s 11568 has been researched along with dihydropyridines in 15 studies
Studies (s 11568) | Trials (s 11568) | Recent Studies (post-2010) (s 11568) | Studies (dihydropyridines) | Trials (dihydropyridines) | Recent Studies (post-2010) (dihydropyridines) |
---|---|---|---|---|---|
16 | 0 | 0 | 5,022 | 529 | 969 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 13 (86.67) | 18.2507 |
2000's | 2 (13.33) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Mikkelsen, EO; Nyborg, NB; Poulsen, SH | 1 |
Atkinson, J; Bray-des Boscs, L; Capdeville-Atkinson, C; Chillon, JM; Hoffman, M; Lartaud, I; Makki, T; Nicolas, JP | 1 |
Giesen-Crouse, E; Morain, P; Peglion, JL | 1 |
Biondi, ML; Feletou, M; Peglion, JL; Vanhoutte, PM; Vilaine, JP; Villeneuve, N | 1 |
Abraham, C; Aptel, H; Lombet, A; Nagel, N; Peglion, JL; Randle, JC; Renaud, JF | 1 |
Péglion, JL; Randle, JC; Renaud, JF | 1 |
McFalls, EO; Sassen, LM; Van der Zande, J; Verdouw, PD | 1 |
Mulvany, MJ; Nyborg, NC; Prieto, D | 2 |
Eleno, N; Flores, O; López-Novoa, JM; Montañés, I | 1 |
Bourachot, ML; Crouzel, C; Fuseau, C; Syrota, A; Valette, H | 1 |
Crouzel, C; Dollé, F; Duval, R; Fuseau, C; Hinnen, F; Péglion, JL; Valette, H | 1 |
Crouzel, C; Dollé, F; Fuseau, C; Hinnen, F; Péglion, JL; Valette, H | 1 |
Coulon, C; Crouzel, C; Dollé, F; Fuseau, C; Guenther, I; Hinnen, F; Péglion, JL; Valette, H | 2 |
15 other study(ies) available for s 11568 and dihydropyridines
Article | Year |
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Stereoselective pharmacodynamic action of (+)-S-12967 and (-)-S-12968, isomers of a new slow acting 1,4-dihydropyridine derivative with calcium channel agonistic and antagonistic effects on rat aorta.
Topics: Animals; Aorta; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; In Vitro Techniques; Male; Nifedipine; Potassium Chloride; Rats; Rats, Inbred Strains; Stereoisomerism; Structure-Activity Relationship; Vasoconstriction | 1992 |
Haemodynamic effects of a new dihydropyridine calcium entry blocker, S-12968-(-), in a rat model of cardiovascular calcium overload.
Topics: Animals; Blood Pressure; Body Weight; Calcium; Calcium Channel Blockers; Cardiac Output; Cholecalciferol; Dihydropyridines; Heart Rate; Hemodynamics; Magnesium; Male; Nicotine; Nifedipine; Nitroprusside; Rats; Stereoisomerism; Vascular Resistance | 1992 |
Ca2+ channel inhibition in a rat osteoblast-like cell line, UMR 106, by a new dihydropyridine derivative, S11568.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Barium; Calcium Channel Blockers; Cell Line; Dihydropyridines; Electrophysiology; Osteoblasts; Rats | 1992 |
The calcium channel antagonist S 11568 causes endothelium-dependent relaxation in canine arteries.
Topics: Animals; Arginine; Calcium Channel Blockers; Cyclic GMP; Dihydropyridines; Dogs; Endothelium, Vascular; Female; Hemoglobins; In Vitro Techniques; Male; Methylene Blue; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; omega-N-Methylarginine | 1991 |
Ca2+ channel inhibition by a new dihydropyridine derivative, S11568, and its enantiomers S12967 and S12968.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Binding, Competitive; Calcium Channel Blockers; Calcium Radioisotopes; Cell Line; Dihydropyridines; Electrophysiology; Guinea Pigs; Heart; In Vitro Techniques; Inosine Triphosphate; Isradipine; Male; Muscle, Smooth, Vascular; Myocardium; Oxadiazoles; Rats; Ryanodine; Stereoisomerism | 1990 |
Inhibition of L-type but not T-type calcium channel current by a new dihydropyridine derivative, S11568.
