Page last updated: 2024-09-03

saclofen and gamma-aminobutyric acid

saclofen has been researched along with gamma-aminobutyric acid in 40 studies

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

Compound Research Comparison

Studies
(saclofen)
Trials
(saclofen)
Recent Studies (post-2010)
(saclofen)
Studies
(gamma-aminobutyric acid)
Trials
(gamma-aminobutyric acid)
Recent Studies (post-2010) (gamma-aminobutyric acid)
10702040,2151,4239,631

Protein Interaction Comparison

ProteinTaxonomysaclofen (IC50)gamma-aminobutyric acid (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 2Rattus norvegicus (Norway rat)0.0292
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0332
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0323
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)2.152
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0333
Sodium- and chloride-dependent GABA transporter 1Homo sapiens (human)5.2623
Sodium- and chloride-dependent taurine transporterHomo sapiens (human)354
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)2.51
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent GABA transporter 1Mus musculus (house mouse)6.349
Sodium- and chloride-dependent GABA transporter 2Mus musculus (house mouse)7.0795
Sodium- and chloride-dependent GABA transporter 3Mus musculus (house mouse)8.1283
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent betaine transporterHomo sapiens (human)6.4082
Sodium- and chloride-dependent GABA transporter 3Homo sapiens (human)3.9953
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0333
GABA theta subunitRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 1Rattus norvegicus (Norway rat)0.0292

Research

Studies (40)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's14 (35.00)18.2507
2000's21 (52.50)29.6817
2010's5 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Angst, C; Bettler, B; Bischoff, S; Bittiger, H; Flor, PJ; Froestl, W; Heid, J; Huggel, K; Kaupmann, K; McMaster, G; Mickel, SJ1
Olausson, B; Shyu, BC; Xu, ZQ1
Hei, DL; Mitsushima, D; Terasawa, E1
Denavit-Saubié, M; Foutz, AS; Pierrefiche, O1
Billard, JM; Deisz, RA; Zieglgänsberger, W1
Hoebel, BG; Mark, GP; Rada, PV1
Chapman, C; Herbison, AE; Poulain, DA; Voisin, DL1
Celada, P; Paladini, CA; Tepper, JM2
Fukuoka, M; Kubo, H; Muraki, M; Nakajima, S; Ohkawa, K; Tohda, Y1
Higashi, H; Maeda, H; Shoji, Y; Tanaka, E; Yamamoto, S1
Burrello, N; Calogero, AE; D'Agata, R; Ferrara, E; Fishel, S; Hall, J1
Ajima, A; Kim, DS; Matsuda, Y; Ohki, K; Tanaka, S1
Ezure, K; Miyazaki, M; Tanaka, I1
Bargas, J; Barral, J; Galarraga, E; Toro, S1
Chen, P; Chen, S; Lin, X1
Park, HJ; Park, HS1
Barker, JL; Behar, TN; Greene, CL; Schaffner, AE; Scott, CA1
Elshourbagy, NA; Gager, TL; Hirst, WD; Jenkins, O; Minton, J; Murkitt, KL; Pangalos, M; Price, GW; Punia, PK; Rice, SQ; Shabon, U; Stammers, M; Taylor, SJ; Testa, T; Wood, MD1
Bodnar, RJ; Christian, G; Echo, JA; Lamonte, N; Ragnauth, A; Znamensky, V1
Asahi, Y; Yonehara, N1
Hattori, T; Hida, W; Kikuchi, Y; Kurosawa, H; Ogawa, H; Okabe, S; Shirato, K; Tabata, M; Tun, Y1
Hayakawa, K; Kamata, K; Kimura, M1
Gómez-Villafuertes, R; Gualix, J; Miras-Portugal, MT; Pintor, J2
Boudah, A; Granato, A; Jasmin, L; Ohara, PT; Rabkin, SD1
Fernández-Pascual, S; Martín Del Río, R; Mukala-Nsengu-Tshibangu, A; Tamarit-Rodríguez, J1
Allen, CN; Gompf, HS1
Ovsepian, SV; Vesselkin, NP1
Boehm, S; Dorostkar, MM1
Ghijsen, WE; Lopes da Silva, FH; Zuiderwijk, M1
Archer, DP; Nguyen, KQ; Roth, SH; Samanani, N1
Beitz, AJ; Han, HJ; Kim, HW; Kwon, YB; Lee, JH; Roh, DH; Seo, HS; Yoon, SY1
Aceves, J; Erlij, D; Florán, B; Nava-Asbell, C; Paz-Bermudez, F1
Balon, N; Deschaseaux, F; Maddens, S; Tiberghien, P; Versaux-Botteri, C; Zangiacomi, V1
Faraji, F; Ghasemi, A; Motamedi, F; Zahediasl, S1
Glinka, Y; Hasilo, C; Paraskevas, S; Prud'homme, GJ; Udovyk, O; Wang, Q1
Borisova, T; Dudarenko, M; Pozdnyakova, N1
Jiang, H; Jin, Q; Li, G; Li, Y; Lv, J; Wan, P; Wang, J1
Chang, CH; Grace, AA1

