Page last updated: 2024-09-05

sb 203580 and brefeldin a

sb 203580 has been researched along with brefeldin a in 8 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(brefeldin a)
Trials
(brefeldin a)
Recent Studies (post-2010) (brefeldin a)
3,48941,1372,6001456

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)brefeldin a (IC50)
major prion protein preproprotein Prp precursorHomo sapiens (human)3.505
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)0.1343

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (62.50)29.6817
2010's3 (37.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bilter, GK; Dias, J; Huang, Z; Keon, BH; Lamerdin, J; MacDonald, ML; Michnick, SW; Minami, T; Owens, S; Shang, Z; Westwick, JK; Yu, H1
Cruciani, V; Mikalsen, SO1
Andreka, P; Bishopric, NH; Evans, WH; Haywood, GA; Martin, PE; Turner, MS; Webster, KA; You, L1
Aizu-Yokota, E; Kasahara, T; Murakami, Y; Ohta, S; Sonoda, Y1
Choi, KH; Eo, SK; Kim, K; Kim, SM; Lee, KA; Moon, YS; Rhim, BY; Son, YH; Sung, SC1
Chae, HJ; Chae, SW; Kim, DS; Kim, HR; Kim, HT; Kim, JH; Lee, GH; Lim, JM1
Goto, K; Hozumi, Y; Nakano, T; Wakabayashi, I1
Ansorena, E; de Galarreta, MR; Garzón, AG; Iraburu, MJ; López-Zabalza, MJ; Martínez-Irujo, JJ; Mòdol, T; Navarro, A1

Other Studies

8 other study(ies) available for sb 203580 and brefeldin a

ArticleYear
Identifying off-target effects and hidden phenotypes of drugs in human cells.
    Nature chemical biology, 2006, Volume: 2, Issue:6

    Topics: Bacterial Proteins; Cell Line; Cell Proliferation; Cluster Analysis; Drug Design; Drug Evaluation, Preclinical; Genetics; Humans; Luminescent Proteins; Molecular Structure; Phenotype; Recombinant Fusion Proteins; Signal Transduction; Structure-Activity Relationship

2006
Mechanisms involved in responses to the poroxisome proliferator WY-14,643 on gap junctional intercellular communication in V79 hamster fibroblasts.
    Toxicology and applied pharmacology, 2002, Jul-01, Volume: 182, Issue:1

    Topics: Acetophenones; Androstadienes; Animals; Benzopyrans; Brefeldin A; Butadienes; Cell Communication; Cells, Cultured; Cricetinae; Cricetulus; Enzyme Inhibitors; Flavonoids; Gap Junctions; Imidazoles; Indoles; Maleimides; Mesocricetus; Mitogen-Activated Protein Kinases; Nitriles; Peroxisome Proliferators; Protein Kinase C; Protein Synthesis Inhibitors; Pyridines; Pyrimidines; Signal Transduction; Sirolimus; Wortmannin

2002
Reversible connexin 43 dephosphorylation during hypoxia and reoxygenation is linked to cellular ATP levels.
    Circulation research, 2004, Oct-01, Volume: 95, Issue:7

    Topics: Adenosine Triphosphate; Alkaloids; Aminoimidazole Carboxamide; Animals; Antimycin A; Benzophenanthridines; Brefeldin A; Carbazoles; Cell Hypoxia; Cells, Cultured; Connexin 43; Cycloheximide; Deoxyglucose; Flavonoids; Imidazoles; Indoles; JNK Mitogen-Activated Protein Kinases; Maleimides; Myocardial Contraction; Myocytes, Cardiac; Okadaic Acid; Ouabain; Phenanthridines; Phosphorylation; Potassium Cyanide; Protein Processing, Post-Translational; Pyridines; Pyrroles; Rats; Recombinant Fusion Proteins; Ribonucleotides; Staurosporine; Tacrolimus; Tetradecanoylphorbol Acetate

2004
Suppression of endoplasmic reticulum stress-induced caspase activation and cell death by the overexpression of Bcl-xL or Bcl-2.
    Journal of biochemistry, 2007, Volume: 141, Issue:3

    Topics: Animals; Anthracenes; Apoptosis; bcl-X Protein; Brefeldin A; Caspase 2; Caspase 9; Cytochromes c; Endoplasmic Reticulum; Enzyme Activation; Imidazoles; JNK Mitogen-Activated Protein Kinases; NFI Transcription Factors; PC12 Cells; Proto-Oncogene Proteins c-bcl-2; Pyridines; Rats; Transfection

2007
7-Ketocholesterol upregulates interleukin-6 via mechanisms that are distinct from those of tumor necrosis factor-alpha, in vascular smooth muscle cells.
    Journal of vascular research, 2009, Volume: 46, Issue:1

    Topics: Animals; Anthracenes; Brefeldin A; CCAAT-Enhancer-Binding Proteins; Cells, Cultured; Dactinomycin; ELAV Proteins; Humans; Imidazoles; Interleukin-6; Ketocholesterols; Muscle, Smooth, Vascular; NF-kappa B; Pyridines; Rats; RNA, Messenger; Tumor Necrosis Factor-alpha; Up-Regulation

2009
p38 Mitogen-activated protein kinase is involved in endoplasmic reticulum stress-induced cell death and autophagy in human gingival fibroblasts.
    Biological & pharmaceutical bulletin, 2010, Volume: 33, Issue:4

    Topics: Autophagy; Brefeldin A; Cell Death; Endoplasmic Reticulum; Endoplasmic Reticulum Chaperone BiP; Enzyme Inhibitors; Fibroblasts; Gingiva; Heat-Shock Proteins; Humans; Imidazoles; Microtubule-Associated Proteins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Synthesis Inhibitors; Pyridines; Thapsigargin; Transcription Factor CHOP; Tunicamycin

2010
Involvement of diacylglycerol kinase γ in modulation of iNOS synthesis in Golgi apparatus of vascular endothelial cells.
    Naunyn-Schmiedeberg's archives of pharmacology, 2012, Volume: 385, Issue:8

    Topics: Animals; Aorta, Thoracic; Blotting, Western; Brefeldin A; Diacylglycerol Kinase; Endothelial Cells; Enzyme Inhibitors; Golgi Apparatus; Imidazoles; Immunohistochemistry; Interleukin-1beta; Isoenzymes; Male; Nitric Oxide Synthase Type II; Nocodazole; Piperidines; Protein Synthesis Inhibitors; Pyridines; Quinazolinones; Rats; Rats, Wistar; Real-Time Polymerase Chain Reaction; RNA, Messenger

2012
Unfolded protein response induced by Brefeldin A increases collagen type I levels in hepatic stellate cells through an IRE1α, p38 MAPK and Smad-dependent pathway.
    Biochimica et biophysica acta, 2016, Volume: 1863, Issue:8

    Topics: Animals; Brefeldin A; Cell Line; Collagen Type I; Endoplasmic Reticulum Stress; Endoribonucleases; Fibrosis; Gene Expression Regulation; Hepatic Stellate Cells; Imidazoles; MAP Kinase Signaling System; Multienzyme Complexes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Pyridines; Rats; RNA, Messenger; Smad3 Protein; Unfolded Protein Response

2016