Page last updated: 2024-09-05

sb 203580 and bucladesine

sb 203580 has been researched along with bucladesine in 13 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(bucladesine)
Trials
(bucladesine)
Recent Studies (post-2010) (bucladesine)
3,48941,1379,77513210

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (23.08)18.2507
2000's7 (53.85)29.6817
2010's3 (23.08)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burchell, A; Schmoll, D; Walther, R; Wasner, C; Watkins, SL1
Brooks, DP; Francis, J; Nambi, P; Parameswaran, N; Pullen, M; Spielman, WS1
Ikeda, K; Kawada, N; Kuroki, T; Seki, S1
Lahiri, T; Laporte, JD; Moore, PE; Panettieri, RA; Schwartzman, IN; Shore, SA1
Asakura, M; Asanuma, H; Fukushima, T; Hori, M; Kitakaze, M; Kuzuya, T; Liao, Y; Mori, H; Node, K; Ogai, A; Ogita, H; Papst, PJ; Sakata, Y; Sanada, S; Shinozaki, Y; Takashima, S; Terada, N; Yamada, J1
Castro-Caldas, M; Duarte, CB; Lopes, MC; Mendes, AF1
Itoh, M; Kakita, A; Miura, Y; Oiso, Y; Ono, Y; Suzuki, A1
Allen, JM; Bertrand, C; Jacob, C; Lagente, V; Szilagyi, C1
Hirade, K; Ishisaki, A; Kanno, Y; Katagiri, Y; Kitajima, Y; Kozawa, O; Matsuno, H; Nakajima, K; Shu, E; Suga, H1
Iijima, R; Ishida, A; Kobayashi, A; Maeda, M1
Fortes, B; Hurley, DJ; Linden, J; Moore, JN; Sun, WC; Thompson, R; Vandenplas, ML1
Avni, D; Meijler, MM; Philosoph, A; Zor, T1
Chetkovich, D; Golding, NL; Khurana, S; Lewis, AS; Liu, Z; Rosa, K1

Other Studies

13 other study(ies) available for sb 203580 and bucladesine

ArticleYear
Glucose induces glucose 6-phosphatase hydrolytic subunit gene transcription in an insulinoma cell line (INS-1).
    FEBS letters, 1999, Jan-22, Volume: 443, Issue:1

    Topics: Bucladesine; Calcium-Calmodulin-Dependent Protein Kinases; Dexamethasone; Enzyme Induction; Genes, Reporter; Glucose; Glucose-6-Phosphatase; Humans; Imidazoles; Insulinoma; Islets of Langerhans; Liver; Luciferases; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Pyridines; Transcription, Genetic; Tumor Cells, Cultured

1999
Mechanism of adrenomedullin-stimulated hyaluronic acid release in rat mesangial cells.
    European journal of pharmacology, 1999, Apr-16, Volume: 370, Issue:3

    Topics: Adrenomedullin; Animals; Bucladesine; Cell Culture Techniques; Colforsin; Drug Interactions; Enzyme Inhibitors; Glomerular Mesangium; Hyaluronic Acid; Imidazoles; Kidney Cortex; Male; Peptides; Phosphotransferases; Pyridines; Rats; Rats, Sprague-Dawley; Vasodilator Agents

1999
Expression of cyclins D1, D2 and E correlates with proliferation of rat stellate cells in culture.
    Journal of hepatology, 1999, Volume: 30, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Blotting, Northern; Blotting, Western; Bromodeoxyuridine; Bucladesine; Cell Cycle; Cell Division; Cells, Cultured; Chromones; Cyclin D1; Cyclin D2; Cyclin E; Cyclin-Dependent Kinase 4; Cyclin-Dependent Kinases; Cyclins; DNA; Enzyme Inhibitors; Flavonoids; G1 Phase; Imidazoles; Liver; Male; Morpholines; Phosphoinositide-3 Kinase Inhibitors; Proto-Oncogene Proteins; Pyridines; Rats; Rats, Wistar; Receptors, Platelet-Derived Growth Factor; RNA, Messenger; S Phase; Thymidine; Tritium

1999
p38 MAP kinase regulates IL-1 beta responses in cultured airway smooth muscle cells.
    American journal of physiology. Lung cellular and molecular physiology, 2000, Volume: 279, Issue:5

    Topics: Bucladesine; Cells, Cultured; Cyclooxygenase 2; Dinoprostone; Enzyme Inhibitors; Humans; Imidazoles; Interleukin-1; Isoenzymes; Isoproterenol; Leupeptins; Membrane Proteins; Mitogen-Activated Protein Kinases; NF-kappa B; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Prostaglandin-Endoperoxide Synthases; Pyridines; Transcription Factor AP-1

2000
Cardioprotective effect afforded by transient exposure to phosphodiesterase III inhibitors: the role of protein kinase A and p38 mitogen-activated protein kinase.
    Circulation, 2001, Aug-07, Volume: 104, Issue:6

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Blood Flow Velocity; Bucladesine; Calcium-Calmodulin-Dependent Protein Kinases; Cardiovascular Agents; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 3; Dogs; Enzyme Inhibitors; Flavonoids; Hemodynamics; Imidazoles; Indoles; Isoquinolines; Maleimides; Milrinone; Mitogen-Activated Protein Kinases; Myocardial Infarction; p38 Mitogen-Activated Protein Kinases; Phosphodiesterase Inhibitors; Protein Kinase C; Pyridines; Pyridones; Sulfonamides; Ventricular Fibrillation

