sb 203580 has been researched along with ag-490 in 28 studies
Studies (sb 203580) | Trials (sb 203580) | Recent Studies (post-2010) (sb 203580) | Studies (ag-490) | Trials (ag-490) | Recent Studies (post-2010) (ag-490) |
---|---|---|---|---|---|
3,489 | 4 | 1,137 | 732 | 2 | 322 |
Protein | Taxonomy | sb 203580 (IC50) | ag-490 (IC50) |
---|---|---|---|
Epidermal growth factor receptor | Homo sapiens (human) | 1.9224 | |
Tyrosine-protein kinase JAK1 | Homo sapiens (human) | 3.38 | |
large T antigen | Betapolyomavirus macacae | 14.61 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (3.57) | 18.2507 |
2000's | 19 (67.86) | 29.6817 |
2010's | 8 (28.57) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M | 1 |
Augustin, M; Davies, SP; Gao, Y; Harvey, KJ; Kovelman, R; Patel, UA; Woodward, A | 1 |
Carvalho, AP; Cruz, MT; Duarte, CB; Gonçalo, M; Lopes, MC | 1 |
Bertoglio, J; David, M; Ford, D; Maizel, AL; Pierre, J | 1 |
Duan, J; Norby, FL; Relling, DP; Ren, J; Wold, LE | 1 |
Caramona, MM; Carvalho, AP; Lopes, MC; Mendes, AF | 1 |
Alarcon-Vargas, D; Ronai, Z; Tansey, WP | 1 |
Aberle, NS; Hintz, KK; Ren, J | 1 |
Angelovska, T; Borowiec, AM; Dixon, IM; Freed, DH | 1 |
Ingelfinger, JR; Moini, B; Zhang, SL | 1 |
De Girolamo, S; Li, RK; Madani, S; Muñoz, DM; Sweeney, G | 1 |
Fu, Y; He, S; Luo, J; Wang, L | 1 |
Ip, WK; Lam, CW; Wong, CK | 1 |
Cao, Q; Lieber, CS; Mak, KM | 1 |
Figulla, HR; Foerster, M; Fritzenwanger, M; Krack, A; Kuethe, F; Meusel, K | 1 |
Chiasson, S; Girard, D; Pelletier, M; Ratthé, C | 1 |
Chen, S; He, S; Lin, Q; Yang, H; Yang, P; Yang, X; Zhang, H; Zhang, Z; Zheng, Y | 1 |
Ceylan-Isik, AF; Esberg, LB; Relling, DP; Ren, J; Zhu, BH | 1 |
Di Rosa, M; Li Volti, G; Malaguarnera, L; Marsullo, AR; Zambito, AM | 1 |
Descoteaux, A; Diallo, TO; Hardy, PO; Matte, C | 1 |
Chang, CW; Chuang, WJ; Lin, MT; Lin, YS; Liu, CC; Tsai, PJ; Tsai, WH; Wu, JJ | 1 |
Chachadi, VB; Inamdar, SR; Nagre, NN; Pujari, R; Shastry, P; Swamy, BM | 1 |
Chen, YE; Han, JY; Huang, Y; Ji, L; Liu, D; Pan, B; Pennathur, S; Tong, X; Zhang, Y; Zheng, L | 1 |
Dahmer, MK; Park, SK; Quasney, MW | 1 |
Bornstein, SR; Graessler, J; Kopprasch, S; Saha, S; Schwarz, PE | 1 |
Jia, CZ; Luo, JM; Wang, L; Zhu, ZY | 1 |
Chen, KL; Li, XF; Luo, J; Niu, HQ; Qin, KL; Zhao, WP; Zhao, XC | 1 |
Jiang, X; Li, SH; Li, ZH; Liang, JX; Liao, X; Liu, HW; Wu, F; Wu, YD; Xu, Y; Yan, JX | 1 |
28 other study(ies) available for sb 203580 and ag-490
Article | Year |
---|---|
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases | 2007 |
A broad activity screen in support of a chemogenomic map for kinase signalling research and drug discovery.