Other Studies

40 other study(ies) available for saclofen and gamma-aminobutyric acid

ArticleYear
Expression cloning of GABA(B) receptors uncovers similarity to metabotropic glutamate receptors.
    Nature, 1997, Mar-20, Volume: 386, Issue:6622

    Topics: Adenylyl Cyclases; Affinity Labels; Amino Acid Sequence; Animals; Azides; Benzoates; Cell Line; Central Nervous System; Cloning, Molecular; COS Cells; DNA, Complementary; Escherichia coli; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Situ Hybridization; Ligands; Molecular Sequence Data; Organophosphorus Compounds; Radioligand Assay; Rats; Receptors, GABA; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Recombinant Proteins; RNA, Messenger; Sequence Alignment

1997
Dorsal column inhibition of nociceptive thalamic cells mediated by gamma-aminobutyric acid mechanisms in the cat.
    Acta physiologica Scandinavica, 1994, Volume: 152, Issue:3

    Topics: Afferent Pathways; Animals; Baclofen; Cats; Dental Pulp; Electric Stimulation; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Homocysteine; Pain; Picrotoxin; Spinal Cord; Thalamus

1994
gamma-Aminobutyric acid is an inhibitory neurotransmitter restricting the release of luteinizing hormone-releasing hormone before the onset of puberty.
    Proceedings of the National Academy of Sciences of the United States of America, 1994, Jan-04, Volume: 91, Issue:1

    Topics: Animals; Baclofen; Behavior, Animal; Bicuculline; Female; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Macaca mulatta; Ovariectomy; Secretory Rate; Sexual Maturation; Statistics as Topic

1994
Effects of GABAB receptor agonists and antagonists on the bulbar respiratory network in cat.
    Brain research, 1993, Mar-05, Volume: 605, Issue:1

    Topics: Animals; Baclofen; Cats; Decerebrate State; Dizocilpine Maleate; Evoked Potentials; Extracellular Space; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Iontophoresis; Medulla Oblongata; Nerve Net; Organophosphorus Compounds; Plethysmography; Receptors, GABA-A; Respiration

1993
Pre- and postsynaptic GABAB receptors of rat neocortical neurons differ in their pharmacological properties.
    Neuroscience letters, 1993, May-14, Volume: 154, Issue:1-2

    Topics: Animals; Baclofen; Cerebral Cortex; Electric Stimulation; Feedback; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Male; Membrane Potentials; Neurons; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Synapses

1993
In vivo modulation of acetylcholine in the nucleus accumbens of freely moving rats: II. Inhibition by gamma-aminobutyric acid.
    Brain research, 1993, Aug-13, Volume: 619, Issue:1-2

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Choline; Dose-Response Relationship, Drug; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Infusions, Parenteral; Kinetics; Male; Muscimol; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Time Factors

1993
Effects of central GABAB receptor modulation upon the milk ejection reflex in the rat.
    Neuroendocrinology, 1996, Volume: 63, Issue:4

