Page last updated: 2024-09-03

saclofen and 2-amino-5-phosphonovalerate

saclofen has been researched along with 2-amino-5-phosphonovalerate in 8 studies

Compound Research Comparison

Studies
(saclofen)
Trials
(saclofen)
Recent Studies (post-2010)
(saclofen)
Studies
(2-amino-5-phosphonovalerate)
Trials
(2-amino-5-phosphonovalerate)
Recent Studies (post-2010) (2-amino-5-phosphonovalerate)
1070204,3931539

Protein Interaction Comparison

ProteinTaxonomysaclofen (IC50)2-amino-5-phosphonovalerate (IC50)
Glutamate receptor ionotropic, NMDA 1 Rattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2A Rattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2BRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2CRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 2DRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 3BRattus norvegicus (Norway rat)0.29
Glutamate receptor ionotropic, NMDA 3ARattus norvegicus (Norway rat)0.29

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (37.50)18.2507
2000's5 (62.50)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, H; Gustafsson, B; Pananceau, M1
Higashi, H; Maeda, H; Shoji, Y; Tanaka, E; Yamamoto, S1
Ezure, K; Miyazaki, M; Tanaka, I1
Kato, K; Mikoshiba, K; Shin, RM1
Greenfield, SA; Mann, EO1
Allen, CN; Gompf, HS1
Ivenshitz, M; Segal, M1
Heinmiller, A; Ting-A-Kee, R; van der Kooy, D; Vargas-Perez, H; Yeh, A1

Other Studies

8 other study(ies) available for saclofen and 2-amino-5-phosphonovalerate

ArticleYear
Short-term facilitation evoked during brief afferent tetani is not altered by long-term potentiation in the guinea-pig hippocampal CA1 region.
    The Journal of physiology, 1998, Apr-15, Volume: 508 ( Pt 2)

    Topics: 2-Amino-5-phosphonovalerate; Adenosine; Animals; Baclofen; Electric Stimulation; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Guinea Pigs; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Membrane Potentials; Neurons, Afferent; Patch-Clamp Techniques; Picrotoxin; Receptors, N-Methyl-D-Aspartate; Synaptic Membranes

1998
Mechanisms underlying the enhancement of excitatory synaptic transmission in basolateral amygdala neurons of the kindling rat.
    Journal of neurophysiology, 1998, Volume: 80, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Amygdala; Animals; Baclofen; Bicuculline; Epilepsy; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Kindling, Neurologic; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin

1998
Excitatory and inhibitory synaptic inputs shape the discharge pattern of pump neurons of the nucleus tractus solitarii in the rat.
    Experimental brain research, 1999, Volume: 129, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Animals; Baclofen; Bicuculline; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Glycine Agents; Neural Inhibition; Neurons; Rats; Rats, Wistar; Reaction Time; Receptors, N-Methyl-D-Aspartate; Solitary Nucleus; Strychnine; Synapses

1999
Polysynaptic excitatory pathways induce heterosynaptic depression in the rat auditory cortex.
    Neuroscience research, 2001, Volume: 40, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Auditory Cortex; Baclofen; Bicuculline; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABA Antagonists; Male; Neural Inhibition; Neural Pathways; Neuronal Plasticity; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Synapses; Synaptic Transmission

2001
Novel modulatory mechanisms revealed by the sustained application of nicotine in the guinea-pig hippocampus in vitro.
    The Journal of physiology, 2003, Sep-01, Volume: 551, Issue:Pt 2

    Topics: 2-Amino-5-phosphonovalerate; alpha7 Nicotinic Acetylcholine Receptor; Animals; Baclofen; Electrophysiology; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; Guinea Pigs; Hippocampus; In Vitro Techniques; Long-Term Potentiation; Male; Neuronal Plasticity; Nicotine; Nicotinic Agonists; Picrotoxin; Receptors, N-Methyl-D-Aspartate; Receptors, Nicotinic

2003
GABAergic synapses of the suprachiasmatic nucleus exhibit a diurnal rhythm of short-term synaptic plasticity.
    The European journal of neuroscience, 2004, Volume: 19, Issue:10

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Analysis of Variance; Animals; Baclofen; Calcium; Circadian Rhythm; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethylmaleimide; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Magnesium; Male; Membrane Potentials; Models, Neurological; Neural Inhibition; Neuronal Plasticity; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Suprachiasmatic Nucleus; Synapses; Time Factors

2004
Simultaneous NMDA-dependent long-term potentiation of EPSCs and long-term depression of IPSCs in cultured rat hippocampal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-25, Volume: 26, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Evoked Potentials; Hippocampus; Long-Term Potentiation; Long-Term Synaptic Depression; Neuronal Plasticity; Neurons; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Quinoxalines; Rats; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin; Thionucleotides; Time Factors

2006
Tegmental pedunculopontine glutamate and GABA-B synapses mediate morphine reward.
    Behavioral neuroscience, 2009, Volume: 123, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Analysis of Variance; Animals; Baclofen; Behavior, Animal; Bicuculline; Conditioning, Operant; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; Male; Morphine; N-Methylaspartate; Narcotics; Pedunculopontine Tegmental Nucleus; Rats; Rats, Wistar; Receptors, GABA-B; Receptors, Glutamate; Reward

2009