Topics: Aurora Kinases; Cluster Analysis; Drug Design; Drug Discovery; Drug Evaluation, Preclinical; ErbB Receptors; Humans; Intracellular Signaling Peptides and Proteins; MAP Kinase Kinase 4; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptors, Vascular Endothelial Growth Factor; Recombinant Proteins; Reproducibility of Results; Signal Transduction; Small Molecule Libraries; Structure-Activity Relationship; Syk Kinase | 2013 |
Involvement of JAK2 and MAPK on type II nitric oxide synthase expression in skin-derived dendritic cells.
Topics: Animals; Cell Nucleus; Cells, Cultured; Dendritic Cells; Enzyme Inhibitors; Fetus; Flavonoids; Fluorescent Antibody Technique; Genistein; Granulocyte-Macrophage Colony-Stimulating Factor; Imidazoles; Interleukin-1; Janus Kinase 2; Lipopolysaccharides; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinases; NF-kappa B; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; p38 Mitogen-Activated Protein Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Pyridines; Skin; Tumor Necrosis Factor-alpha; Tyrphostins | 1999 |
Induction of the IL-13 receptor alpha2-chain by IL-4 and IL-13 in human keratinocytes: involvement of STAT6, ERK and p38 MAPK pathways.
Topics: Antineoplastic Agents; Blotting, Western; Butadienes; Cross-Linking Reagents; Enzyme Inhibitors; Gene Expression Regulation, Neoplastic; Imidazoles; Interleukin-13; Interleukin-13 Receptor alpha1 Subunit; Interleukin-4; Keratinocytes; Kinetics; Ligands; Mitogen-Activated Protein Kinases; Nitriles; p38 Mitogen-Activated Protein Kinases; Plasmids; Precipitin Tests; Protein Binding; Pyridines; Receptors, Interleukin; Receptors, Interleukin-13; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; STAT6 Transcription Factor; Time Factors; Trans-Activators; Transcription, Genetic; Tumor Cells, Cultured; Tyrphostins | 2001 |
Abrogated leptin-induced cardiac contractile response in ventricular myocytes under spontaneous hypertension: role of Jak/STAT pathway.
Topics: Animals; Blood Pressure; Calcium; Carrier Proteins; Cell Size; DNA-Binding Proteins; Enzyme Inhibitors; Heart Ventricles; Hypertension; Imidazoles; Janus Kinase 2; Leptin; Mitogen-Activated Protein Kinase Kinases; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phosphorylation; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Pyridines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Cell Surface; Receptors, Leptin; Signal Transduction; STAT3 Transcription Factor; Trans-Activators; Tyrphostins; Ventricular Dysfunction, Left | 2002 |
Role of mitogen-activated protein kinases and tyrosine kinases on IL-1-Induced NF-kappaB activation and iNOS expression in bovine articular chondrocytes.
Topics: Animals; Cartilage, Articular; Cattle; Chondrocytes; Enzyme Inhibitors; Genistein; Humans; Imidazoles; Interleukin-1; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; NF-kappa B; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; p38 Mitogen-Activated Protein Kinases; Protein-Tyrosine Kinases; Pyridines; Signal Transduction; Transcription Factor AP-1; Tyrphostins | 2002 |
Regulation of c-myc stability by selective stress conditions and by MEKK1 requires aa 127-189 of c-myc.
Topics: Antineoplastic Agents; Apoptosis; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Cycloheximide; Dactinomycin; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Fibroblasts; Flavonoids; Humans; Imidazoles; MAP Kinase Kinase Kinase 1; Oligopeptides; Peptide Fragments; Protein Serine-Threonine Kinases; Protein Synthesis Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-myc; Pyridines; Stress, Physiological; Tumor Necrosis Factor-alpha; Tyrphostins; Ultraviolet Rays | 2002 |
Insulin resistance induces hyperleptinemia, cardiac contractile dysfunction but not cardiac leptin resistance in ventricular myocytes.
Topics: Animals; Blood Glucose; Calcium; Enzyme Inhibitors; Glucose Tolerance Test; Imidazoles; Insulin Resistance; Leptin; Male; Myocardial Contraction; Myocytes, Cardiac; NG-Nitroarginine Methyl Ester; Pyridines; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Tyrphostins; Ventricular Function | 2003 |
Induction of protein synthesis in cardiac fibroblasts by cardiotrophin-1: integration of multiple signaling pathways.
