Page last updated: 2024-09-03

salvinorin a and etorphine

salvinorin a has been researched along with etorphine in 2 studies

Compound Research Comparison

Studies
(salvinorin a)
Trials
(salvinorin a)
Recent Studies (post-2010)
(salvinorin a)
Studies
(etorphine)
Trials
(etorphine)
Recent Studies (post-2010) (etorphine)
24771287982363
24771281201

Protein Interaction Comparison

ProteinTaxonomysalvinorin a (IC50)etorphine (IC50)
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0074
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0001
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.0018

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Benaderet, TS; Bishop-Mathis, K; Dersch, CM; Partilla, JS; Prisinzano, TE; Rothman, RB; Simpson, DS; Wang, X; Xu, H1
Dai, R; Deng, G; Lee, DY; Liu, J; Liu-Chen, LY; Ma, Z; Xu, W; Yang, L1

Other Studies

2 other study(ies) available for salvinorin a and etorphine

ArticleYear
Differential effects of opioid agonists on G protein expression in CHO cells expressing cloned human opioid receptors.
    Brain research bulletin, 2008, Sep-05, Volume: 77, Issue:1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Benzamides; Blotting, Western; CHO Cells; Cricetinae; Cricetulus; Diterpenes, Clerodane; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Ethylketocyclazocine; Etorphine; Female; Furans; Gene Expression; GTP-Binding Protein alpha Subunits, G12-G13; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Morphine; Oligopeptides; Piperazines; Pyrones; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

2008
Synthesis and biological evaluation of 2-alkyl-2-methoxymethyl-salvinorin ethers as selective κ-opioid receptor agonists.
    Bioorganic & medicinal chemistry letters, 2015, Oct-15, Volume: 25, Issue:20

    Topics: Diterpenes; Dose-Response Relationship, Drug; Humans; Molecular Conformation; Receptors, Opioid, kappa; Structure-Activity Relationship

2015