Page last updated: 2024-09-05

sb 203580 and mifepristone

sb 203580 has been researched along with mifepristone in 3 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(mifepristone)
Trials
(mifepristone)
Recent Studies (post-2010) (mifepristone)
3,48941,1376,5365951,758

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)mifepristone (IC50)
Glucocorticoid receptor Canis lupus familiaris (dog)0.0264
Bile salt export pumpHomo sapiens (human)2.02
Estrogen receptorHomo sapiens (human)4.311
Glucocorticoid receptorHomo sapiens (human)0.0249
Prostaglandin G/H synthase 1Ovis aries (sheep)0.0003
Progesterone receptorHomo sapiens (human)0.1347
Glucocorticoid receptorRattus norvegicus (Norway rat)0.774
Glucocorticoid receptorMus musculus (house mouse)0.0022
Glycine receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0022
Mineralocorticoid receptor Homo sapiens (human)2.0938
Cytochrome P450 3A4Homo sapiens (human)9.5
Coagulation factor VIIHomo sapiens (human)0.0003
Androgen receptorHomo sapiens (human)0.2988
Cytochrome P450 2C8Homo sapiens (human)1.5
Cytochrome P450 2C9 Homo sapiens (human)4.9
Steroid 17-alpha-hydroxylase/17,20 lyase Rattus norvegicus (Norway rat)0.0016
Polyunsaturated fatty acid lipoxygenase ALOX15Oryctolagus cuniculus (rabbit)0.555
Tissue factorHomo sapiens (human)0.0003
Androgen receptorRattus norvegicus (Norway rat)0.0083
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0014
Glycine receptor subunit betaRattus norvegicus (Norway rat)0.0022
Glycine receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0022
Prostaglandin G/H synthase 1Homo sapiens (human)0.0078
Glycine receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0022
Substance-P receptorCavia porcellus (domestic guinea pig)0.0015
Mu-type opioid receptorHomo sapiens (human)2.457
Estrogen receptor betaHomo sapiens (human)1.528
Glucocorticoid receptorSus scrofa (pig)0.0153

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, YP; Luo, Y; Rui, HL1
Chen, Y; Feng, C; Xiao, L1
Harada, H; Heidari, N; Hicks, MA; Marking, CB; Miller, AV1

Other Studies

3 other study(ies) available for sb 203580 and mifepristone

ArticleYear
[The role of MAPK/ERK1/2 signaling pathway in aldosterone stimulated transforming growth factor-beta1 synthesis in renal tubular epithelial cells].
    Zhonghua yi xue za zhi, 2006, Nov-28, Volume: 86, Issue:44

    Topics: Aldosterone; Anthracenes; Blotting, Western; Butadienes; Cells, Cultured; Dose-Response Relationship, Drug; Epithelial Cells; Extracellular Signal-Regulated MAP Kinases; Humans; Imidazoles; Kidney Tubules, Proximal; Mifepristone; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Nitriles; Phosphorylation; Pyridines; Signal Transduction; Time Factors; Transforming Growth Factor beta1

2006
Glucocorticoid rapidly enhances NMDA-evoked neurotoxicity by attenuating the NR2A-containing NMDA receptor-mediated ERK1/2 activation.
    Molecular endocrinology (Baltimore, Md.), 2010, Volume: 24, Issue:3

    Topics: Animals; Blotting, Western; Calcium; Cells, Cultured; Enzyme Inhibitors; Flavonoids; Glucocorticoids; Hippocampus; Imidazoles; Mifepristone; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; N-Methylaspartate; Neurons; p38 Mitogen-Activated Protein Kinases; Pyridines; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

2010
Glucocorticoid-mediated BIM induction and apoptosis are regulated by Runx2 and c-Jun in leukemia cells.
    Cell death & disease, 2012, Jul-19, Volume: 3

    Topics: Apoptosis; Apoptosis Regulatory Proteins; Bcl-2-Like Protein 11; Binding Sites; Cell Line, Tumor; Core Binding Factor Alpha 1 Subunit; Dexamethasone; Glucocorticoids; HEK293 Cells; Humans; Imidazoles; JNK Mitogen-Activated Protein Kinases; Jurkat Cells; Membrane Proteins; Mifepristone; p38 Mitogen-Activated Protein Kinases; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Promoter Regions, Genetic; Protein Kinase Inhibitors; Proto-Oncogene Proteins; Pyridines; Receptors, Glucocorticoid; RNA Interference; RNA, Small Interfering; Signal Transduction; Transcription Factor AP-1

2012