Topics: Animals; Blotting, Western; Cells, Cultured; Chromones; Cytokines; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Flavonoids; Imidazoles; Janus Kinase 1; Male; MAP Kinase Signaling System; Morpholines; Myocardium; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Precipitin Tests; Protein Biosynthesis; Protein-Tyrosine Kinases; Pyridines; Rats; Rats, Sprague-Dawley; Signal Transduction; Sirolimus; Tyrphostins | 2003 |
Angiotensin II increases Pax-2 expression in fetal kidney cells via the AT2 receptor.
Topics: Angiotensin II; Animals; Anthracenes; Blotting, Western; Cells, Cultured; DNA-Binding Proteins; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fibroblasts; Flavonoids; Genistein; Imidazoles; Kidney; Losartan; Mice; Microscopy, Fluorescence; Onium Compounds; PAX2 Transcription Factor; Phosphorylation; Plasmids; Pyridines; Receptors, Angiotensin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Time Factors; Transcription Factors; Tyrphostins; Up-Regulation | 2004 |
Direct effects of leptin on size and extracellular matrix components of human pediatric ventricular myocytes.
Topics: Cell Size; Cells, Cultured; Extracellular Matrix Proteins; Flavonoids; Heart Ventricles; Humans; Imidazoles; Infant; Janus Kinase 1; Leptin; Microscopy, Phase-Contrast; Mitogen-Activated Protein Kinase Kinases; Myocytes, Cardiac; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein-Tyrosine Kinases; Pyridines; Tyrphostins | 2006 |
Induction of interleukin-8 secretion and activation of ERK1/2, p38 MAPK signaling pathways by thrombin in dermal fibroblasts.
Topics: Adolescent; Adult; Butadienes; Chromones; Fibroblasts; Flavonoids; Humans; Imidazoles; Interleukin-8; Male; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Morpholines; Nitriles; p38 Mitogen-Activated Protein Kinases; Pyridines; Receptors, Proteinase-Activated; Signal Transduction; Skin; STAT3 Transcription Factor; Thrombin; Tyrphostins | 2006 |
Interleukin (IL)-4 and IL-13 up-regulate monocyte chemoattractant protein-1 expression in human bronchial epithelial cells: involvement of p38 mitogen-activated protein kinase, extracellular signal-regulated kinase 1/2 and Janus kinase-2 but not c-Jun NH2
Topics: Blotting, Western; Bronchi; Cell Line, Transformed; Cell Survival; Chemokine CCL2; Dose-Response Relationship, Drug; Enzyme Activation; Epithelial Cells; Flavonoids; Gene Expression; Humans; Imidazoles; Interleukin-13; Interleukin-4; Interleukins; Janus Kinase 2; JNK Mitogen-Activated Protein Kinases; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 3; p38 Mitogen-Activated Protein Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; Tyrphostins; Up-Regulation | 2006 |
Leptin represses matrix metalloproteinase-1 gene expression in LX2 human hepatic stellate cells.
Topics: Base Sequence; Catalase; Cell Line; Down-Regulation; Enzyme Inhibitors; Hepatocytes; Humans; Hydrogen Peroxide; Imidazoles; Janus Kinases; Leptin; Liver Cirrhosis; MAP Kinase Signaling System; Matrix Metalloproteinase 1; Models, Biological; Oligodeoxyribonucleotides, Antisense; Pyridines; RNA, Messenger; STAT3 Transcription Factor; STAT5 Transcription Factor; Tyrphostins | 2007 |
Cardiotrophin-1 induces interleukin-6 synthesis in human umbilical vein endothelial cells.
Topics: Antibodies, Monoclonal; Cells, Cultured; Cycloheximide; Cytokines; Dose-Response Relationship, Drug; Endothelial Cells; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Gene Expression; Humans; Imidazoles; Interleukin-6; Janus Kinase 2; Kinetics; NF-kappa B; p38 Mitogen-Activated Protein Kinases; Pyridines; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sesquiterpenes; STAT3 Transcription Factor; Stilbenes; Tyrphostins; Umbilical Cord | 2006 |
Molecular mechanisms involved in interleukin-4-induced human neutrophils: expression and regulation of suppressor of cytokine signaling.
