Page last updated: 2024-09-03

salvinorin a and naltrindole

salvinorin a has been researched along with naltrindole in 6 studies

Compound Research Comparison

Studies
(salvinorin a)
Trials
(salvinorin a)
Recent Studies (post-2010)
(salvinorin a)
Studies
(naltrindole)
Trials
(naltrindole)
Recent Studies (post-2010) (naltrindole)
24771288010139

Protein Interaction Comparison

ProteinTaxonomysalvinorin a (IC50)naltrindole (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0007
Delta-type opioid receptorHomo sapiens (human)0.0006

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (50.00)29.6817
2010's3 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Azar, MR; Cashman, JR; Ghirmai, S1
Fichna, J; Lewellyn, K; Roth, BL; Yan, F; Zjawiony, JK1
Ferreira, D; Polepally, PR; Roth, BL; Vardy, E; White, K; Zjawiony, JK1
Huben, K; Mosier, PD; Polepally, PR; Roth, BL; Setola, V; Vardy, E; Zjawiony, JK1
Fantegrossi, WE; Koreeda, M; Kugle, KM; Valdes, LJ; Woods, JH1
Erlichman, JS; French, LG; John, TF1

Other Studies

6 other study(ies) available for salvinorin a and naltrindole

ArticleYear
Synthesis and pharmacological evaluation of 6-naltrexamine analogs for alcohol cessation.
    Bioorganic & medicinal chemistry, 2009, Sep-15, Volume: 17, Issue:18

    Topics: Alcohol Deterrents; Alcoholism; Animals; Humans; Liver; Male; Mice; Naltrexone; Nociceptin Receptor; Protein Binding; Rats; Rats, Wistar; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Structure-Activity Relationship

2009
Synthesis and biological evaluation of new salvinorin A analogues incorporating natural amino acids.
    Bioorganic & medicinal chemistry letters, 2011, Jan-01, Volume: 21, Issue:1

    Topics: Amino Acids; Diterpenes, Clerodane; Protein Binding; Receptors, Opioid, kappa; Structure-Activity Relationship; Valine

2011
Kappa-opioid receptor-selective dicarboxylic ester-derived salvinorin A ligands.
    Bioorganic & medicinal chemistry letters, 2013, May-15, Volume: 23, Issue:10

    Topics: Camphanes; Diterpenes, Clerodane; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; HEK293 Cells; Humans; Molecular Conformation; Panax notoginseng; Receptors, Opioid, kappa; Salvia; Salvia miltiorrhiza; Structure-Activity Relationship

2013
Michael acceptor approach to the design of new salvinorin A-based high affinity ligands for the kappa-opioid receptor.
    European journal of medicinal chemistry, 2014, Oct-06, Volume: 85

    Topics: Diterpenes, Clerodane; Drug Design; HEK293 Cells; Humans; Ligands; Models, Molecular; Protein Binding; Protein Conformation; Receptors, Opioid, kappa

2014
Kappa-opioid receptor-mediated effects of the plant-derived hallucinogen, salvinorin A, on inverted screen performance in the mouse.
    Behavioural pharmacology, 2005, Volume: 16, Issue:8

    Topics: Analgesics, Opioid; Animals; Behavior, Animal; Benzeneacetamides; Diterpenes; Diterpenes, Clerodane; Hallucinogens; Male; Mice; Naloxone; Naltrexone; Narcotic Antagonists; Piperidines; Psychotropic Drugs; Pyrrolidines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Remifentanil

2005
The antinociceptive effect of salvinorin A in mice.
    European journal of pharmacology, 2006, Sep-18, Volume: 545, Issue:2-3

    Topics: Analgesics; Animals; Diterpenes; Diterpenes, Clerodane; Injections, Spinal; Male; Mice; Naltrexone

2006