Page last updated: 2024-09-03

saclofen and 6-cyano-7-nitroquinoxaline-2,3-dione

saclofen has been researched along with 6-cyano-7-nitroquinoxaline-2,3-dione in 5 studies

Compound Research Comparison

Studies
(saclofen)
Trials
(saclofen)
Recent Studies (post-2010)
(saclofen)
Studies
(6-cyano-7-nitroquinoxaline-2,3-dione)
Trials
(6-cyano-7-nitroquinoxaline-2,3-dione)
Recent Studies (post-2010) (6-cyano-7-nitroquinoxaline-2,3-dione)
1070202,6981353

Protein Interaction Comparison

ProteinTaxonomysaclofen (IC50)6-cyano-7-nitroquinoxaline-2,3-dione (IC50)
Glutamate receptor 1Homo sapiens (human)1.02
Glutamate receptor 2Homo sapiens (human)1.02
Glutamate receptor 3Homo sapiens (human)1.02
Glutamate receptor 4Homo sapiens (human)1.02

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (60.00)18.2507
2000's2 (40.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Higashi, H; Maeda, H; Shoji, Y; Tanaka, E; Yamamoto, S1
Ibrahim, N; Kabashima, N; Setiadji, VS; Shibuya, I; Ueta, Y; Yamashita, H1
Ezure, K; Miyazaki, M; Tanaka, I1
Allen, CN; Gompf, HS1
Boehm, S; Dorostkar, MM1

Other Studies

5 other study(ies) available for saclofen and 6-cyano-7-nitroquinoxaline-2,3-dione

ArticleYear
Mechanisms underlying the enhancement of excitatory synaptic transmission in basolateral amygdala neurons of the kindling rat.
    Journal of neurophysiology, 1998, Volume: 80, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Epilepsy; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin

1998
GABAB receptor-mediated inhibition of spontaneous action potential discharge in rat supraoptic neurons in vitro.
    Brain research, 1998, Nov-30, Volume: 813, Issue:1

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Female; GABA Agonists; GABA Antagonists; In Vitro Techniques; Male; Neural Inhibition; Picrotoxin; Rats; Rats, Wistar; Receptors, GABA-B; Supraoptic Nucleus

1998
Excitatory and inhibitory synaptic inputs shape the discharge pattern of pump neurons of the nucleus tractus solitarii in the rat.
    Experimental brain research, 1999, Volume: 129, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; Neural Inhibition; Neurons; Rats; Rats, Wistar; Reaction Time; Receptors, N-Methyl-D-Aspartate; Solitary Nucleus; Strychnine; Synapses

1999
GABAergic synapses of the suprachiasmatic nucleus exhibit a diurnal rhythm of short-term synaptic plasticity.
    The European journal of neuroscience, 2004, Volume: 19, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Baclofen; Calcium; Circadian Rhythm; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethylmaleimide; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Male; Membrane Potentials; Models, Neurological; Neural Inhibition; Neuronal Plasticity; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Suprachiasmatic Nucleus; Synapses; Time Factors

2004
Opposite effects of presynaptic 5-HT3 receptor activation on spontaneous and action potential-evoked GABA release at hippocampal synapses.
    Journal of neurochemistry, 2007, Volume: 100, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Animals, Newborn; Baclofen; Bicuculline; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Hippocampus; Indoles; Inhibitory Postsynaptic Potentials; Neurons; Patch-Clamp Techniques; Potassium Chloride; Presynaptic Terminals; Rats; Rats, Sprague-Dawley; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Tropisetron

2007