Page last updated: 2024-09-05

sb 203580 and calcimycin

sb 203580 has been researched along with calcimycin in 12 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(calcimycin)
Trials
(calcimycin)
Recent Studies (post-2010) (calcimycin)
3,48941,13711,94640444

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)calcimycin (IC50)
XBP1Homo sapiens (human)1.41
DNA damage-inducible transcript 3 proteinMus musculus (house mouse)0.16

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (16.67)18.2507
2000's10 (83.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kozawa, O; Matsuno, H; Tokuda, H; Uematsu, T1
Creanor, J; Flatman, PW1
Cruise, L; Fuller, G; Ho, LK; Morris, BJ; Veitch, K1
Ammon, HP; Bertsche, T; Boden, SE; Safayhi, H1
Kozawa, O; Tokuda, H; Uematsu, T1
Linch, DC; Mollapour, E; Roberts, PJ1
Klemm, J; Rådmark, O; Samuelsson, B; Werz, O1
Gibbs, BF; Grabbe, J; Plath, KE; Wolff, HH1
Hsu, SC; Lai, MZ; Shih, HM; Wu, CC1
Febbraio, MA; Holmes, AG; Southgate, RJ; Watt, MJ1
Brunius, G; Domeij, H; Gustavsson, A; Yucel-Lindberg, T1
Caimmi, PP; Grossini, E; Mary, DA; Molinari, C; Ribichini, F; Uberti, F; Vacca, G1

Other Studies

12 other study(ies) available for sb 203580 and calcimycin

ArticleYear
Involvement of p38 mitogen-activated protein kinase in basic fibroblast growth factor-induced interleukin-6 synthesis in osteoblasts.
    Journal of cellular biochemistry, 1999, Sep-01, Volume: 74, Issue:3

    Topics: Animals; Calcimycin; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Diglycerides; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fibroblast Growth Factor 2; Imidazoles; Interleukin-6; Ionophores; Mice; Mitogen-Activated Protein Kinases; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Pyridines; Time Factors

1999
Stimulation of Na+-K+-2Cl- cotransport by arsenite in ferret erythrocytes.
    The Journal of physiology, 1999, Aug-15, Volume: 519 Pt 1

    Topics: Animals; Arsenites; Bumetanide; Calcimycin; Calcium-Calmodulin-Dependent Protein Kinases; Carrier Proteins; Chlorides; Edetic Acid; Enzyme Inhibitors; Erythrocytes; Ferrets; Flavonoids; Genistein; Homeostasis; Imidazoles; In Vitro Techniques; Models, Biological; Potassium; Pyridines; Rubidium; Rubidium Radioisotopes; Sodium; Sodium-Potassium-Chloride Symporters; Staurosporine

1999
Kainate receptors activate NF-kappaB via MAP kinase in striatal neurones.
    Neuroreport, 2000, Feb-07, Volume: 11, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Calcimycin; Calcium; Cells, Cultured; Corpus Striatum; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Flavonoids; Imidazoles; Immunohistochemistry; In Vitro Techniques; Ionophores; Kainic Acid; Mitogen-Activated Protein Kinases; N-Methylaspartate; Neurons; NF-kappa B; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Kainic Acid; Transcription Factor RelA

2000
MEK-1/2 inhibition prevents 5-lipoxygenase translocation in N-formylpeptide-challenged human neutrophils.
    The international journal of biochemistry & cell biology, 2000, Volume: 32, Issue:10

    Topics: Arachidonate 5-Lipoxygenase; Butadienes; Calcimycin; Calcium; Cell-Free System; Enzyme Activation; Flavonoids; Humans; Imidazoles; MAP Kinase Kinase 1; MAP Kinase Kinase 2; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase Kinases; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Nitriles; Phosphorylation; Protein Serine-Threonine Kinases; Protein Transport; Protein-Tyrosine Kinases; Pyridines

2000
Basic fibroblast growth factor stimulates vascular endothelial growth factor release in osteoblasts: divergent regulation by p42/p44 mitogen-activated protein kinase and p38 mitogen-activated protein kinase.
    Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 2000, Volume: 15, Issue:12

    Topics: Animals; Calcimycin; Calcium; Endothelial Growth Factors; Enzyme Inhibitors; Fibroblast Growth Factor 2; Flavonoids; Imidazoles; In Vitro Techniques; Ionophores; Lymphokines; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Thapsigargin; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2000
Activation and priming of neutrophil nicotinamide adenine dinucleotide phosphate oxidase and phospholipase A(2) are dissociated by inhibitors of the kinases p42(ERK2) and p38(SAPK) and by methyl arachidonyl fluorophosphonate, the dual inhibitor of cytosol
    Blood, 2001, Apr-15, Volume: 97, Issue:8

    Topics: Arachidonic Acid; Arachidonic Acids; Calcimycin; Complement C5a; Cytosol; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Granulocyte-Macrophage Colony-Stimulating Factor; Group VI Phospholipases A2; Humans; Imidazoles; Ionophores; Isoenzymes; MAP Kinase Kinase Kinase 1; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; Neutrophils; Organophosphonates; p38 Mitogen-Activated Protein Kinases; Phospholipases A; Protein Serine-Threonine Kinases; Pyridines; Respiratory Burst; Superoxides; Tumor Necrosis Factor-alpha