    Topics: Animals; Baclofen; Electric Stimulation; Electroencephalography; Female; GABA Agonists; GABA Antagonists; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Injections; Injections, Intraventricular; Microdialysis; Milk Ejection; Oxytocin; Rats; Rats, Wistar; Receptors, GABA-A; Supraoptic Nucleus

1996
GABAergic control of the firing pattern of substantia nigra dopaminergic neurons.
    Advances in pharmacology (San Diego, Calif.), 1998, Volume: 42

    Topics: Animals; Baclofen; Bicuculline; Evoked Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Kinetics; Muscimol; Neurons; Rats; Receptors, GABA-A; Receptors, GABA-B; Substantia Nigra

1998
Role of GABA receptors in the bronchial response: studies in sensitized guinea-pigs.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 1998, Volume: 28, Issue:6

    Topics: Acetylcholine; Animals; Baclofen; Bicuculline; Bronchi; Electric Stimulation; GABA Agonists; gamma-Aminobutyric Acid; Guinea Pigs; Male; Muscimol; Muscle Contraction; Muscle, Smooth; Ovalbumin; Trachea

1998
Mechanisms underlying the enhancement of excitatory synaptic transmission in basolateral amygdala neurons of the kindling rat.
    Journal of neurophysiology, 1998, Volume: 80, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Epilepsy; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin

1998
Striatal, pallidal, and pars reticulata evoked inhibition of nigrostriatal dopaminergic neurons is mediated by GABA(A) receptors in vivo.
    Neuroscience, 1999, Volume: 89, Issue:3

    Topics: Afferent Pathways; Animals; Baclofen; Bicuculline; Corpus Striatum; Dopamine; Electric Stimulation; GABA Antagonists; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Nerve Degeneration; Neurons; Phosphinic Acids; Picrotoxin; Propanolamines; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, GABA-B; Receptors, Presynaptic; Substantia Nigra

1999
Gamma-aminobutyric acid (GABA) A and B receptors mediate the stimulatory effects of GABA on the human sperm acrosome reaction: interaction with progesterone.
    Fertility and sterility, 1999, Volume: 71, Issue:5

    Topics: Acrosome; Analysis of Variance; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Picrotoxin; Progesterone; Prospective Studies; Receptors, GABA-A; Receptors, GABA-B

1999
GABA-mediated representation of temporal information in rat barrel cortex.
    Neuroreport, 1999, Jun-23, Volume: 10, Issue:9

    Topics: Animals; Baclofen; Bicuculline; Brain Chemistry; Evoked Potentials, Somatosensory; GABA Antagonists; gamma-Aminobutyric Acid; Iontophoresis; Rats; Rats, Long-Evans; Somatosensory Cortex; Time Perception; Vibrissae

1999
Excitatory and inhibitory synaptic inputs shape the discharge pattern of pump neurons of the nucleus tractus solitarii in the rat.
    Experimental brain research, 1999, Volume: 129, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; Neural Inhibition; Neurons; Rats; Rats, Wistar; Reaction Time; Receptors, N-Methyl-D-Aspartate; Solitary Nucleus; Strychnine; Synapses

1999
GABAergic presynaptic inhibition of rat neostriatal afferents is mediated by Q-type Ca(2+) channels.
    Neuroscience letters, 2000, Mar-31, Volume: 283, Issue:1

    Topics: Animals; Baclofen; Calcium Channel Blockers; Calcium Channels, Q-Type; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Neostriatum; Neural Inhibition; Presynaptic Terminals; Rats; Rats, Wistar; Receptors, GABA-B

2000
Activation of metabotropic GABAB receptors inhibited glutamate responses in spiral ganglion neurons of mice.
    Neuroreport, 2000, Apr-07, Volume: 11, Issue:5

    Topics: Age Factors; Animals; Animals, Newborn; Auditory Pathways; Baclofen; Bicuculline; Cells, Cultured; Cochlea; Dose-Response Relationship, Drug; Embryo, Mammalian; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hair Cells, Auditory; Mice; Neurons; Polymerase Chain Reaction; Receptors, GABA-B; Spiral Ganglion

