Page last updated: 2024-09-05

sb 203580 and dinaciclib

sb 203580 has been researched along with dinaciclib in 4 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(dinaciclib)
Trials
(dinaciclib)
Recent Studies (post-2010) (dinaciclib)
3,48941,13713312129

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)dinaciclib (IC50)
Cyclin-T1Homo sapiens (human)0.0272
Cyclin-KHomo sapiens (human)0.0227
Cyclin-dependent kinase 1Homo sapiens (human)0.0162
Cyclin-dependent kinase 4Homo sapiens (human)0.0742
G2/mitotic-specific cyclin-B1Homo sapiens (human)0.049
Cyclin-A2Homo sapiens (human)0.002
G1/S-specific cyclin-D1Homo sapiens (human)0.119
G1/S-specific cyclin-E1Homo sapiens (human)0.0028
Cyclin-dependent kinase 2Homo sapiens (human)0.0074
Aldo-keto reductase family 1 member C3Homo sapiens (human)0.23
Cyclin-dependent kinase 8Homo sapiens (human)0.0039
Glycogen synthase kinase-3 alphaHomo sapiens (human)0.414
Glycogen synthase kinase-3 betaHomo sapiens (human)0.324
Cyclin-dependent kinase 7Homo sapiens (human)0.1273
Cyclin-dependent kinase 9Homo sapiens (human)0.0227
Cyclin-HHomo sapiens (human)0.17
CDK-activating kinase assembly factor MAT1Homo sapiens (human)0.17
Cyclin-A1Homo sapiens (human)0.003
Cyclin-dependent-like kinase 5 Homo sapiens (human)0.011
Heat shock factor protein 1Homo sapiens (human)0.007
Cyclin-dependent kinase 13Homo sapiens (human)0.021
Cyclin-dependent kinase 5 activator 1Homo sapiens (human)0.0219
Cyclin-dependent kinase 12Homo sapiens (human)0.0323

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (25.00)24.3611
2020's3 (75.00)2.80

Authors

AuthorsStudies
Munoz, L1
Bharate, SB; Raghuvanshi, R1
Caballero, E; García-Cárceles, J; Gil, C; Martínez, A1
Laufer, S; Pillaiyar, T1

Reviews

3 review(s) available for sb 203580 and dinaciclib

ArticleYear
Non-kinase targets of protein kinase inhibitors.
    Nature reviews. Drug discovery, 2017, Volume: 16, Issue:6

    Topics: Animals; Drug Design; Drug Evaluation, Preclinical; Humans; Molecular Targeted Therapy; Protein Kinase Inhibitors; Protein Kinases

2017
Kinase Inhibitors as Underexplored Antiviral Agents.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Animals; Antiviral Agents; Drug Repositioning; Humans; Protein Kinase Inhibitors; Virus Diseases; Viruses

2022
Kinases as Potential Therapeutic Targets for Anti-coronaviral Therapy.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Antiviral Agents; COVID-19; COVID-19 Drug Treatment; Humans; Protein Kinase Inhibitors; SARS-CoV-2; Signal Transduction; Virus Replication

2022

Other Studies

1 other study(ies) available for sb 203580 and dinaciclib

ArticleYear
Recent Developments in the Use of Kinase Inhibitors for Management of Viral Infections.
    Journal of medicinal chemistry, 2022, 01-27, Volume: 65, Issue:2

    Topics: Antiviral Agents; COVID-19; COVID-19 Drug Treatment; Drug Approval; Drug Repositioning; High-Throughput Screening Assays; Humans; Protein Kinase Inhibitors; SARS-CoV-2; United States; United States Food and Drug Administration; Virus Diseases

2022