Page last updated: 2024-09-02

rx 821002 and yohimbine

rx 821002 has been researched along with yohimbine in 61 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(yohimbine)
Trials
(yohimbine)
Recent Studies (post-2010) (yohimbine)
3170455,893253532

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)yohimbine (IC50)
Alpha-2A adrenergic receptorHomo sapiens (human)0.0353
Cytochrome P450 2D6Homo sapiens (human)1.02
D(2) dopamine receptorHomo sapiens (human)2.06
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)1.3
Alpha-2B adrenergic receptorHomo sapiens (human)0.0428
Alpha-2C adrenergic receptorHomo sapiens (human)0.0466
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.126
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.0682
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)1.3
Alpha-1D adrenergic receptorHomo sapiens (human)1.013
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.126
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.074
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)1.3
5-hydroxytryptamine receptor 6Homo sapiens (human)1.689

Research

Studies (61)

TimeframeStudies, this research(%)All Research%
pre-19902 (3.28)18.7374
1990's44 (72.13)18.2507
2000's12 (19.67)29.6817
2010's3 (4.92)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Denis-Pouxviel, C; Devedjian, JC; Esclapez, F; Paris, H1
Neubig, RR; Porter, AC; Uhlén, S1
Harms, GS; Lohse, MJ; Steinmeyer, R; Vilardaga, JP1
Paris, H; Remaury, A1
Leslie, FM; Raymon, HK; Smith, TD1
Blaxall, HS; Bylund, DB; Lawhead, RG1
Litthauer, D; Oelofsen, W; van de Venter, M1
Uhlén, S; Wikberg, JE1
Czerwiec, E; De Backer, JP; De Potter, W; De Vos, H; Vauquelin, G1
Berlan, M; Galitzky, J; Montastruc, P; Tran, MA1
Berlan, M; Galitzky, J; Lafontan, M; Larrouy, D1
Lafontan, M; Langin, D; Paris, H1
Carpéné, C; Galitzky, J; Lafontan, M; Langin, D; Larrouy, D1
Berlan, M; Galitzky, J; Lafontan, M; Montastruc, JL; Senard, JM; Stillings, M1
Berlan, M; Estan, L; Montastruc, JL; Senard, JM; Tran, MA1
Lafontan, M; Langin, D; Paris, H; Stillings, MR1
Carpéné, C; Lafontan, M; Langin, D; Saulnier-Blache, JS1
Hussain, JF; Kendall, DA; Pinthong, D; Wilson, VG1
Berlie, JR; Blaxall, HS; Bylund, DB; Chacko, DM; Cooley, ME; Iversen, LJ1
Szabo, B; Urban, R1
Blaylock, NA; Kendall, DA; Wilson, VG; Wright, IK1
Halme, M; Savola, JM; Scheinin, M; Sjöholm, B1
Erdbrügger, W; Michel, MC; Otto, T; Raulf, M1
Evans, RG; Haynes, JM1
Starke, K; Szabo, B; Urban, R1
Blaxall, HS; Bylund, DB; Iversen, LJ; O'Rourke, MF1
Ala-Uotila, S; Kurose, H; Marjamäki, A; Oker-Blom, C; Pohjanoksa, K; Scheinin, M; Sizmann, D1
Bylund, DB; Iversen, LJ; Lomasney, JW; O'Rourke, MF1
Berlan, M; Galitzky, J; Le Corre, P; Le Verge, R1
Etgen, AM; Karkanias, GB1
Clarke, RW; Harris, J1
De Backer, JP; De Keyser, J; De Vos, H; Van Liefde, I; Vauquelin, G1
Blandizzi, C; Carignani, D; Colucci, R; Crema, F; Del Tacca, M; Lazzeri, G; Natale, G1
Savola, JM; Savola, MK1
Bylund, DB; Cerutis, DR; Deupree, JD; Hinton, KA1
Elliott, J1
Goldstein, I; Huang, YH; Moreland, RB; Traish, AM1
Akerman, KE; Cockcroft, V; Huifang, G; Jansson, CC; Kukkonen, JP; Savola, JM; Wurster, S1
Dambrova, M; Gu, Y; Näsman, J; Schiöth, HB; Uhlén, S; Wikberg, JE; Wikberg-Matsson, A1
Birdsall, NJ; Lazareno, S; Leppik, RA; Mynett, A1
Bach, KB; Mitchell, GS1
Cleale, RM; Hadcock, JR; Ingling, JM; Pausch, MH; Search, DJ1
Audinot, V; Chaput, C; Gavaudan, S; Millan, MJ; Newman-Tancredi, A; Nicolas, JP; Richard, N; Touzard, M; Verrièle, L1
Caramona, MM; Figueiredo, IV; Guimarães, S; Moura, D; Paiva, MQ1
Holmberg, M; Kurose, H; Miettinen, R; Scheinin, M1
Hillilä, M; Lähdesmäki, J; Pyykkö, K; Scheinin, M; Sjöholm, B1
McAllister, KH; Rey, B1
Cockcroft, V; Frang, H; Marjamäki, A; Pihlavisto, M; Scheinin, M1
Benamour, K; Chang-Fong, J; Cussac, M; Morand, JM; Szymonski, B; Thomasson, F1
Bylund, DB; Gerety, ME; Happe, HK; Murrin, LC1
Akerman, KE; Jansson, CC; Kukkonen, JP1
McAllister, KH1
De Luca, LA; Menani, JV; Moreira, Tdos S; Renzi, A; Takakura, AC1
De Luca, LA; dos Santos Moreira, T; Menani, JV; Renzi, A; Takakura, AC1
Fagerholm, V; Holmberg, M; Scheinin, M1
Fagerholm, V; Hein, L; Philipp, M; Scheinin, M1
Amano, T; Ebiko, M; Kimura, Y; Sakurada, S; Yonezawa, A; Yoshizumii, M1
de Castro Perez, A; de Francischi, JN; Gama Duarte, ID; Romero, TR1
Arszol, C; Bartenstein, P; Böning, G; Cumming, P; Josef Gildehaus, F; Mille, E; Rominger, A; Wängler, B1
Almeida, RL; Constancio, J; David, RB; De Luca, LA; Fracasso, JF; Menani, JV1
Alves, TB; Antunes, VR; Colombari, E; Ferreira-Neto, HC; Menani, JV; Moreira, TS; Takakura, AC; Totola, LT1