2000
Effects of GABA on pancreatic exocrine secretion of rats.
    Journal of Korean medical science, 2000, Volume: 15 Suppl

    Topics: Amylases; Animals; Baclofen; Bicuculline; Cholecystokinin; Dose-Response Relationship, Drug; Electric Stimulation; GABA Antagonists; gamma-Aminobutyric Acid; Gastrin-Releasing Peptide; Hormones; In Vitro Techniques; Pancreas; Rats; Receptors, GABA-A; Secretin; Somatostatin; Tetrodotoxin

2000
GABA receptor antagonists modulate postmitotic cell migration in slice cultures of embryonic rat cortex.
    Cerebral cortex (New York, N.Y. : 1991), 2000, Volume: 10, Issue:9

    Topics: Animals; Baclofen; Bicuculline; Bromodeoxyuridine; Cell Movement; Cellular Senescence; Cerebral Cortex; Chemotaxis; Female; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Intermediate Filament Proteins; Mitosis; Nerve Tissue Proteins; Nestin; Neuroglia; Neurons; Organ Culture Techniques; Picrotoxin; Pregnancy; Rats; Receptors, GABA-A

2000
The human GABA(B1b) and GABA(B2) heterodimeric recombinant receptor shows low sensitivity to phaclofen and saclofen.
    British journal of pharmacology, 2000, Volume: 131, Issue:6

    Topics: Animals; Baclofen; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Humans; Receptors, GABA; Receptors, GABA-B

2000
gamma-Aminobutyric acid receptor subtype antagonists differentially alter opioid-induced feeding in the shell region of the nucleus accumbens in rats.
    Brain research, 2001, Jul-06, Volume: 906, Issue:1-2

    Topics: Animals; Baclofen; Bicuculline; Eating; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; GABA Agonists; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Male; Naltrexone; Narcotic Antagonists; Narcotics; Neurons; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-A; Receptors, GABA-B; Receptors, Opioid

2001
Involvement of GABAergic systems in manifestation of pharmacological activity of desipramine.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:3

    Topics: Animals; Antidepressive Agents, Tricyclic; Baclofen; Desipramine; Freund's Adjuvant; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Muscimol; Picrotoxin; Rats; Rats, Sprague-Dawley; Reaction Time

2001
Role of GABA within the nucleus tractus solitarii in the hypoxic ventilatory decline of awake rats.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2001, Volume: 281, Issue:5

    Topics: Animals; Baclofen; Bicuculline; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Hypoxia; Male; Microdialysis; Microinjections; Muscimol; Neurons; Organophosphorus Compounds; Pulmonary Ventilation; Rats; Rats, Sprague-Dawley; Solitary Nucleus

2001
Mechanism underlying gamma-aminobutyric acid-induced antihypertensive effect in spontaneously hypertensive rats.
    European journal of pharmacology, 2002, Mar-01, Volume: 438, Issue:1-2

    Topics: Animals; Antihypertensive Agents; Baclofen; Blood Pressure; Dose-Response Relationship, Drug; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Muscimol; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Species Specificity; Systole; Time Factors; Vasoconstriction; Vasoconstrictor Agents

2002
GABAB receptor-mediated presynaptic potentiation of ATP ionotropic receptors in rat midbrain synaptosomes.
    Neuropharmacology, 2003, Volume: 44, Issue:3

    Topics: Adenosine Triphosphate; Animals; Baclofen; Calcium; Colforsin; Competitive Bidding; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Fura-2; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Immunohistochemistry; In Vitro Techniques; Mesencephalon; Muscimol; Nerve Tissue Proteins; Picrotoxin; Rats; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X; Synaptosomes; Time Factors

2003
Analgesia and hyperalgesia from GABA-mediated modulation of the cerebral cortex.
    Nature, 2003, Jul-17, Volume: 424, Issue:6946

