Page last updated: 2024-09-05

sb 203580 and colforsin

sb 203580 has been researched along with colforsin in 25 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
3,48941,13713,460461,298

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (8.00)18.2507
2000's21 (84.00)29.6817
2010's2 (8.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burns, CJ; Howell, SL; Jones, PM; Persaud, SJ1
Brooks, DP; Francis, J; Nambi, P; Parameswaran, N; Pullen, M; Spielman, WS1
Hansen, TO; Nielsen, FC; Rehfeld, JF1
Lee, JK; Suh, HW; Won, JS1
Caivano, M; Cohen, P; Gorgoni, B; Poli, V1
Kandolf, R; Küpper, JH; Meyer, RG; Rodemann, HP1
Eisen, TG; Smalley, KS1
Gauldie, J; Howe, K; McKay, DM1
Coulonval, K; Dumont, JE; Lamy, F; Perpete, S; Vandeput, F1
Dhein, S; Hagendorff, A; Pfeiffer, D; Polontchouk, L; Salameh, A1
Damiano, N; Galdiero, E; Galdiero, M; Longanella, A; Tortora, A; Vitiello, M1
Itoh, M; Kakita, A; Miura, Y; Oiso, Y; Ono, Y; Suzuki, A1
Ishisaki, A; Kanno, Y; Kozawa, O; Nakajima, K; Numata, O; Shibata, T; Tokuda, H1
Egashira, K; Fukuyama, K; Ichiki, T; Iino, N; Masuda, S; Ono, H; Takeshita, A1
Hirade, K; Ishisaki, A; Kanno, Y; Katagiri, Y; Kitajima, Y; Kozawa, O; Matsuno, H; Nakajima, K; Shu, E; Suga, H1
Blondeau, JP; Corrèze, C; Pomérance, M1
Creaven, BS; Egan, DA; Finn, GJ1
Becker, TC; Cao, W; Collins, QF; Collins, S; Daniel, KW; Floering, L; Lupo, EG; Robidoux, J; Xiong, Y1
Blume, N; Friedrichsen, BN; Gram, VK; Lee, YC; Møldrup, A; Neubauer, N; Nielsen, JH; Petersen, JS1
Bhat, NR; Mohanty, SB; Zhang, P1
Hanada, K; Iwasaki, Y; Kageyama, K; Nigawara, T; Sakihara, S; Suda, T; Takayasu, S1
Caimmi, PP; Grossini, E; Mary, DA; Molinari, C; Ribichini, F; Uberti, F; Vacca, G1
Derebecka-Holysz, N; Holysz, M; Lehmann, TP; Trzeciak, WH1
Chetkovich, D; Golding, NL; Khurana, S; Lewis, AS; Liu, Z; Rosa, K1
Campos-Toimil, M; Cuíñas, A; Elíes, J; Orallo, F1

Other Studies

25 other study(ies) available for sb 203580 and colforsin

ArticleYear
The p38 mitogen-activated protein kinase cascade is not required for the stimulation of insulin secretion from rat islets of Langerhans.
    Molecular and cellular endocrinology, 1999, Feb-25, Volume: 148, Issue:1-2

    Topics: Animals; Arsenites; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cells, Cultured; Colforsin; Enzyme Inhibitors; Glucose; Homeostasis; Imidazoles; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Mitogen-Activated Protein Kinases; Okadaic Acid; p38 Mitogen-Activated Protein Kinases; Phosphoprotein Phosphatases; Pyridines; Rats; Rats, Sprague-Dawley; Signal Transduction; Sodium Compounds; Sorbitol; Tetradecanoylphorbol Acetate; Vanadates

1999
Mechanism of adrenomedullin-stimulated hyaluronic acid release in rat mesangial cells.
    European journal of pharmacology, 1999, Apr-16, Volume: 370, Issue:3

    Topics: Adrenomedullin; Animals; Bucladesine; Cell Culture Techniques; Colforsin; Drug Interactions; Enzyme Inhibitors; Glomerular Mesangium; Hyaluronic Acid; Imidazoles; Kidney Cortex; Male; Peptides; Phosphotransferases; Pyridines; Rats; Rats, Sprague-Dawley; Vasodilator Agents

1999
Cyclic AMP-induced neuronal differentiation via activation of p38 mitogen-activated protein kinase.
    Journal of neurochemistry, 2000, Volume: 75, Issue:5