Topics: Apoptosis; Cycloheximide; Dose-Response Relationship, Drug; Flavonoids; Gene Expression Profiling; Granulocyte Colony-Stimulating Factor; Granulocyte-Macrophage Colony-Stimulating Factor; Humans; Imidazoles; Interleukin-4; Leupeptins; Neutrophils; Pyridines; Receptors, Interleukin-4, Type I; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship; Suppressor of Cytokine Signaling Proteins; Tyrphostins | 2007 |
Modulation of mast cell proteinase-activated receptor expression and IL-4 release by IL-12.
Topics: Animals; Butadienes; Cells, Cultured; Chromones; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Gene Expression Regulation; Imidazoles; Interleukin-12; Interleukin-4; Mast Cells; Mice; Morpholines; Nitriles; Proto-Oncogene Proteins c-akt; Pyridines; Receptors, Proteinase-Activated; RNA, Messenger; Trypsin; Tryptases; Tyrphostins | 2007 |
High-fat diet-induced obesity leads to resistance to leptin-induced cardiomyocyte contractile response.
Topics: Animals; Calcium; Cells, Cultured; Diet, Fat-Restricted; Dietary Fats; Enzyme Inhibitors; Imidazoles; Leptin; Male; Myocardial Contraction; Myocardium; Myocytes, Cardiac; NG-Nitroarginine Methyl Ester; Obesity; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Leptin; Tyrphostins | 2008 |
Prolactin induces chitotriosidase expression in human macrophages through PTK, PI3-K, and MAPK pathways.
Topics: Acetophenones; Benzopyrans; Butadienes; Chromones; Gene Expression Regulation, Enzymologic; Genistein; Hexosaminidases; Humans; Imidazoles; Macrophages; MAP Kinase Signaling System; Monocytes; Morpholines; Nitriles; Phosphatidylinositol 3-Kinases; Phosphorylation; Prolactin; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-akt; Pyridines; Pyrimidines; RNA, Messenger; Tyrphostins | 2009 |
Roles of phosphatidylinositol 3-kinase and p38 mitogen-activated protein kinase in the regulation of protein kinase C-alpha activation in interferon-gamma-stimulated macrophages.
Topics: Animals; Cell Line; Cell Nucleus; Chromones; Enzyme Activation; Enzyme Inhibitors; Female; Imidazoles; Interferon-gamma; Janus Kinase 2; Macrophages; Mice; Mice, Inbred BALB C; Morpholines; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase C-alpha; Pyridines; Signal Transduction; STAT1 Transcription Factor; Trans-Activators; Tyrphostins | 2009 |
Procaspase 8 and Bax are up-regulated by distinct pathways in Streptococcal pyrogenic exotoxin B-induced apoptosis.
Topics: Antibodies; Apoptosis; Bacterial Proteins; bcl-2-Associated X Protein; Caspase 8; Cell Line, Tumor; Enzyme Inhibitors; Exotoxins; fas Receptor; Humans; Imidazoles; Immunoblotting; Integrin alphaVbeta3; Janus Kinase 2; Models, Biological; Mutant Proteins; Phosphorylation; Pyridines; Recombinant Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA Interference; Signal Transduction; STAT1 Transcription Factor; Tyrphostins; Up-Regulation | 2009 |
Rhizoctonia bataticola lectin (RBL) induces mitogenesis and cytokine production in human PBMC via p38 MAPK and STAT-5 signaling pathways.
Topics: Blotting, Western; Cell Proliferation; Cytokines; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Flow Cytometry; Fungal Proteins; Humans; Imidazoles; Interferon-gamma; Interleukin-10; Interleukin-2; Interleukin-2 Receptor alpha Subunit; Interleukin-4; Lectins; Leukocytes, Mononuclear; Mitogens; p38 Mitogen-Activated Protein Kinases; Protein Binding; Pyridines; Rhizoctonia; Signal Transduction; STAT5 Transcription Factor; Tyrphostins | 2010 |
Human apolipoprotein A-I induces cyclooxygenase-2 expression and prostaglandin I-2 release in endothelial cells through ATP-binding cassette transporter A1.