    Topics: Animals; Baclofen; Bupivacaine; Cerebral Cortex; gamma-Aminobutyric Acid; Hot Temperature; Hyperalgesia; Male; Models, Neurological; Neurons; Pain Threshold; Phentolamine; Rats; Rats, Sprague-Dawley; Synaptic Transmission; Vigabatrin

2003
GABA modulates presynaptic signalling mediated by dinucleotides on rat synaptic terminals.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 308, Issue:3

    Topics: Animals; Baclofen; Calcium; Calcium Signaling; Cyclic AMP-Dependent Protein Kinases; Dinucleoside Phosphates; GABA Agonists; gamma-Aminobutyric Acid; Mesencephalon; Nerve Endings; Presynaptic Terminals; Rats; Receptors, GABA-B

2004
Conversion into GABA (gamma-aminobutyric acid) may reduce the capacity of L-glutamine as an insulin secretagogue.
    The Biochemical journal, 2004, May-01, Volume: 379, Issue:Pt 3

    Topics: 4-Aminobutyrate Transaminase; Adenosine Triphosphate; Allylglycine; Amination; Animals; Aspartic Acid; Baclofen; Bicuculline; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Glutamic Acid; Glutamine; Insulin; Insulin Secretion; Islets of Langerhans; Ketoglutaric Acids; Leucine; Male; Oxidation-Reduction; Perfusion; Potassium Chloride; Rats; Rats, Wistar; Receptors, GABA

2004
GABAergic synapses of the suprachiasmatic nucleus exhibit a diurnal rhythm of short-term synaptic plasticity.
    The European journal of neuroscience, 2004, Volume: 19, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Baclofen; Calcium; Circadian Rhythm; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethylmaleimide; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Male; Membrane Potentials; Models, Neurological; Neural Inhibition; Neuronal Plasticity; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Suprachiasmatic Nucleus; Synapses; Time Factors

2004
Dual effect of GABA on descending monosynaptic excitatory postsynaptic potential in frog lumbar motoneurons.
    Neuroscience, 2004, Volume: 129, Issue:3

    Topics: Animals; Baclofen; Drug Interactions; Electric Stimulation; Evoked Potentials; Excitatory Postsynaptic Potentials; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Lumbosacral Region; Motor Neurons; Rana ridibunda; Spinal Cord; Synapses; Synaptic Transmission

2004
Opposite effects of presynaptic 5-HT3 receptor activation on spontaneous and action potential-evoked GABA release at hippocampal synapses.
    Journal of neurochemistry, 2007, Volume: 100, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Animals, Newborn; Baclofen; Bicuculline; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Indoles; Inhibitory Postsynaptic Potentials; Neurons; Patch-Clamp Techniques; Potassium Chloride; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Tropisetron

2007
Electrically evoked GABA release in rat hippocampus CA1 region and its changes during kindling epileptogenesis.
    Brain research, 2007, Mar-02, Volume: 1135, Issue:1

    Topics: Animals; Anticonvulsants; Baclofen; Electric Stimulation; Epilepsy; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Kindling, Neurologic; Male; Nipecotic Acids; Rats; Rats, Wistar

2007
Pentobarbital enhances gamma-aminobutyric acid-mediated excitation without altering synaptic plasticity in rat hippocampus.
    Anesthesia and analgesia, 2007, Volume: 104, Issue:4

    Topics: Adjuvants, Anesthesia; Animals; Baclofen; Bicarbonates; Bicuculline; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA Modulators; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Neuronal Plasticity; Neurons; Pentobarbital; Rats; Receptors, GABA-A; Receptors, GABA-B; Synaptic Transmission; Time Factors

2007
A spinal muscarinic M2 receptor-GABAergic disinhibition pathway that modulates peripheral inflammation in mice.
    Neuropharmacology, 2007, Volume: 53, Issue:5

