Page last updated: 2024-09-02

s 9788 and cyclosporine

s 9788 has been researched along with cyclosporine in 12 studies

Compound Research Comparison

Studies
(s 9788)
Trials
(s 9788)
Recent Studies (post-2010)
(s 9788)
Studies
(cyclosporine)
Trials
(cyclosporine)
Recent Studies (post-2010) (cyclosporine)
49403772170
494030,5473,8026,558

Protein Interaction Comparison

ProteinTaxonomys 9788 (IC50)cyclosporine (IC50)
ATP-binding cassette sub-family C member 3Homo sapiens (human)0.6315
Bile salt export pumpRattus norvegicus (Norway rat)0.6
Bile salt export pumpHomo sapiens (human)3.5
Interleukin-2Mus musculus (house mouse)0.005
ATP-dependent translocase ABCB1Mus musculus (house mouse)0.7
ATP-dependent translocase ABCB1Homo sapiens (human)1.6792
Cytochrome P450 3A4Homo sapiens (human)3.734
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 25.82
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)9.34
Cytochrome P450 3A5Homo sapiens (human)2.06
ATP-dependent translocase ABCB1Mus musculus (house mouse)4.8
Substance-K receptorHomo sapiens (human)4.139
Peptidyl-prolyl cis-trans isomerase BHomo sapiens (human)0.0088
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)9.34
Cytochrome P450 3A7Homo sapiens (human)2.06
Cytochrome P450 2C19Homo sapiens (human)7
Multidrug resistance-associated protein 1 Homo sapiens (human)3.5082
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)9.34
Peptidyl-prolyl cis-trans isomerase A Homo sapiens (human)0.0252
Peptidyl-prolyl cis-trans isomerase FKBP4Homo sapiens (human)0.016
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoformHomo sapiens (human)0.183
Peptidyl-prolyl cis-trans isomerase DHomo sapiens (human)0.0036
Sodium/bile acid cotransporterHomo sapiens (human)1
Reverse transcriptase/RNaseH Human immunodeficiency virus 10.455
Cytochrome P450 3A43 Homo sapiens (human)2.06
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform Mus musculus (house mouse)0.57
Solute carrier organic anion transporter family member 1B3Homo sapiens (human)1.3
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)4.3
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)0.95

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's12 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Atassi, G; Dhainaut, A; Guilbaud, N; Kraus-Berthier, L; Leonce, S; Pierre, A; Regnier, G; Tizot, A1
Faussat, AM; Kühnel, JM; Marie, JP; Perrot, JY; Schwaller, MA1
Berlion, M; Dieterlen, A; Lucas, C; Marchal, S; Merlin, JL; Poullain, MG; Ramacci, C; Schultz, G1
Lucas, C; Marchal, S; Merlin, JL; Paraire, M; Poullain, MG; Ramacci, C1
Gibassier, J; Leclech, G; Lucas, C; Massart, C; Pourquier, P; Raoul, M; Robert, J1
Guerci, A; Guerci, O; Humbert, JC; Marchal, S; Merlin, JL; Missoum, N; Ramacci, C; Tsuruo, T1
Berlion, M; Kernaleguen, D; Le Bot, MA; Riché, C; Robert, J1
Hill, BT; Hosking, LK1
Berlion, M; Kernaleguen, D; Le Bot, MA; Riché, C; Simon, I1
Chapey, C; Hu, YP; Robert, J1
Buée-Scherrer, V; Cecchelli, R; Dehouck, MP; Descamps, L; Duhem, C; Fenart, L; Poullain, MG1

Other Studies

12 other study(ies) available for s 9788 and cyclosporine

ArticleYear
New purines and purine analogs as modulators of multidrug resistance.
    Journal of medicinal chemistry, 1996, Sep-27, Volume: 39, Issue:20

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channels; Doxorubicin; Drug Resistance, Multiple; Female; Leukemia P388; Leukemia, Experimental; Mice; Molecular Structure; Neoplasm Transplantation; Piperidines; Purines; Structure-Activity Relationship; Triazines; Tumor Cells, Cultured; Vincristine

1996
Functional assay of multidrug resistant cells using JC-1, a carbocyanine fluorescent probe.
    Leukemia, 1997, Volume: 11, Issue:7

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Carbocyanines; Drug Resistance, Multiple; Flow Cytometry; Fluorescent Dyes; Humans; Rhodamine 123; Rhodamines; Spectrometry, Fluorescence; Tumor Cells, Cultured

1997
Influence of S9788, a new modulator of multidrug resistance, on the cellular accumulation and subcellular distribution of daunorubicin in P-glycoprotein-expressing MCF7 human breast adenocarcinoma cells.
    Cytometry, 1995, Aug-01, Volume: 20, Issue:4

