Page last updated: 2024-09-05

sb 203580 and l 365260

sb 203580 has been researched along with l 365260 in 2 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(l 365260)
Trials
(l 365260)
Recent Studies (post-2010) (l 365260)
3,48941,137422108

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)l 365260 (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0081
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0081
Cholecystokinin receptor type ARattus norvegicus (Norway rat)0.4981
Gastrin/cholecystokinin type B receptorRattus norvegicus (Norway rat)0.039
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0081
Histamine H1 receptorCavia porcellus (domestic guinea pig)5
Cholecystokinin receptor type AHomo sapiens (human)0.1585
Gastrin/cholecystokinin type B receptorHomo sapiens (human)0.0079
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5
Cholecystokinin receptor type ACavia porcellus (domestic guinea pig)0.044
Cysteinyl leukotriene receptor 2Homo sapiens (human)5
Cysteinyl leukotriene receptor 1Homo sapiens (human)5

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bergé, G; Carnazzi, E; Gagne, D; Galleyrand, JC; Ibarz, G; Martinez, J; Morel, C; Oiry, C1
Cao, J; Luo, HS; Ming, M; Song, WC; Yu, HG; Yu, JP; Zhou, YH1

Other Studies

2 other study(ies) available for sb 203580 and l 365260

ArticleYear
Cross-interactions of two p38 mitogen-activated protein (MAP) kinase inhibitors and two cholecystokinin (CCK) receptor antagonists with the CCK1 receptor and p38 MAP kinase.
    The Journal of biological chemistry, 2005, Jun-03, Volume: 280, Issue:22

    Topics: Adenosine Triphosphate; Animals; Benzodiazepinones; Binding Sites; Blotting, Western; COS Cells; Devazepide; Dose-Response Relationship, Drug; Enzyme Inhibitors; Genes, Reporter; Hormone Antagonists; Imidazoles; Immunoblotting; Inositol Phosphates; Kinetics; Ligands; MAP Kinase Signaling System; Models, Chemical; Models, Molecular; p38 Mitogen-Activated Protein Kinases; Phenylurea Compounds; Protein Binding; Protein Conformation; Pyridines; Rats; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Signal Transduction; Time Factors; Transfection

2005
[The role of p38 MAPK in gastrin-induced u-PA expression in human colon cancer cells].
    Zhonghua zhong liu za zhi [Chinese journal of oncology], 2007, Volume: 29, Issue:1

    Topics: Benzodiazepinones; Blotting, Western; Cell Line, Tumor; Colonic Neoplasms; Gastrins; Gene Expression Regulation, Neoplastic; Genetic Vectors; Humans; Imidazoles; p38 Mitogen-Activated Protein Kinases; Phenylurea Compounds; Phosphorylation; Pyridines; Receptor, Cholecystokinin B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Transfection; Urokinase-Type Plasminogen Activator

2007