    Topics: Animals; Cell Differentiation; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; Fibroblast Growth Factor 2; Genes, Dominant; Humans; Imidazoles; Mitogen-Activated Protein Kinases; Mutation; Neurites; Neurons; p38 Mitogen-Activated Protein Kinases; PC12 Cells; Phosphorylation; Pyridines; Rats; Signal Transduction; Transfection; Tumor Cells, Cultured

2000
Forskolin inhibits expression of inducible nitric oxide synthase mRNA via inhibiting the mitogen activated protein kinase in C6 cells.
    Brain research. Molecular brain research, 2001, Apr-18, Volume: 89, Issue:1-2

    Topics: Animals; Colforsin; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation, Enzymologic; Glioma; Imidazoles; Isoquinolines; Lipopolysaccharides; Mitogen-Activated Protein Kinases; NF-kappa B; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; p38 Mitogen-Activated Protein Kinases; Pyridines; Rats; RNA, Messenger; Sulfonamides; Transcription, Genetic; Tumor Cells, Cultured

2001
The induction of cyclooxygenase-2 mRNA in macrophages is biphasic and requires both CCAAT enhancer-binding protein beta (C/EBP beta ) and C/EBP delta transcription factors.
    The Journal of biological chemistry, 2001, Dec-28, Volume: 276, Issue:52

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Butadienes; CCAAT-Enhancer-Binding Proteins; Cell Fractionation; Cell Line; Colforsin; Cyclic AMP Response Element-Binding Protein; Cyclooxygenase 2; DNA; Enzyme Induction; Enzyme Inhibitors; Imidazoles; Isoenzymes; Lipopolysaccharides; Macrophage Activation; Macrophages; Mice; Models, Biological; NF-kappa B; Nitriles; Promoter Regions, Genetic; Prostaglandin-Endoperoxide Synthases; Protein Binding; Pyridines; RNA, Messenger; Transcription Factors

2001
Early growth response-1 gene (Egr-1) promoter induction by ionizing radiation in U87 malignant glioma cells in vitro.
    European journal of biochemistry, 2002, Volume: 269, Issue:1

    Topics: Androstadienes; Anisomycin; Blotting, Western; Colforsin; DNA-Binding Proteins; Early Growth Response Protein 1; Epidermal Growth Factor; Flavonoids; Glioma; Humans; Imidazoles; Immediate-Early Proteins; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Pyridines; Suramin; Transcription Factors; Wortmannin

2002
Differentiation of human melanoma cells through p38 MAP kinase is associated with decreased retinoblastoma protein phosphorylation and cell cycle arrest.
    Melanoma research, 2002, Volume: 12, Issue:3

    Topics: alpha-MSH; Cell Differentiation; Colforsin; Dose-Response Relationship, Drug; Enzyme Inhibitors; G1 Phase; Humans; Imidazoles; Kinetics; MAP Kinase Signaling System; Melanins; Melanoma; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neoplasm Proteins; Phosphorylation; Protein Processing, Post-Translational; Pyridines; Retinoblastoma Protein; Tumor Cells, Cultured

2002
TGF-beta effects on epithelial ion transport and barrier: reduced Cl- secretion blocked by a p38 MAPK inhibitor.
    American journal of physiology. Cell physiology, 2002, Volume: 283, Issue:6

    Topics: Biological Transport; Chlorides; Colforsin; Colon; Cyclic AMP; Electric Conductivity; Enzyme Inhibitors; Gene Transfer Techniques; Humans; Imidazoles; Intestinal Mucosa; Ions; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Permeability; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Transforming Growth Factor beta; Tumor Cells, Cultured

2002
Role of the different mitogen-activated protein kinase subfamilies in the stimulation of dog and human thyroid epithelial cell proliferation by cyclic adenosine 5'-monophosphate and growth factors.
    Endocrinology, 2003, Volume: 144, Issue:4

    Topics: Animals; Arsenites; Carcinogens; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Dogs; Enzyme Inhibitors; Epidermal Growth Factor; Epithelial Cells; Flavonoids; Hepatocyte Growth Factor; Humans; Hypoglycemic Agents; Imidazoles; Insulin; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Sodium Compounds; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin

2003
Chronic regulation of the expression of the gap junction protein connexin 43 in transfected HeLa cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 2003, Volume: 368, Issue:1

    Topics: Adenylyl Cyclases; Blotting, Western; Colforsin; Connexin 43; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Flavonoids; Fluorescent Antibody Technique; Gap Junctions; Gene Expression Regulation; HeLa Cells; Humans; Imidazoles; Protein Kinase C; Protein-Tyrosine Kinases; Pyridines; Receptors, Tumor Necrosis Factor; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Transfection; Tumor Necrosis Factor-alpha