    Topics: Adenocarcinoma; ATP Binding Cassette Transporter, Subfamily B, Member 1; Breast Neoplasms; Cell Nucleus; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Female; Flow Cytometry; Humans; Neoplasm Proteins; Piperidines; Subcellular Fractions; Triazines; Tumor Cells, Cultured; Verapamil

1995
[Effect of the modality of exposure on the action of S9788 on the modulation of multidrug resistance of human tumor cell lines].
    Bulletin du cancer, 1994, Volume: 81, Issue:10

    Topics: Adenocarcinoma; Antineoplastic Agents; Breast Neoplasms; Cyclosporine; Daunorubicin; Drug Resistance, Multiple; Humans; Leukemia; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1994
Cyclosporin A, verapamil and S9788 reverse doxorubicin resistance in a human medullary thyroid carcinoma cell line.
    Anti-cancer drugs, 1995, Volume: 6, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Carcinoma, Medullary; Cyclosporine; Doxorubicin; Drug Resistance, Multiple; Drug Synergism; Glutathione; Glutathione Transferase; Humans; Neoplasm Proteins; Piperidines; Polymerase Chain Reaction; RNA, Messenger; RNA, Neoplasm; Thyroid Neoplasms; Triazines; Verapamil

1995
[Pharmacological properties of S9788, a new modulator of multidrug resistance].
    Bulletin du cancer, 1994, Volume: 81, Issue:2

    Topics: Adjuvants, Immunologic; Antineoplastic Agents; Cyclosporine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Humans; Piperidines; Spectrometry, Fluorescence; Triazines; Tumor Cells, Cultured; Vinblastine; Vincristine

1994
Comparative evaluation of S9788, verapamil, and cyclosporine A in K562 human leukemia cell lines and in P-glycoprotein-expressing samples from patients with hematologic malignancies.
    Blood, 1994, Jul-01, Volume: 84, Issue:1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Cyclosporine; Doxorubicin; Drug Resistance; Female; Humans; Leukemia; Male; Membrane Glycoproteins; Middle Aged; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1994
Modulation of anthracycline accumulation and metabolism in rat hepatocytes in culture by three revertants of multidrug resistance.
    Cancer chemotherapy and pharmacology, 1994, Volume: 35, Issue:1

    Topics: Animals; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cells, Cultured; Cyclosporine; Drug Resistance, Multiple; Liver; Male; Piperidines; Rats; Rats, Sprague-Dawley; Triazines; Up-Regulation; Verapamil

1994
Differential effectiveness of a range of novel drug-resistance modulators, relative to verapamil, in influencing vinblastine or teniposide cytotoxicity in human lymphoblastoid CCRF-CEM sublines expressing classic or atypical multidrug resistance.
    Cancer chemotherapy and pharmacology, 1994, Volume: 33, Issue:4

    Topics: Cyclosporine; Dihydropyridines; Dose-Response Relationship, Drug; Drug Resistance; Drug Screening Assays, Antitumor; Flunarizine; Humans; Leukemia, T-Cell; Piperidines; Quinidine; Teniposide; Triazines; Tumor Cells, Cultured; Verapamil; Vinblastine

1994
[Effect of S9788, cyclosporin A and verapamil on intracellular accumulation of doxorubicin, daunorubicin and daunorubicinol in primary rat hepatocyte culture].
    Annales de biologie clinique, 1996, Volume: 54, Issue:1

    Topics: Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cells, Cultured; Cyclosporine; Daunorubicin; Doxorubicin; Drug Resistance, Multiple; Liver; Piperidines; Rats; Rats, Sprague-Dawley; Triazines; Verapamil

1996
Relationship between the inhibition of azidopine binding to P-glycoprotein by MDR modulators and their efficiency in restoring doxorubicin intracellular accumulation.
    Cancer letters, 1996, Dec-03, Volume: 109, Issue:1-2

    Topics: Affinity Labels; Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cyclosporine; Cyclosporins; Dihydropyridines; Doxorubicin; Drug Resistance, Multiple; Humans; Mice; Nicardipine; Piperidines; Triazines; Tumor Cells, Cultured; Verapamil

1996
Inhibition of P-glycoprotein: rapid assessment of its implication in blood-brain barrier integrity and drug transport to the brain by an in vitro model of the blood-brain barrier.
    Pharmaceutical research, 1998, Volume: 15, Issue:7

    Topics: Animals; Antibiotics, Antineoplastic; Antineoplastic Agents; Antineoplastic Agents, Phytogenic; Astrocytes; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Blood-Brain Barrier; Brain; Calcium Channel Blockers; Cattle; Coculture Techniques; Cyclosporine; Doxorubicin; Endothelium, Vascular; Immunosuppressive Agents; Piperidines; Predictive Value of Tests; Rats; Triazines; Verapamil; Vincristine

1998