Other Studies

61 other study(ies) available for rx 821002 and yohimbine

ArticleYear
Further characterization of human alpha 2-adrenoceptor subtypes: [3H]RX821002 binding and definition of additional selective drugs.
    European journal of pharmacology, 1994, Jan-24, Volume: 252, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cell Line; Dioxanes; Humans; Idazoxan; Plasmids; Radioligand Assay; Receptors, Adrenergic, alpha; Transfection

1994
The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Dibenzazepines; Humans; Imidazoles; Indoles; Isoindoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2

1994
Molecular basis of inverse agonism in a G protein-coupled receptor.
    Nature chemical biology, 2005, Volume: 1, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Cell Line; Fluorescence Resonance Energy Transfer; Humans; Ligands; Protein Binding; Receptors, Adrenergic, alpha-2; Receptors, G-Protein-Coupled; Signal Transduction

2005
The insulin-secreting cell line, RINm5F, expresses an alpha-2D adrenoceptor and nonadrenergic idazoxan-binding sites.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:1

    Topics: Adenosine Diphosphate; Adrenergic alpha-Antagonists; Animals; Binding Sites; Brimonidine Tartrate; Cell Line; Cyclic AMP; Dioxanes; GTP-Binding Proteins; Idazoxan; Immunoblotting; Insulin; Insulin Secretion; Kinetics; Membranes; Pertussis Toxin; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Tritium; Virulence Factors, Bordetella; Yohimbine

1992
Further pharmacological characterization of [3H]idazoxan binding sites in rat brain: evidence for predominant labeling of alpha 2-adrenergic receptors.
    Brain research, 1992, Jun-12, Volume: 582, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Buffers; Dioxanes; Epinephrine; Idazoxan; Male; Phentolamine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Receptors, Drug; Tritium; Yohimbine

1992
Alpha-2A is the predominant alpha-2 adrenergic receptor subtype in human spinal cord.
    Anesthesiology, 1992, Volume: 77, Issue:5

    Topics: Adrenergic alpha-Antagonists; Dioxanes; Humans; Idazoxan; In Vitro Techniques; Indicators and Reagents; Receptors, Adrenergic, alpha; Spinal Cord; Yohimbine

