Page last updated: 2024-09-03

safinamide and lazabemide

safinamide has been researched along with lazabemide in 5 studies

Compound Research Comparison

Studies
(safinamide)
Trials
(safinamide)
Recent Studies (post-2010)
(safinamide)
Studies
(lazabemide)
Trials
(lazabemide)
Recent Studies (post-2010) (lazabemide)
199291591141128

Protein Interaction Comparison

ProteinTaxonomysafinamide (IC50)lazabemide (IC50)
Amine oxidase [flavin-containing] BRattus norvegicus (Norway rat)0.03
Amine oxidase [flavin-containing] BHomo sapiens (human)0.077

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's5 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Almos, T; Edmondson, DE; Massari, ME; Rojas, RJ; Scott, R1
Mostert, S; Petzer, A; Petzer, JP2
Abramov, IG; Chirkova, ZV; Filimonov, SI; Kabanova, MV; Petzer, A; Petzer, JP; Suponitsky, KY1
Baykov, S; Chirkova, Z; Engelbrecht, I; Korsakov, M; Osipyan, A; Petzer, A; Petzer, JP; Sapegin, A; Shetnev, A1

Other Studies

5 other study(ies) available for safinamide and lazabemide

ArticleYear
Reversible and irreversible small molecule inhibitors of monoamine oxidase B (MAO-B) investigated by biophysical techniques.
    Bioorganic & medicinal chemistry, 2015, Feb-15, Volume: 23, Issue:4

    Topics: Humans; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Parkinson Disease; Small Molecule Libraries; Thermodynamics

2015
Inhibition of monoamine oxidase by benzoxathiolone analogues.
    Bioorganic & medicinal chemistry letters, 2016, Feb-15, Volume: 26, Issue:4

    Topics: Benzoxazoles; Humans; Inhibitory Concentration 50; Kinetics; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Protein Binding; Protein Isoforms; Structure-Activity Relationship

2016
An evaluation of synthetic indole derivatives as inhibitors of monoamine oxidase.
    Bioorganic & medicinal chemistry letters, 2016, May-01, Volume: 26, Issue:9

    Topics: Crystallography, X-Ray; Models, Molecular; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2016
The evaluation of 1,4-benzoquinones as inhibitors of human monoamine oxidase.
    European journal of medicinal chemistry, 2017, Jul-28, Volume: 135

    Topics: Benzoquinones; Dose-Response Relationship, Drug; Humans; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Structure-Activity Relationship

2017
Novel monoamine oxidase inhibitors based on the privileged 2-imidazoline molecular framework.
    Bioorganic & medicinal chemistry letters, 2019, 01-01, Volume: 29, Issue:1

    Topics: Dose-Response Relationship, Drug; Humans; Imidazoles; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Neurodegenerative Diseases; Structure-Activity Relationship

2019