Page last updated: 2024-09-05

sb 203580 and gdc-0068

sb 203580 has been researched along with gdc-0068 in 1 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(gdc-0068)
Trials
(gdc-0068)
Recent Studies (post-2010) (gdc-0068)
3,48941,137621760

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)gdc-0068 (IC50)
Cytochrome P450 2D6Homo sapiens (human)0.157
RAC-alpha serine/threonine-protein kinaseHomo sapiens (human)0.0418
RAC-beta serine/threonine-protein kinaseHomo sapiens (human)0.0255
cGMP-dependent protein kinase 1 Homo sapiens (human)0.0835
RAC-gamma serine/threonine-protein kinaseHomo sapiens (human)0.0187

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hamilton, BJ; Stan, RV; Tse, D1

Other Studies

1 other study(ies) available for sb 203580 and gdc-0068

ArticleYear
Phorbol esters induce PLVAP expression via VEGF and additional secreted molecules in MEK1-dependent and p38, JNK and PI3K/Akt-independent manner.
    Journal of cellular and molecular medicine, 2019, Volume: 23, Issue:2

    Topics: Anthracenes; Autocrine Communication; Axitinib; Butadienes; Flavonoids; Gene Expression Regulation; Human Umbilical Vein Endothelial Cells; Humans; Imidazoles; Indazoles; MAP Kinase Kinase 1; MAP Kinase Kinase 4; Membrane Proteins; Nitriles; Phosphatidylinositol 3-Kinases; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Pyridines; Pyrimidines; RNA, Small Interfering; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factor Receptor-2

2019