Page last updated: 2024-09-05

sb 203580 and carbachol

sb 203580 has been researched along with carbachol in 5 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
3,48941,13713,91881968

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (20.00)18.2507
2000's4 (80.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gerthoffer, WT; Larsen, JK; Weber, LA; Yamboliev, IA1
del Valle, J; Pausawasdi, N; Ramamoorthy, S; Stepan, V; Todisco, A1
Abdel-Latif, AA; Gao, G; Yousufzai, SY1
Askari, FK; Crofford, LJ; Pausawasdi, N; Ramamoorthy, S; Todisco, A1
Barrett, KE; Carlstrom, K; Chow, JY1

Other Studies

5 other study(ies) available for sb 203580 and carbachol

ArticleYear
Phosphorylation of the 27-kDa heat shock protein via p38 MAP kinase and MAPKAP kinase in smooth muscle.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Amino Acid Sequence; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carbachol; Colon; Cricetinae; Dogs; Enzyme Activation; Female; Gene Library; Heat-Shock Proteins; Humans; Imidazoles; Intracellular Signaling Peptides and Proteins; Kinetics; Male; Mice; Mitogen-Activated Protein Kinases; Molecular Sequence Data; Muscle, Smooth; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Phosphotyrosine; Protein Serine-Threonine Kinases; Pyridines; Rats; Recombinant Proteins; Sequence Alignment; Sequence Homology, Amino Acid

1997
Regulation and function of p38 protein kinase in isolated canine gastric parietal cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2000, Volume: 278, Issue:1

    Topics: ADP Ribose Transferases; Aminopyrine; Animals; Botulinum Toxins; Calcium; Carbachol; Cell Separation; Cells, Cultured; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Imidazoles; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Parietal Cells, Gastric; Pyridines; rho GTP-Binding Proteins; Time Factors

2000
Mitogen-activated protein kinase inhibitors suppress prostaglandin F(2alpha)-induced myosin-light chain phosphorylation and contraction in iris sphincter smooth muscle.
    European journal of pharmacology, 2000, Oct-27, Volume: 407, Issue:1-2

    Topics: Animals; Carbachol; Cats; Dinoprost; Enzyme Inhibitors; Flavonoids; Imidazoles; Iris; Miotics; Mitogen-Activated Protein Kinases; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Oxytocics; Phosphorylation; Pyridines

2000
Regulation and function of COX-2 gene expression in isolated gastric parietal cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:6

    Topics: Animals; Carbachol; Cells, Cultured; Cholinergic Agonists; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dogs; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Histamine; Imidazoles; Indoles; Isoenzymes; Maleimides; NF-kappa B; Nitrobenzenes; Parietal Cells, Gastric; Prostaglandin-Endoperoxide Synthases; Prostaglandins; Pyridines; Sulfonamides

2002
Growth hormone reduces chloride secretion in human colonic epithelial cells via EGF receptor and extracellular regulated kinase.
    Gastroenterology, 2003, Volume: 125, Issue:4

    Topics: Biological Transport; Carbachol; Cell Line; Chlorides; Cholinergic Agonists; Enzyme Inhibitors; Epithelial Cells; ErbB Receptors; Flavonoids; Human Growth Hormone; Humans; Imidazoles; Intestinal Mucosa; Janus Kinase 2; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphorylation; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Pyridines; Tyrosine

2003