1992
The effect of high concentrations of alpha 2-adrenoceptor antagonists on the lipolytic responsiveness of isolated human adipocytes.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 103, Issue:2

    Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Dioxanes; Female; Humans; Idazoxan; Isoproterenol; Lipolysis; Norepinephrine; Propanolamines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine

1992
Delineation of three pharmacological subtypes of alpha 2-adrenoceptor in the rat kidney.
    British journal of pharmacology, 1991, Volume: 104, Issue:3

    Topics: Animals; Binding, Competitive; Computer Simulation; Dioxanes; Guanabenz; Idazoxan; In Vitro Techniques; Kidney; Male; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1991
[3H]rauwolscine behaves as an agonist for the 5-HT1A receptors in human frontal cortex membranes.
    European journal of pharmacology, 1991, May-25, Volume: 207, Issue:1

    Topics: Adrenergic alpha-Antagonists; Aged; Dioxanes; Frontal Lobe; GTP-Binding Proteins; Guanine Nucleotides; Humans; Idazoxan; In Vitro Techniques; Kinetics; Membranes; Middle Aged; Mollusk Venoms; Phentolamine; Receptors, Adrenergic, alpha; Receptors, Serotonin; Yohimbine

1991
Anorectic effect of alpha 2-antagonists in dog: effect of acute and chronic treatment.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 39, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Appetite Depressants; Blood Glucose; Blood Platelets; Body Weight; Catecholamines; Cell Membrane; Dioxanes; Dogs; Fatty Acids, Nonesterified; Feeding Behavior; Idazoxan; Imidazoles; Insulin; Male; Nadolol; Yohimbine

1991
New tools for human fat cell alpha-2A adrenoceptor characterization. Identification on membranes and on intact cells using the new antagonist [3H]RX821002.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 252, Issue:1

    Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Adult; Dioxanes; Dioxins; Female; Guanosine Triphosphate; Humans; Idazoxan; In Vitro Techniques; Kinetics; Magnesium; Middle Aged; Receptors, Adrenergic, alpha; Tritium; Yohimbine

1990
Binding of [3H]idazoxan and of its methoxy derivative [3H] RX821002 in human fat cells: [3H]idazoxan but not [3H] RX821002 labels additional non-alpha 2-adrenergic binding sites.
    Molecular pharmacology, 1990, Volume: 37, Issue:6

    Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Binding Sites; Brimonidine Tartrate; Cell Membrane; Cystamine; Dioxanes; Dioxins; Epinephrine; Female; Humans; Idazoxan; Magnesium Chloride; Phenoxybenzamine; Potassium Chloride; Quinoxalines; Tritium; Yohimbine

1990
Non-adrenergic sites for imidazolines are not directly involved in the alpha 2-adrenergic antilipolytic effect of UK 14304 in rat adipocytes.
    Biochemical pharmacology, 1990, Aug-01, Volume: 40, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Bucladesine; Cell Membrane; Colforsin; Dioxanes; Idazoxan; Kinetics; Lipolysis; Phentolamine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1990
Identification of human platelet alpha 2-adrenoceptors with a new antagonist [3H]-RX821002, a 2-methoxy derivative of idazoxan.
    British journal of pharmacology, 1990, Volume: 100, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Blood Platelets; Brimonidine Tartrate; Dioxanes; Epinephrine; Humans; Idazoxan; In Vitro Techniques; Kinetics; Male; Membranes; Oxymetazoline; Prazosin; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha; Yohimbine

1990
Reserpine induces vascular alpha 2-adrenergic supersensitivity and platelet alpha 2-adrenoceptor up-regulation in dog.
    British journal of pharmacology, 1990, Volume: 101, Issue:2

    Topics: Adipose Tissue; Animals; Blood Platelets; Blood Pressure; Cardiovascular System; Catecholamines; Cell Membrane; Clonidine; Dioxanes; Dogs; Heart Rate; Idazoxan; Male; Norepinephrine; Posture; Prazosin; Receptors, Adrenergic, alpha; Reserpine; Up-Regulation; Yohimbine

