Page last updated: 2024-09-03

saclofen and desipramine

saclofen has been researched along with desipramine in 1 studies

Compound Research Comparison

Studies
(saclofen)
Trials
(saclofen)
Recent Studies (post-2010)
(saclofen)
Studies
(desipramine)
Trials
(desipramine)
Recent Studies (post-2010) (desipramine)
1070205,775487414

Protein Interaction Comparison

ProteinTaxonomysaclofen (IC50)desipramine (IC50)
Solute carrier family 22 member 1 Homo sapiens (human)9.18
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.35
Alpha-2A adrenergic receptorHomo sapiens (human)0.0003
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.35
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.0034
Alpha-2B adrenergic receptorHomo sapiens (human)0.0003
Alpha-2C adrenergic receptorHomo sapiens (human)0.0003
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.35
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.0031
Sodium-dependent dopamine transporterRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 6Rattus norvegicus (Norway rat)0.35
Histamine H1 receptorRattus norvegicus (Norway rat)0.0008
Sodium-dependent serotonin transporterHomo sapiens (human)0.1961
5-hydroxytryptamine receptor 7 Rattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 5ARattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 5BRattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.35
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.0003
Histamine H2 receptorCavia porcellus (domestic guinea pig)3.8
Sodium-dependent dopamine transporter Homo sapiens (human)9.9
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.4035
Sodium channel protein type 5 subunit alphaHomo sapiens (human)1.52
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)0.35
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.35
Solute carrier family 22 member 2Rattus norvegicus (Norway rat)10
TransporterRattus norvegicus (Norway rat)7.8

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Asahi, Y; Yonehara, N1

Other Studies

1 other study(ies) available for saclofen and desipramine

ArticleYear
Involvement of GABAergic systems in manifestation of pharmacological activity of desipramine.
    Japanese journal of pharmacology, 2001, Volume: 86, Issue:3

    Topics: Animals; Antidepressive Agents, Tricyclic; Baclofen; Desipramine; Freund's Adjuvant; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Muscimol; Picrotoxin; Rats; Rats, Sprague-Dawley; Reaction Time

2001