Topics: Animals; Barium; Calcium Channel Blockers; Calcium Channels; Chick Embryo; Dihydropyridines; Heart | 1991 |
Cardiovascular profile of the new dihydropyridine derivative S12968.
Topics: Anesthesia; Animals; Calcium Channel Blockers; Dihydropyridines; Female; Heart; Heart Conduction System; Hemodynamics; Male; Muscle, Smooth, Vascular; Myocardial Contraction; Myocardium; Oxygen Consumption; Regional Blood Flow; Swine | 1991 |
(+)-S-12967 and (-)-S-12968: 1,4-dihydropyridine stereoisomers with calcium channel agonistic and antagonistic properties in rat resistance arteries.
Topics: Animals; Calcium; Calcium Channel Agonists; Calcium Channel Blockers; Dihydropyridines; In Vitro Techniques; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Rats; Rats, Inbred Strains; Vascular Resistance | 1991 |
Effects of a new dihydropyridine derivative, S12968 (pranedipine), and its stereoisomer, S12967, on renal effects of endothelin-1.
Topics: Animals; Calcium Channel Blockers; Dihydropyridines; Endothelins; Glomerular Filtration Rate; Kidney; Kidney Function Tests; Male; Rats; Rats, Wistar; Renal Circulation; Sodium; Stereoisomerism; Urodynamics; Vascular Resistance | 1994 |
Canine myocardial dihydropyridine binding sites: a positron emission tomographic study with the calcium channel inhibitor 11C-S11568.
Topics: Animals; Binding Sites; Blood Pressure; Calcium Channel Blockers; Carbon Radioisotopes; Coronary Vessels; Dihydropyridines; Dogs; Female; Heart; Heart Rate; Isradipine; Myocardium; Tomography, Emission-Computed | 1994 |
Effects of (+)-S-12967 and (-)-S-12968, two enantiomers of a new slow-acting 1,4-dihydropyridine, on rat coronary resistance arteries.
Topics: Animals; Calcium Channel Blockers; Calcium Chloride; Coronary Vessels; Dihydropyridines; Dose-Response Relationship, Drug; Hydrogen-Ion Concentration; Male; Muscle Contraction; Muscle, Smooth, Vascular; Potassium Chloride; Rats; Rats, Wistar; Serotonin; Stereoisomerism; Vascular Resistance; Vasodilator Agents | 1993 |
Synthesis of two optically active calcium channel antagonists labelled with carbon-11 for in vivo cardiac PET imaging.
Topics: Amlodipine; Animals; Binding, Competitive; Calcium Channel Blockers; Carbon Radioisotopes; Chromatography, High Pressure Liquid; Dihydropyridines; Dogs; Heart; Heart Diseases; Isotope Labeling; Isradipine; Magnetic Resonance Spectroscopy; Muscle, Smooth, Vascular; Myocardium; Reproducibility of Results; Stereoisomerism; Tomography, Emission-Computed | 1997 |
Synthesis and characterization of a 11C-labelled derivative of S12968: an attempt to image in vivo brain calcium channels.
Topics: Animals; Blood-Brain Barrier; Brain; Calcium Channel Blockers; Calcium Channels; Dihydropyridines; Male; Rats; Rats, Sprague-Dawley; Stereoisomerism; Structure-Activity Relationship; Tissue Distribution; Tomography, Emission-Computed | 1998 |
Myocardial kinetics of the (11)C-labeled enantiomers of the Ca(2+) channel inhibitor S11568: an in vivo study.
Topics: Animals; Calcium Channel Blockers; Carbon Radioisotopes; Coronary Circulation; Dihydropyridines; Dogs; Female; Heart; Male; Myocardium; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tomography, Emission-Computed | 2001 |
In vivo quantification of myocardial dihydropyridine binding sites: a PET study in dogs.
Topics: Animals; Binding Sites; Calcium Channel Blockers; Calcium Channels, L-Type; Carbon Radioisotopes; Dihydropyridines; Dogs; Female; Heart; Myocardium; Time Factors; Tomography, Emission-Computed | 2002 |