38 MAPK in formalin-induced temporomandibular joint nociception in rats.
    Journal of orofacial pain, 2012,Spring, Volume: 26, Issue:2

    Topics: Analysis of Variance; Animals; Arthralgia; Cisterna Magna; Endpoint Determination; Formaldehyde; Imidazoles; Injections, Intra-Articular; Male; Microglia; Minocycline; Motor Activity; Nociception; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Posterior Horn Cells; Protease Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley; Temporomandibular Joint; Temporomandibular Joint Disorders

2012
Orofacial neuropathic pain mouse model induced by Trigeminal Inflammatory Compression (TIC) of the infraorbital nerve.
    Molecular brain, 2012, Dec-28, Volume: 5

    Topics: Animals; Behavior, Animal; Disease Models, Animal; Facial Pain; Hyperalgesia; Imidazoles; Inflammation; Male; Mice; Mice, Inbred C57BL; Microglia; Minocycline; Nerve Compression Syndromes; Neuralgia; Neurons; Orbit; p38 Mitogen-Activated Protein Kinases; Purinergic P2X Receptor Antagonists; Pyridines; Tetrazoles; Trigeminal Ganglion; Trigeminal Nerve; Trigeminal Neuralgia; Trigeminal Nucleus, Spinal

2012
Depressing interleukin-1β contributed to the synergistic effects of tramadol and minocycline on spinal nerve ligation-induced neuropathic pain.
    Neuro-Signals, 2014, Volume: 22, Issue:1

    Topics: Analgesics; Animals; Antibodies; Drug Combinations; Hyperalgesia; Imidazoles; Interleukin-1beta; Ligation; Male; Microglia; Minocycline; Neuralgia; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Posterior Horn Cells; Pyridines; Rats, Sprague-Dawley; Rotarod Performance Test; Signal Transduction; Spinal Nerves; Tramadol

2014
Crosstalk between Activated Microglia and Neurons in the Spinal Dorsal Horn Contributes to Stress-induced Hyperalgesia.
    Scientific reports, 2016, 12-20, Volume: 6

    Topics: Animals; Genes, fos; Hyperalgesia; Imidazoles; Interleukin-6; Male; Microglia; Minocycline; Neurons; Pain; Pain Threshold; Pyridines; Rats; Rats, Sprague-Dawley; Spinal Cord; Spinal Cord Dorsal Horn; Stress, Physiological

2016
Potentiation of spinal glutamatergic response in the neuron-glia interactions underlies the intrathecal IL-1β-induced thermal hyperalgesia in rats.
    CNS neuroscience & therapeutics, 2017, Volume: 23, Issue:7

    Topics: Animals; Disease Models, Animal; Dizocilpine Maleate; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glutamate Plasma Membrane Transport Proteins; Glutamic Acid; Hot Temperature; Hyperalgesia; Imidazoles; Interleukin-1beta; Male; Microglia; Minocycline; Neurons; Nitric Oxide; Nociceptive Pain; Phosphorylation; Pyridines; Random Allocation; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Spinal Cord

2017
Paclitaxel-induced HMGB1 release from macrophages and its implication for peripheral neuropathy in mice: Evidence for a neuroimmune crosstalk.
    Neuropharmacology, 2018, Volume: 141

    Topics: Acetylcysteine; Animals; Antibodies; Cells, Cultured; Clodronic Acid; Coculture Techniques; Ganglia, Spinal; HMGB1 Protein; Hyperalgesia; Imidazoles; Macrophages; Male; Membrane Proteins; Mice; Minocycline; Neurons; p300-CBP Transcription Factors; Paclitaxel; Peripheral Nervous System Diseases; Phosphoproteins; Phosphorylation; Proline; Pyridines; Pyruvates; Reactive Oxygen Species; Receptor for Advanced Glycation End Products; Receptors, CXCR4; Recombinant Proteins; Sciatic Nerve; Thiocarbamates; Thrombomodulin; Up-Regulation

2018
Priming of Adult Incision Response by Early-Life Injury: Neonatal Microglial Inhibition Has Persistent But Sexually Dimorphic Effects in Adult Rats.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2019, 04-17, Volume: 39, Issue:16

    Topics: Animals; Enzyme Inhibitors; Female; Hyperalgesia; Imidazoles; Interferon Regulatory Factors; Male; Microglia; Minocycline; Neurons; Pain; Pain Threshold; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Sex Factors; Spinal Cord

2019
Activation of spinal PDGFRβ in microglia promotes neuronal autophagy via p38 MAPK pathway in morphine-tolerant rats.
    Journal of neurochemistry, 2021, Volume: 158, Issue:2

    Topics: Adenine; Animals; Autophagy; Drug Tolerance; Imatinib Mesylate; Imidazoles; Injections, Spinal; Male; MAP Kinase Signaling System; Microglia; Minocycline; Morphine; Narcotics; Neurons; p38 Mitogen-Activated Protein Kinases; Pain Measurement; Protein Kinase Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Platelet-Derived Growth Factor beta

2021