Page last updated: 2024-09-05

sb 203580 and bq 123

sb 203580 has been researched along with bq 123 in 7 studies

Compound Research Comparison

Studies
(sb 203580)
Trials
(sb 203580)
Recent Studies (post-2010)
(sb 203580)
Studies
(bq 123)
Trials
(bq 123)
Recent Studies (post-2010) (bq 123)
3,48941,1371,39163152

Protein Interaction Comparison

ProteinTaxonomysb 203580 (IC50)bq 123 (IC50)
Endothelin-1 receptorHomo sapiens (human)0.017
Endothelin-1 receptorRattus norvegicus (Norway rat)0.014

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (28.57)18.2507
2000's2 (28.57)29.6817
2010's3 (42.86)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ishida, T; Kawai, M; Kawashima, S; Namiki, M; Rikitake, Y; Sakoda, T; Ueyama, T; Yokoyama, M1
Kato, K; Kawamura, H; Kozawa, O; Matsui, N; Matsuno, H; Niwa, M; Otsuka, T; Uematsu, T1
Bagnato, A; Di Castro, V; Elia, G; Natali, PG; Rosanò, L; Spinella, F1
Calderone, A; Dupuis, J; Préfontaine, A1
Forman, SP; Katzenberg, G; Ohanian, J; Ohanian, V1
Cheng, M; Li, M; Meng, W; She, T; Shi, C; Wang, B; Yu, L1
E, LL; Liang, L; Liu, H; Liu, N; Wang, DS; Yu, J; Zhou, W1

Other Studies

7 other study(ies) available for sb 203580 and bq 123

ArticleYear
Endothelin-1 activates p38 mitogen-activated protein kinase via endothelin-A receptor in rat myocardial cells.
    Molecular and cellular biochemistry, 1999, Volume: 199, Issue:1-2

    Topics: Animals; Blotting, Western; Cardiomegaly; Cells, Cultured; Dose-Response Relationship, Drug; Endothelin-1; Enzyme Activation; Enzyme Inhibitors; Imidazoles; Leucine; Mitogen-Activated Protein Kinases; Myocardium; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phosphorylation; Piperidines; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptors, Endothelin; Sarcomeres

1999
Endothelin-1 stimulates heat shock protein 27 induction in osteoblasts: involvement of p38 MAP kinase.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: Animals; Antihypertensive Agents; Blotting, Northern; Carcinogens; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Estrenes; Flavonoids; Gene Expression Regulation, Enzymologic; Genistein; Heat-Shock Proteins; Imidazoles; Mice; Mitogen-Activated Protein Kinases; Naphthalenes; Oligopeptides; Osteoblasts; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phorbol Esters; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Propranolol; Protein Kinase C; Pyridines; Pyrrolidinones; RNA, Messenger; Skull; Staurosporine

1999
Endothelin-1 stimulates cyclooxygenase-2 expression in ovarian cancer cells through multiple signaling pathways: evidence for involvement of transactivation of the epidermal growth factor receptor.
    Journal of cardiovascular pharmacology, 2004, Volume: 44 Suppl 1

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cyclooxygenase 1; Cyclooxygenase 2; Dinoprostone; Endothelin A Receptor Antagonists; Endothelin-1; Enzyme Induction; ErbB Receptors; Female; Flavonoids; Gene Expression Regulation, Neoplastic; Humans; Imidazoles; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Ovarian Neoplasms; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Protein Kinase Inhibitors; Pyridines; Quinazolines; Receptor, Endothelin A; Signal Transduction; Transcriptional Activation; Tyrphostins

2004
Role of endothelin receptors on basal and endothelin-1-stimulated lung myofibroblast proliferation.
    Canadian journal of physiology and pharmacology, 2008, Volume: 86, Issue:6

    Topics: Animals; Cell Proliferation; Cells, Cultured; Chromones; Endothelin A Receptor Antagonists; Endothelin B Receptor Antagonists; Endothelin-1; Enzyme Inhibitors; Fibroblasts; Imidazoles; Lung; Male; Morpholines; Myoblasts, Smooth Muscle; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Phosphoinositide-3 Kinase Inhibitors; Piperidines; Pyridines; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B

2008
Endothelin-1 stimulates small artery VCAM-1 expression through p38MAPK-dependent neutral sphingomyelinase.
    Journal of vascular research, 2012, Volume: 49, Issue:4

    Topics: Aniline Compounds; Animals; Benzylidene Compounds; Endothelin B Receptor Antagonists; Endothelin-1; HSP27 Heat-Shock Proteins; Imidazoles; Mesenteric Arteries; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Piperidines; Pyridines; Rats; Sphingomyelin Phosphodiesterase; Vascular Cell Adhesion Molecule-1

2012
Endothelin-1 stimulates the expression of L-type Ca2+ channels in neonatal rat cardiomyocytes via the extracellular signal-regulated kinase 1/2 pathway.
    The Journal of membrane biology, 2013, Volume: 246, Issue:4

    Topics: Animals; Animals, Newborn; Anthracenes; Blotting, Western; Cells, Cultured; Endothelin-1; Enzyme Inhibitors; Flavonoids; Imidazoles; JNK Mitogen-Activated Protein Kinases; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocytes, Cardiac; Oligopeptides; Patch-Clamp Techniques; Peptides, Cyclic; Piperidines; Pyridines; Rats; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction

2013
Endothelin-1 stimulates proinflammatory cytokine expression in human periodontal ligament cells via mitogen-activated protein kinase pathway.
    Journal of periodontology, 2014, Volume: 85, Issue:4

    Topics: Adult; Anthracenes; Calcium-Calmodulin-Dependent Protein Kinases; Cell Culture Techniques; Cells, Cultured; Cytokines; Dose-Response Relationship, Drug; Endothelin B Receptor Antagonists; Endothelin Receptor Antagonists; Endothelin-1; Female; Flavonoids; Humans; Imidazoles; Interleukin-1beta; Interleukin-6; JNK Mitogen-Activated Protein Kinases; Male; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Oligopeptides; p38 Mitogen-Activated Protein Kinases; Peptides, Cyclic; Periodontal Ligament; Periodontitis; Piperidines; Pyridines; Time Factors; Tumor Necrosis Factor-alpha

2014