Topics: Apolipoprotein A-I; Apolipoproteins; ATP Binding Cassette Transporter 1; ATP-Binding Cassette Transporters; Cells, Cultured; Cholesterol; Cyclooxygenase 2; Down-Regulation; Drug Synergism; Epoprostenol; Extracellular Signal-Regulated MAP Kinases; Fatty Acids, Nonesterified; Flavonoids; Gene Expression; Human Umbilical Vein Endothelial Cells; Humans; Imidazoles; Janus Kinase 2; Lipoproteins, HDL; Lysophospholipids; p38 Mitogen-Activated Protein Kinases; Pertussis Toxin; Phospholipids; Phosphorylation; Protein Kinase Inhibitors; Pyridines; RNA, Small Interfering; Signal Transduction; Sphingosine; Trypsin; Tyrphostins; Up-Regulation | 2011 |
MAPK and JAK-STAT signaling pathways are involved in the oxidative stress-induced decrease in expression of surfactant protein genes.
Topics: Acetylcysteine; Antioxidants; ATP-Binding Cassette Transporters; Butadienes; Cell Line, Tumor; DNA-Binding Proteins; Humans; Hydrogen Peroxide; Imidazoles; Janus Kinases; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nitriles; Oxidative Stress; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Promoter Regions, Genetic; Protein Binding; Pulmonary Surfactant-Associated Protein A; Pulmonary Surfactant-Associated Protein B; Pulmonary Surfactant-Associated Protein D; Pyridines; RNA, Messenger; Signal Transduction; STAT3 Transcription Factor; Transcription Factors; Tyrphostins | 2012 |
Stimulation of phagocyte adhesion to endothelial cells by modified VLDL and HDL requires scavenger receptor BI.
Topics: Biomarkers; Butadienes; Cell Adhesion; Cyclopentanes; Human Umbilical Vein Endothelial Cells; Humans; Imidazoles; Janus Kinase 2; Lipoproteins, HDL; Lipoproteins, VLDL; Mitogen-Activated Protein Kinases; Neutrophil Activation; Neutrophils; Nitriles; Phagocytes; Pyridines; Scavenger Receptors, Class B; Thiosemicarbazones; Tyrphostins | 2013 |
Polyriboinosinic-polyribocytidylic acid facilitates interleukin-6, and interleukin-8 secretion in human dermal fibroblasts via the JAK/STAT3 and p38 MAPK signal transduction pathways.
Topics: Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fibroblasts; Humans; Imidazoles; Interleukin-6; Interleukin-8; MAP Kinase Signaling System; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Poly I-C; Pyridines; Skin; STAT3 Transcription Factor; Tyrphostins | 2018 |
Combination of 4-hydroperoxy cyclophosphamide and methotrexate inhibits IL-6/sIL-6R-induced RANKL expression in fibroblast-like synoviocytes via suppression of the JAK2/STAT3 and p38MAPK signaling pathway.
Topics: Arthritis, Rheumatoid; Cells, Cultured; Cyclophosphamide; Drug Therapy, Combination; Fibroblasts; Gene Expression Regulation; Humans; Imidazoles; Interleukin-6; Janus Kinase 2; Methotrexate; p38 Mitogen-Activated Protein Kinases; Pyridines; RANK Ligand; Receptors, Interleukin-6; Signal Transduction; STAT3 Transcription Factor; Synoviocytes; Tyrphostins | 2018 |
A novel role of angiotensin II in epidermal cell lineage determination: Angiotensin II promotes the differentiation of mesenchymal stem cells into keratinocytes through the p38 MAPK, JNK and JAK2 signalling pathways.
Topics: Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Angiotensin II Type 2 Receptor Blockers; Animals; Anthracenes; Bone Marrow Cells; Cell Differentiation; Cell Lineage; Cell Movement; Imidazoles; Janus Kinase 2; Janus Kinases; Keratinocytes; Losartan; Male; MAP Kinase Signaling System; Mesenchymal Stem Cells; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Pyridines; Rats; Rats, Wistar; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Tyrphostins | 2019 |