Page last updated: 2024-09-03

salvinorin a and cep-32496

salvinorin a has been researched along with cep-32496 in 2 studies

Compound Research Comparison

Studies
(salvinorin a)
Trials
(salvinorin a)
Recent Studies (post-2010)
(salvinorin a)
Studies
(cep-32496)
Trials
(cep-32496)
Recent Studies (post-2010) (cep-32496)
247712818016

Protein Interaction Comparison

ProteinTaxonomysalvinorin a (IC50)cep-32496 (IC50)
Tyrosine-protein kinase ABL1Homo sapiens (human)0.006
RAF proto-oncogene serine/threonine-protein kinaseHomo sapiens (human)0.146
Proto-oncogene tyrosine-protein kinase receptor RetHomo sapiens (human)0.0543
Serine/threonine-protein kinase B-rafHomo sapiens (human)0.082
Ephrin type-A receptor 2Homo sapiens (human)0.028
Cytochrome P450 2C19Homo sapiens (human)3.4
Vascular endothelial growth factor receptor 2Homo sapiens (human)0.03
Nuclear receptor coactivator 4Homo sapiens (human)0.0004
Coiled-coil domain-containing protein 6Homo sapiens (human)0.0037

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Kabir, M; Kerns, E; Nguyen, K; Shah, P; Sun, H; Wang, Y; Xu, X; Yu, KR1
Itkin, M; Kabir, M; Mathé, EA; Nguyễn, ÐT; Padilha, EC; Shah, P; Shinn, P; Siramshetty, V; Wang, AQ; Williams, J; Xu, X; Yu, KR; Zhao, T1

Reviews

1 review(s) available for salvinorin a and cep-32496

ArticleYear
Using in vitro ADME data for lead compound selection: An emphasis on PAMPA pH 5 permeability and oral bioavailability.
    Bioorganic & medicinal chemistry, 2022, 02-15, Volume: 56

    Topics: Administration, Oral; Animals; Betamethasone; Biological Availability; Caco-2 Cells; Cell Membrane Permeability; Cells, Cultured; Dexamethasone; Dogs; Dose-Response Relationship, Drug; Humans; Hydrogen-Ion Concentration; Madin Darby Canine Kidney Cells; Mice; Molecular Structure; Neural Networks, Computer; Ranitidine; Rats; Structure-Activity Relationship; Verapamil

2022

Other Studies

1 other study(ies) available for salvinorin a and cep-32496

ArticleYear
Predictive models of aqueous solubility of organic compounds built on A large dataset of high integrity.
    Bioorganic & medicinal chemistry, 2019, 07-15, Volume: 27, Issue:14

    Topics: Drug Discovery; Organic Chemicals; Pharmaceutical Preparations; Solubility

2019