Page last updated: 2024-09-05

sb 203580 and glycine

sb 203580 has been researched along with glycine in 6 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(glycine)
Trials
(glycine)
Recent Studies (post-2010) (glycine)
3,48941,13735,1637568,415

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)glycine (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)1.4852
Sodium- and chloride-dependent glycine transporter 1Homo sapiens (human)106
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.3253
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.3253
Sodium- and chloride-dependent glycine transporter 2Homo sapiens (human)128

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (66.67)29.6817
2010's1 (16.67)24.3611
2020's1 (16.67)2.80

Authors

AuthorsStudies
Becker, JW; Cameron, PM; Fitzgerald, CE; O'Keefe, SJ; Patel, SB; Pikounis, VB; Scapin, G; Zaller, D1
Anwyl, R; Gisabella, B; Rowan, MJ1
Chalothorn, D; Faber, JE; Jackson, LF; Lee, DC; Zhang, H1
Clay, WC; Condreay, JP; Hall, M; Holbrook, J; Livermore, D; Michel, AD; Ng, SW; Roman, S; Senger, S; Thompson, K1
Chen, Q; Fan, L; He, Z; Jiang, L; Liu, L; Lu, Y; Qin, X; Zhong, X1
Ameen, M; Arthur Ataam, J; Bharucha, N; Bruyneel, AAN; Diecke, S; Feyen, DAM; Furihata, T; Gavidia, AA; Karakikes, I; Kaur, B; Lim, EW; Martinez-Amador, N; Mercola, M; Metallo, CM; Monte, E; Nair, P; Perea-Gil, I; Seeger, T; Serrano, R; Snyder, MP; Termglinchan, V; Vadgama, N1

Other Studies

6 other study(ies) available for sb 203580 and glycine

ArticleYear
Structural basis for p38alpha MAP kinase quinazolinone and pyridol-pyrimidine inhibitor specificity.
    Nature structural biology, 2003, Volume: 10, Issue:9

    Topics: Amino Acid Sequence; Animals; Cloning, Molecular; Enzyme Inhibitors; Glycine; Imidazoles; Inhibitory Concentration 50; Kinetics; Mice; Mitogen-Activated Protein Kinase 14; Mitogen-Activated Protein Kinases; Models, Chemical; Models, Molecular; Molecular Sequence Data; Mutation; Peptides; Protein Binding; Protein Isoforms; Protein Structure, Tertiary; Pyridazines; Pyridines; Pyrimidines; Quinazolines; Sequence Homology, Amino Acid

2003
Mechanisms underlying the inhibition of long-term potentiation by preconditioning stimulation in the hippocampus in vitro.
    Neuroscience, 2003, Volume: 121, Issue:2

    Topics: Animals; Anticonvulsants; Cyclopropanes; Electric Stimulation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Flavonoids; Glycine; Hippocampus; Imidazoles; In Vitro Techniques; Long-Term Potentiation; Male; Methoxyhydroxyphenylglycol; Neural Inhibition; Pyridines; Rats; Rats, Wistar; Synapses; Time Factors

2003
Transactivation of epidermal growth factor receptor mediates catecholamine-induced growth of vascular smooth muscle.
    Circulation research, 2004, Nov-12, Volume: 95, Issue:10

    Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Anthracenes; Aorta, Thoracic; Bacterial Proteins; Benzopyrans; Butadienes; Catheterization; Cell Division; Dipeptides; ErbB Receptors; Flavonoids; Glycine; Hydroxamic Acids; Imidazoles; MAP Kinase Kinase 1; MAP Kinase Kinase 2; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nitriles; Organ Culture Techniques; Phenylephrine; Phosphorylation; Protein Processing, Post-Translational; Pyridines; Quinazolines; Rats; Receptors, Adrenergic, alpha-1; Thrombin; Tyrphostins

2004
Identification of regions of the P2X(7) receptor that contribute to human and rat species differences in antagonist effects.
    British journal of pharmacology, 2008, Volume: 155, Issue:5

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Allosteric Regulation; Allosteric Site; Amino Acid Sequence; Animals; Cell Line; Cloning, Molecular; Dose-Response Relationship, Drug; Glycine; Humans; Imidazoles; Molecular Sequence Data; Mutagenesis, Site-Directed; Piperazines; Plasmids; Polymorphism, Single Nucleotide; Protein Binding; Protein Structure, Tertiary; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Pyridines; Pyridoxal Phosphate; Radioligand Assay; Rats; Receptors, Purinergic P2; Receptors, Purinergic P2X7; Sequence Alignment; Species Specificity; Transfection

2008
Glycine-induced cytoprotection is mediated by ERK1/2 and AKT in renal cells with ATP depletion.
    European journal of cell biology, 2011, Volume: 90, Issue:4

    Topics: Adenosine Triphosphate; Animals; Cell Death; Cytoprotection; Dogs; Glycine; HEK293 Cells; Humans; Imidazoles; Kidney; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Proto-Oncogene Proteins c-akt; Pyridines; Receptors, Glycine; Signal Transduction

2011
Serine biosynthesis as a novel therapeutic target for dilated cardiomyopathy.
    European heart journal, 2022, 09-21, Volume: 43, Issue:36

    Topics: Activating Transcription Factor 4; Adenosine Triphosphate; Anti-Inflammatory Agents, Non-Steroidal; Carbazoles; Cardiomyopathy, Dilated; Drug Evaluation, Preclinical; Glucose; Glycine; Humans; Imidazoles; Induced Pluripotent Stem Cells; Molecular Targeted Therapy; Mutation; Myocytes, Cardiac; Phosphoglycerate Dehydrogenase; Protein Kinase Inhibitors; Pyridines; Serine; Troponin T

2022