    Topics: Adrenal Cortex Hormones; Adrenal Glands; Animals; Anti-Inflammatory Agents; Autonomic Fibers, Preganglionic; Baclofen; Catecholamines; Cell Proliferation; Exudates and Transudates; GABA Antagonists; gamma-Aminobutyric Acid; Image Interpretation, Computer-Assisted; Immunohistochemistry; Inflammation; Male; Mice; Mice, Inbred ICR; Neural Pathways; Neurons; Receptor, Muscarinic M2; Receptors, GABA-A; Receptors, GABA-B; Spinal Cord

2007
GABA(B) receptor activation inhibits dopamine D1 receptor-mediated facilitation of [(3)H]GABA release in substantia nigra pars reticulata.
    Neuropharmacology, 2007, Volume: 53, Issue:5

    Topics: Animals; Baclofen; Benzazepines; Cyclic AMP-Dependent Protein Kinases; Data Interpretation, Statistical; Dopamine Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, GABA-B; Reserpine; Substantia Nigra

2007
Human cord blood-derived hematopoietic and neural-like stem/progenitor cells are attracted by the neurotransmitter GABA.
    Stem cells and development, 2009, Volume: 18, Issue:9

    Topics: AC133 Antigen; Antigens, CD; Baclofen; Bicuculline; Cell Differentiation; Cell Line; Cells, Cultured; Chemotaxis; Colony-Forming Units Assay; Fetal Blood; Flow Cytometry; Fluorescent Antibody Technique; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression; Glycoproteins; Hematopoietic Stem Cells; Humans; Neurons; Peptides; Receptors, GABA-A; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; Stem Cells

2009
Time-dependent effect of GABA on glucose-stimulated insulin secretion from isolated islets in rat.
    Scandinavian journal of clinical and laboratory investigation, 2011, Volume: 71, Issue:6

    Topics: Animals; Baclofen; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Wistar; Time Factors

2011
GABA protects pancreatic beta cells against apoptosis by increasing SIRT1 expression and activity.
    Biochemical and biophysical research communications, 2014, Sep-26, Volume: 452, Issue:3

    Topics: Animals; Apoptosis; Baclofen; Cell Line, Tumor; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression Regulation; Humans; Insulin-Secreting Cells; Muscimol; NAD; Picrotoxin; Primary Cell Culture; Rats; Receptors, GABA-A; Receptors, GABA-B; Signal Transduction; Sirtuin 1; Transcription Factor RelA

2014
New effects of GABAB receptor allosteric modulator rac-BHFF on ambient GABA, uptake/release, Em and synaptic vesicle acidification in nerve terminals.
    Neuroscience, 2015, Sep-24, Volume: 304

    Topics: Allosteric Regulation; Animals; Baclofen; Benzofurans; Cerebral Cortex; Dose-Response Relationship, Drug; Extracellular Space; GABA Agents; gamma-Aminobutyric Acid; Hippocampus; Male; Membrane Potentials; Protons; Rats, Wistar; Receptors, GABA-B; Synaptic Vesicles; Synaptosomes; Tritium

2015
GABAB receptors in the hippocampal dentate gyrus are involved in spatial learning and memory impairment in a rat model of vascular dementia.
    Brain research bulletin, 2016, Volume: 124

    Topics: Animals; Baclofen; Dementia, Vascular; Dentate Gyrus; Disease Models, Animal; GABA Antagonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Male; Memory Disorders; Myocardial Ischemia; Rats; Rats, Sprague-Dawley; Reaction Time; Receptors, GABA-B; Spatial Learning

2016
Inhibitory Modulation of Orbitofrontal Cortex on Medial Prefrontal Cortex-Amygdala Information Flow.
    Cerebral cortex (New York, N.Y. : 1991), 2018, 01-01, Volume: 28, Issue:1

    Topics: Amygdala; Anesthesia; Animals; Baclofen; Bicuculline; Electric Stimulation; Emotions; Excitatory Amino Acid Agonists; Frontal Lobe; GABA Antagonists; gamma-Aminobutyric Acid; Male; Microelectrodes; N-Methylaspartate; Neural Inhibition; Neural Pathways; Neurons; Rats, Sprague-Dawley; Receptors, GABA

2018