Page last updated: 2024-09-05

sb 203580 and calyculin a

sb 203580 has been researched along with calyculin a in 5 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(calyculin a)
Trials
(calyculin a)
Recent Studies (post-2010) (calyculin a)
3,48941,1379150110

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)calyculin a (IC50)
Tyrosine-protein phosphatase non-receptor type 1Homo sapiens (human)0.0009
Serine/threonine-protein phosphatase PP1-gamma catalytic subunitHomo sapiens (human)0.0182
Serine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B Gallus gallus (chicken)0.0032

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, KD; Chen, LY; Cho, JH; Lai, MT; Lai, YK1
Armstrong, SC; Ganote, CE; Shivell, CL1
Grethe, S; Pörn-Ares, MI1
Bavec, A; Corda, D; Di Girolamo, M; Mariggiò, S; Natale, E; Salmona, M; Zizza, P1
Leslie, NR; Mackintosh, C; Murphy, J; Pozuelo-Rubio, M1

Other Studies

5 other study(ies) available for sb 203580 and calyculin a

ArticleYear
Activation of p38 mitogen-activated protein kinase and mitochondrial Ca(2+)-mediated oxidative stress are essential for the enhanced expression of grp78 induced by the protein phosphatase inhibitors okadaic acid and calyculin A.
    Journal of cellular biochemistry, 2000, Volume: 76, Issue:4

    Topics: Acetylcysteine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Carrier Proteins; Egtazic Acid; Endoplasmic Reticulum Chaperone BiP; Enzyme Inhibitors; Heat-Shock Proteins; Imidazoles; Marine Toxins; Mitochondria; Mitogen-Activated Protein Kinases; Molecular Chaperones; Okadaic Acid; Oxazoles; Oxidative Stress; p38 Mitogen-Activated Protein Kinases; Phosphoprotein Phosphatases; Proline; Promoter Regions, Genetic; Pyridines; Rats; RNA, Messenger; Ruthenium Red; Thiocarbamates; Transcriptional Activation; Tumor Cells, Cultured

2000
Differential translocation or phosphorylation of alpha B crystallin cannot be detected in ischemically preconditioned rabbit cardiomyocytes.
    Journal of molecular and cellular cardiology, 2000, Volume: 32, Issue:7

    Topics: Animals; Blotting, Western; Cattle; Cells, Cultured; Crystallins; Cytoskeleton; Cytosol; Enzyme Inhibitors; Flavonoids; Heart Ventricles; Hydrogen-Ion Concentration; Imidazoles; Immunoblotting; Ischemic Preconditioning, Myocardial; Isoelectric Focusing; Lens, Crystalline; Marine Toxins; Mitogen-Activated Protein Kinases; Myocardium; Oxazoles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Isoforms; Pyridines; Rabbits; Time Factors

2000
p38 MAPK regulates phosphorylation of Bad via PP2A-dependent suppression of the MEK1/2-ERK1/2 survival pathway in TNF-alpha induced endothelial apoptosis.
    Cellular signalling, 2006, Volume: 18, Issue:4

    Topics: Alkenes; Apoptosis; bcl-Associated Death Protein; Cell Line; Cell Survival; Cells, Cultured; Down-Regulation; Endothelial Cells; Humans; Imidazoles; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Marine Toxins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Oxazoles; p38 Mitogen-Activated Protein Kinases; Phosphoprotein Phosphatases; Phosphorylation; Polyenes; Protein Phosphatase 2; Pyridines; Pyrones; Signal Transduction; Tumor Necrosis Factor-alpha

2006
Galpha13 mediates activation of the cytosolic phospholipase A2alpha through fine regulation of ERK phosphorylation.
    Cellular signalling, 2006, Volume: 18, Issue:12

    Topics: Animals; Arachidonic Acid; Butadienes; CHO Cells; Cricetinae; Cricetulus; Cytosol; Enzyme Activation; Enzyme Inhibitors; Group IV Phospholipases A2; GTP-Binding Protein alpha Subunits, G12-G13; Imidazoles; Marine Toxins; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Mutation; Nitriles; Oxazoles; Phospholipases A; Phosphoric Monoester Hydrolases; Phosphorylation; Pyridines; Pyrrolidines; rhoA GTP-Binding Protein; Transfection

2006
Mechanism of activation of PKB/Akt by the protein phosphatase inhibitor Calyculin A.
    Cell biochemistry and biophysics, 2010, Volume: 58, Issue:3

    Topics: 3-Phosphoinositide-Dependent Protein Kinases; Animals; Chromones; Embryonic Stem Cells; Enzyme Inhibitors; Imidazoles; Insulin Receptor Substrate Proteins; Insulin-Like Growth Factor I; Marine Toxins; Mice; Mitogen-Activated Protein Kinase 11; Morpholines; Oxazoles; Phosphatidylinositol 3-Kinases; Phosphoprotein Phosphatases; Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-akt; Pyridines

2010