2001
Dexamethasone-induced and estradiol-induced CREB activation and annexin 1 expression in CCRF-CEM lymphoblastic cells: evidence for the involvement of cAMP and p38 MAPK.
    Mediators of inflammation, 2003, Volume: 12, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Annexin A1; Bucladesine; Cells, Cultured; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Dexamethasone; Enzyme Inhibitors; Estradiol; Humans; Imidazoles; Lymphocytes; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Pyridines; Response Elements; Signal Transduction; Thionucleotides

2003
Possible involvement of p38 MAP kinase in prostaglandin E1-induced ALP activity in osteoblast-like cells.
    Prostaglandins, leukotrienes, and essential fatty acids, 2004, Volume: 70, Issue:5

    Topics: Adenylyl Cyclases; Alkaline Phosphatase; Alprostadil; Animals; Bucladesine; Cell Differentiation; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Imidazoles; Isoquinolines; Mice; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Sulfonamides

2004
Role of PDE4 in superoxide anion generation through p44/42MAPK regulation: a cAMP and a PKA-independent mechanism.
    British journal of pharmacology, 2004, Volume: 143, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Bronchoalveolar Lavage Fluid; Bucladesine; CREB-Binding Protein; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclohexanecarboxylic Acids; Flavonoids; Gene Expression Regulation, Enzymologic; Imidazoles; Lipopolysaccharides; Macrophages; Mitogen-Activated Protein Kinases; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Nitriles; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-raf; Pyridines; Rats; Rats, Wistar; Reactive Oxygen Species; Rolipram; Superoxides; Trans-Activators

2004
Akt regulates thrombin-induced HSP27 phosphorylation in aortic smooth muscle cells: function at a point downstream from p38 MAP kinase.
    Life sciences, 2005, May-20, Volume: 77, Issue:1

    Topics: Adenylyl Cyclases; Animals; Aorta; Bucladesine; Cells, Cultured; Colforsin; Cyclic AMP; Heat-Shock Proteins; Imidazoles; Muscle, Smooth, Vascular; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Pyridines; Rats; Thrombin

2005
Characterization of cAMP-dependent proteolysis of GATA-6.
    Biochemical and biophysical research communications, 2005, Jul-15, Volume: 332, Issue:4

    Topics: Animals; Base Sequence; Benzylamines; Binding Sites; Bucladesine; Carbazoles; Cell Nucleus; CHO Cells; Cricetinae; Cyclic AMP; DNA-Binding Proteins; Enzyme Inhibitors; Flavonoids; GATA6 Transcription Factor; Humans; Imidazoles; Indole Alkaloids; Isoquinolines; MAP Kinase Kinase Kinase 1; MAP Kinase Signaling System; Molecular Sequence Data; Mutation; Naphthalenes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Plasmids; Prostaglandin D2; Proteasome Endopeptidase Complex; Protein Binding; Pyridines; src-Family Kinases; Sulfonamides; Transcription Factors

2005
Differential modulation of lipopolysaccharide-induced expression of inflammatory genes in equine monocytes through activation of adenosine A2A receptors.
    Veterinary immunology and immunopathology, 2010, Apr-15, Volume: 134, Issue:3-4

    Topics: Adenosine A2 Receptor Agonists; Animals; Base Sequence; Bucladesine; Cyclooxygenase 2; Cytokines; DNA Primers; Drug Synergism; Gene Expression; Horses; Imidazoles; In Vitro Techniques; Inflammation Mediators; Interleukin-10; Lipopolysaccharides; Monocytes; Piperidines; Pyridines; Receptor, Adenosine A2A

2010
The ceramide-1-phosphate analogue PCERA-1 modulates tumour necrosis factor-alpha and interleukin-10 production in macrophages via the cAMP-PKA-CREB pathway in a GTP-dependent manner.
    Immunology, 2010, Volume: 129, Issue:3

    Topics: Adenylyl Cyclases; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bucladesine; Calcium Signaling; Cell Line; Cell Membrane; Ceramides; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Enzyme Inhibitors; Genes, Reporter; Guanosine Triphosphate; Imidazoles; Indoles; Interleukin-10; Isoquinolines; Lipopolysaccharides; Macrophages; Mice; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Pyridines; Response Elements; Ribosomal Protein S6 Kinases, 90-kDa; Rolipram; Signal Transduction; Sulfonamides; Transfection; Tumor Necrosis Factor-alpha

2010
An essential role for modulation of hyperpolarization-activated current in the development of binaural temporal precision.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Feb-22, Volume: 32, Issue:8

    Topics: Age Factors; Analysis of Variance; Androstadienes; Animals; Biophysical Phenomena; Bucladesine; Colforsin; Cyclic Nucleotide-Gated Cation Channels; Electric Stimulation; Enzyme Inhibitors; Female; Gene Expression Regulation, Developmental; Gerbillinae; Imidazoles; In Vitro Techniques; Ion Channel Gating; Male; Neurons; Olivary Nucleus; Patch-Clamp Techniques; Pyridines; Pyrimidines; Wortmannin

2012