2003
Induction of cytokine mRNA expression in U937 cells by Salmonella typhimurium porins is regulated by different phosphorylation pathways.
    Medical microbiology and immunology, 2005, Volume: 194, Issue:1-2

    Topics: Colforsin; Cytokines; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Humans; Imidazoles; Lipopolysaccharides; Monocytes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Porins; Proto-Oncogene Proteins c-raf; Pyridines; RNA, Messenger; Salmonella typhimurium; U937 Cells

2005
Possible involvement of p38 MAP kinase in prostaglandin E1-induced ALP activity in osteoblast-like cells.
    Prostaglandins, leukotrienes, and essential fatty acids, 2004, Volume: 70, Issue:5

    Topics: Adenylyl Cyclases; Alkaline Phosphatase; Alprostadil; Animals; Bucladesine; Cell Differentiation; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Imidazoles; Isoquinolines; Mice; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Sulfonamides

2004
Involvement of SAPK/JNK in prostaglandin E(1)-induced VEGF synthesis in osteoblast-like cells.
    Molecular and cellular endocrinology, 2004, May-31, Volume: 220, Issue:1-2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Alprostadil; Animals; Anthracenes; Cell Line; Colforsin; Imidazoles; JNK Mitogen-Activated Protein Kinases; Mice; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Proto-Oncogene Proteins c-jun; Pyridines; Vascular Endothelial Growth Factor A

2004
cAMP-response element-binding protein mediates tumor necrosis factor-alpha-induced vascular smooth muscle cell migration.
    Arteriosclerosis, thrombosis, and vascular biology, 2004, Volume: 24, Issue:9

    Topics: Cell Movement; Cells, Cultured; Colforsin; Coronary Vessels; CREB-Binding Protein; Genes, Dominant; Genes, fos; Humans; Imidazoles; Ionomycin; MAP Kinase Signaling System; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Phosphoserine; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Pyridines; rac1 GTP-Binding Protein; Recombinant Fusion Proteins; Trans-Activators; Tumor Necrosis Factor-alpha

2004
Akt regulates thrombin-induced HSP27 phosphorylation in aortic smooth muscle cells: function at a point downstream from p38 MAP kinase.
    Life sciences, 2005, May-20, Volume: 77, Issue:1

    Topics: Adenylyl Cyclases; Animals; Aorta; Bucladesine; Cells, Cultured; Colforsin; Cyclic AMP; Heat-Shock Proteins; Imidazoles; Muscle, Smooth, Vascular; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Rats; Thrombin

2005
p38 mitogen-activated protein kinase contributes to cell cycle regulation by cAMP in FRTL-5 thyroid cells.
    European journal of endocrinology, 2005, Volume: 153, Issue:1

    Topics: Animals; CDC2-CDC28 Kinases; Cells, Cultured; Colforsin; Cyclic AMP; Cyclin-Dependent Kinase 2; Enzyme Inhibitors; G1 Phase; Hypoglycemic Agents; Imidazoles; Insulin; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Rats; S Phase; Signal Transduction; Threonine; Thyroid Gland; Tyrosine

2005
Activation of mitogen activated protein kinase pathways and melanogenesis by novel nitro-derivatives of 7-hydroxycomarin in human malignant melanoma cells.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2005, Volume: 26, Issue:1

    Topics: Antineoplastic Agents; Cell Differentiation; Cell Line, Tumor; Colforsin; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; MAP Kinase Signaling System; Melanins; Melanoma; Mitogen-Activated Protein Kinases; Monophenol Monooxygenase; Nitro Compounds; Pyridines; Umbelliferones

2005
p38 Mitogen-activated protein kinase plays a stimulatory role in hepatic gluconeogenesis.
    The Journal of biological chemistry, 2005, Dec-30, Volume: 280, Issue:52

    Topics: Acetylcysteine; Adenoviridae; Animals; Cell Line, Tumor; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Diabetes Mellitus, Type 1; Disease Models, Animal; Enzyme Inhibitors; Gene Silencing; Glucagon; Gluconeogenesis; Glucose; Glucose-6-Phosphatase; Hepatocytes; Imidazoles; Liver; Mice; p38 Mitogen-Activated Protein Kinases; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Phosphoenolpyruvate Carboxykinase (GTP); Phosphorylation; Promoter Regions, Genetic; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Small Interfering; Streptozocin; Trans-Activators; Transcription Factors; Transfection

2005
Stimulation of pancreatic beta-cell replication by incretins involves transcriptional induction of cyclin D1 via multiple signalling pathways.
    The Journal of endocrinology, 2006, Volume: 188, Issue:3