2001
p38 MAP kinase mediates stress-induced leukotriene synthesis in a human B-lymphocyte cell line.
    Journal of leukocyte biology, 2001, Volume: 70, Issue:5

    Topics: Arachidonate 5-Lipoxygenase; Arachidonic Acid; Arsenites; B-Lymphocytes; Calcimycin; Calcium; Cell Line; Cell-Free System; Enzyme Activation; Enzyme Inhibitors; Hydroxyeicosatetraenoic Acids; Hypertonic Solutions; Imidazoles; Interleukin-1; Intracellular Signaling Peptides and Proteins; Ionophores; Leukotrienes; Lipoxygenase Inhibitors; Mitogen-Activated Protein Kinases; Osmotic Pressure; Oxidative Stress; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinases; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Protein Tyrosine Phosphatases; Pyridines; Sodium Compounds; Sorbitol; Subcellular Fractions; Thapsigargin; Transforming Growth Factor beta; Tumor Necrosis Factor-alpha; Vanadates

2001
Regulation of mediator secretion in human basophils by p38 mitogen-activated protein kinase: phosphorylation is sensitive to the effects of phosphatidylinositol 3-kinase inhibitors and calcium mobilization.
    Journal of leukocyte biology, 2002, Volume: 72, Issue:2

    Topics: Albuterol; Basophils; Calcimycin; Calcium Channel Blockers; Calcium Signaling; Calcium-Calmodulin-Dependent Protein Kinases; Chromones; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Histamine Release; Humans; Imidazoles; Immunoglobulin E; Interleukin-13; Interleukin-4; Interleukins; Leukotriene C4; MAP Kinase Kinase 3; MAP Kinase Kinase 6; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Morpholines; N-Formylmethionine Leucyl-Phenylalanine; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Processing, Post-Translational; Protein-Tyrosine Kinases; Pyridines; Salmeterol Xinafoate; Second Messenger Systems; Theophylline

2002
Nuclear factor of activated T cells c is a target of p38 mitogen-activated protein kinase in T cells.
    Molecular and cellular biology, 2003, Volume: 23, Issue:18

    Topics: Animals; Calcimycin; Carrier Proteins; Cell Nucleus; Cells, Cultured; DNA-Binding Proteins; Enzyme Inhibitors; Humans; Imidazoles; Interleukin-2; Lymphocyte Activation; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinases; NFATC Transcription Factors; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Protein Biosynthesis; Protein Transport; Pyridines; RNA Stability; RNA, Messenger; T-Lymphocytes; Transcription Factors

2003
Suppression of plasma free fatty acids upregulates peroxisome proliferator-activated receptor (PPAR) alpha and delta and PPAR coactivator 1alpha in human skeletal muscle, but not lipid regulatory genes.
    Journal of molecular endocrinology, 2004, Volume: 33, Issue:2

    Topics: Calcimycin; Carnitine O-Palmitoyltransferase; CD36 Antigens; Cells, Cultured; Enzyme Inhibitors; Epinephrine; Exercise Test; Fatty Acids; Forkhead Transcription Factors; Heat-Shock Proteins; Humans; Hypolipidemic Agents; Imidazoles; Lipids; Muscle, Skeletal; Niacin; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Phosphorylation; PPAR alpha; PPAR delta; Protein Kinases; Pyridines; Sterol Esterase; Transcription Factors; Up-Regulation

2004
Bradykinin upregulates IL-8 production in human gingival fibroblasts stimulated by interleukin-1beta and tumor necrosis factor alpha.
    Regulatory peptides, 2005, Mar-30, Volume: 126, Issue:3

    Topics: Adolescent; Bradykinin; Bradykinin B2 Receptor Antagonists; Calcimycin; Cells, Cultured; Child; Fibroblasts; Gingiva; Humans; Imidazoles; Indoles; Interleukin-1; Interleukin-8; Ionophores; Kallidin; Maleimides; MAP Kinase Kinase 2; Protein Kinase C; Pyridines; Receptor, Bradykinin B2; Tumor Necrosis Factor-alpha; Up-Regulation

2005
Urocortin II induces nitric oxide production through cAMP and Ca2+ related pathways in endothelial cells.
    Cellular physiology and biochemistry : international journal of experimental cellular physiology, biochemistry, and pharmacology, 2009, Volume: 23, Issue:1-3

    Topics: Androstadienes; Animals; Aorta; Blotting, Western; Butadienes; Calcimycin; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Dideoxyadenosine; Endothelial Cells; Imidazoles; Ionophores; Mitogen-Activated Protein Kinase 3; Nitric Oxide; Nitriles; Oncogene Protein v-akt; p38 Mitogen-Activated Protein Kinases; Peptide Fragments; Peptides, Cyclic; Pyridines; Signal Transduction; Swine; Urocortins; Wortmannin

2009