Page last updated: 2024-09-03

san 58035 and sirolimus

san 58035 has been researched along with sirolimus in 2 studies

Compound Research Comparison

Studies
(san 58035)
Trials
(san 58035)
Recent Studies (post-2010)
(san 58035)
Studies
(sirolimus)
Trials
(sirolimus)
Recent Studies (post-2010) (sirolimus)
5811220,7112,36811,516

Protein Interaction Comparison

ProteinTaxonomysan 58035 (IC50)sirolimus (IC50)
Bile salt export pumpHomo sapiens (human)10
ATP-dependent translocase ABCB1Homo sapiens (human)1.25
Cytochrome P450 3A4Homo sapiens (human)2
Cytochrome P450 2C9 Homo sapiens (human)2
Peptidyl-prolyl cis-trans isomerase FKBP1AMus musculus (house mouse)0.001
Cytochrome P450 2C19Homo sapiens (human)4
Serine/threonine-protein kinase mTORHomo sapiens (human)0.0897
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)0.0042
Regulatory-associated protein of mTORHomo sapiens (human)0.225
Target of rapamycin complex subunit LST8Homo sapiens (human)0.225
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)1.9
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)1.1

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abete, C; Dessì, S; Fossarello, M; Mulas, C; Norfo, C; Peiretti, E; Putzolu, M1
Abete, C; Dessì, S; Mandas, A; Massidda, B; Mulas, MF; Pani, A; Pulisci, D1

Other Studies

2 other study(ies) available for san 58035 and sirolimus

ArticleYear
Modulation of cholesterol homeostasis by antiproliferative drugs in human pterygium fibroblasts.
    Investigative ophthalmology & visual science, 2007, Volume: 48, Issue:8

    Topics: Aged; Amides; ATP Binding Cassette Transporter, Subfamily B, Member 1; Caveolin 1; Cell Division; Cells, Cultured; Cholesterol; Cholesterol Esters; Enzyme Inhibitors; Everolimus; Female; Fibroblasts; Homeostasis; Humans; Hypoglycemic Agents; Immunosuppressive Agents; In Vitro Techniques; Male; Middle Aged; Organosilicon Compounds; Pioglitazone; Progesterone; Pterygium; RNA, Messenger; Sirolimus; Sterol O-Acyltransferase; Thiazolidinediones

2007
Cholesterol esters as growth regulators of lymphocytic leukaemia cells.
    Cell proliferation, 2011, Volume: 44, Issue:4

    Topics: Adult; Aged; Amides; Antineoplastic Agents; Cell Proliferation; Cholesterol Esters; Cholesterol, HDL; Everolimus; Humans; Leukemia, Lymphocytic, Chronic, B-Cell; Lipid Metabolism; Lipids; Middle Aged; Organosilicon Compounds; Phytohemagglutinins; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Progesterone; Sirolimus

2011