    Topics: Adenylyl Cyclases; Androstadienes; Animals; Animals, Newborn; Cell Line; Cell Proliferation; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclin D1; Enzyme Activation; Flavonoids; Gastric Inhibitory Polypeptide; Glucagon-Like Peptide 1; Human Growth Hormone; Imidazoles; Insulin-Secreting Cells; Isoquinolines; Liraglutide; Mitogen-Activated Protein Kinase Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Rats; Signal Transduction; Stimulation, Chemical; Sulfonamides; Transcription, Genetic; Transduction, Genetic; Wortmannin

2006
p38 MAP kinase regulation of oligodendrocyte differentiation with CREB as a potential target.
    Neurochemical research, 2007, Volume: 32, Issue:2

    Topics: Animals; Cell Differentiation; Cells, Cultured; Colforsin; Cyclic AMP Response Element-Binding Protein; Enzyme Activation; Imidazoles; Myelin Basic Protein; Myelin Proteolipid Protein; Myelin-Associated Glycoprotein; Oligodendroglia; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Rats; RNA, Messenger

2007
Involvement of regulatory elements on corticotropin-releasing factor gene promoter in hypothalamic 4B cells.
    Journal of endocrinological investigation, 2008, Volume: 31, Issue:12

    Topics: Anthracenes; Cell Line; Chromones; Colforsin; Corticotropin-Releasing Hormone; Dexamethasone; Flavonoids; Genes, Reporter; Humans; Hypothalamus; Imidazoles; Isoquinolines; Morpholines; Promoter Regions, Genetic; Protein Kinase Inhibitors; Pyridines; Regulatory Elements, Transcriptional; Sequence Deletion; Sulfonamides; Transfection

2008
Urocortin II induces nitric oxide production through cAMP and Ca2+ related pathways in endothelial cells.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2009, Volume: 23, Issue:1-3

    Topics: Androstadienes; Animals; Aorta; Blotting, Western; Butadienes; Calcimycin; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Dideoxyadenosine; Endothelial Cells; Imidazoles; Ionophores; Mitogen-Activated Protein Kinase 3; Nitric Oxide; Nitriles; Oncogene Protein v-akt; p38 Mitogen-Activated Protein Kinases; Peptide Fragments; Peptides, Cyclic; Pyridines; Signal Transduction; Swine; Urocortins; Wortmannin

2009
TGF-beta inhibits CYP17 transcription in H295R cells acting via activin receptor-like kinase 5.
    Endocrine research, 2009, Volume: 34, Issue:3

    Topics: Activin Receptors; Adrenal Cortex; Benzamides; Cell Line; Colforsin; Cytochromes b5; Dichlororibofuranosylbenzimidazole; Dioxoles; Humans; Imidazoles; MAP Kinase Kinase 1; NADPH-Ferrihemoprotein Reductase; p38 Mitogen-Activated Protein Kinases; Protein Serine-Threonine Kinases; Pyridines; Receptor, Transforming Growth Factor-beta Type I; Receptors, Transforming Growth Factor beta; RNA, Messenger; Steroid 17-alpha-Hydroxylase; Transforming Growth Factor beta

2009
An essential role for modulation of hyperpolarization-activated current in the development of binaural temporal precision.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Feb-22, Volume: 32, Issue:8

    Topics: Age Factors; Analysis of Variance; Androstadienes; Animals; Biophysical Phenomena; Bucladesine; Colforsin; Cyclic Nucleotide-Gated Cation Channels; Electric Stimulation; Enzyme Inhibitors; Female; Gene Expression Regulation, Developmental; Gerbillinae; Imidazoles; In Vitro Techniques; Ion Channel Gating; Male; Neurons; Olivary Nucleus; Patch-Clamp Techniques; Pyridines; Pyrimidines; Wortmannin

2012
Cyclic AMP relaxation of rat aortic smooth muscle is mediated in part by decrease of depletion of intracellular Ca(2+) stores and inhibition of capacitative calcium entry.
    Vascular pharmacology, 2013, Volume: 58, Issue:1-2

    Topics: Animals; Aorta, Thoracic; Calcium; Colforsin; Cyclic AMP; Imidazoles; Male; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Nifedipine; p38 Mitogen-Activated Protein Kinases; Phenylephrine; Phosphodiesterase 4 Inhibitors; Pyridines; Rats; Rats, Inbred WKY; Rolipram; Vasodilation; Vasodilator Agents; Verapamil

2013