1990
[3H]RX821002: a new tool for the identification of alpha 2A-adrenoceptors.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Adrenergic alpha-Antagonists; Binding, Competitive; Catecholamines; Cell Membrane; Colforsin; Cyclic AMP; Dioxanes; Dioxins; Humans; Idazoxan; Kinetics; Radioligand Assay; Receptors, Adrenergic, alpha; Tumor Cells, Cultured; Yohimbine

1989
Imidazolinic radioligands for the identification of hamster adipocyte alpha 2-adrenoceptors.
    European journal of pharmacology, 1989, Nov-21, Volume: 171, Issue:2-3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Clonidine; Cricetinae; Dioxanes; Idazoxan; Imidazoles; In Vitro Techniques; Kinetics; Lipid Metabolism; Lipolysis; Male; Mesocricetus; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha; Yohimbine

1989
Comparison of the interaction of agmatine and crude methanolic extracts of bovine lung and brain with alpha 2-adrenoceptor binding sites.
    British journal of pharmacology, 1995, Volume: 115, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Binding, Competitive; Brimonidine Tartrate; Cattle; Cerebral Cortex; Clonidine; Dioxanes; Idazoxan; Imidazoles; Lung; Methanol; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Yohimbine

1995
Alpha-2 adrenergic receptors in the bovine retina. Presence of only the alpha-2D subtype.
    Investigative ophthalmology & visual science, 1995, Volume: 36, Issue:9

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cattle; Dioxanes; Idazoxan; Pineal Gland; Radioligand Assay; Receptors, Adrenergic, alpha-2; Retina; Yohimbine

1995
Mechanism of sympathoinhibition by imidazolines.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzazepines; Brimonidine Tartrate; Dioxanes; Hemodynamics; Idazoxan; Imidazoles; Oxazoles; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1995
The relationship between density of alpha-adrenoceptor binding sites and contractile responses in several porcine isolated blood vessels.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: 5'-Nucleotidase; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Cell Membrane; Dioxanes; Dose-Response Relationship, Drug; Drug Interactions; Ear, External; Idazoxan; Male; Microscopy, Electron; Muscle Contraction; Muscle, Smooth, Vascular; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Splenic Artery; Structure-Activity Relationship; Swine; Veins; Yohimbine

1995
Recombinant human alpha 2-adrenoceptor subtypes: comparison of [3H]rauwolscine, [3H]atipamezole and [3H]RX821002 as radioligands.
    Biochimica et biophysica acta, 1995, Apr-28, Volume: 1266, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Binding, Competitive; Buffers; Cell Line; Dioxanes; Humans; Idazoxan; Imidazoles; Kinetics; Mice; Radioligand Assay; Recombinant Proteins; Yohimbine

1995
Does [3H]2-methoxy-idazoxan (RX 821002) detect more alpha-2-adrenoceptor agonist high-affinity sites than [3H]rauwolscine? A comparison of nine tissues and cell lines.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 273, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cell Line; Dioxanes; Epinephrine; Female; Guinea Pigs; Humans; Idazoxan; Male; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

1995
Characterization of binding sites for [3H]-idazoxan, [3H]-P-aminoclonidine and [3H]-rauwolscine in the kidney of the dog.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:8

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Clonidine; Dioxanes; Dogs; GTP-Binding Proteins; Idazoxan; Imidazoline Receptors; Kidney; Male; Radioligand Assay; Receptors, Drug; Yohimbine

1994
Sympathoinhibition by rilmenidine in conscious rabbits: involvement of alpha 2-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 348, Issue:6

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Catecholamines; Decerebrate State; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Electrodes, Implanted; Female; Heart Rate; Hemodynamics; Idazoxan; Kidney; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1993
Characterization of [3H]RX821002 binding to alpha-2 adrenergic receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 268, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Cattle; CHO Cells; Cricetinae; Dioxanes; Female; Idazoxan; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

1994
Similar ligand binding in recombinant human alpha 2 C2-adrenoceptors produced in mammalian, insect and yeast cells.
    European journal of pharmacology, 1994, Mar-15, Volume: 267, Issue:1

    Topics: Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Cells, Cultured; Chlorpromazine; Dioxanes; Humans; Idazoxan; Immunoblotting; Mammary Neoplasms, Experimental; Mice; Molecular Sequence Data; Moths; Oxymetazoline; Prazosin; Receptors, Adrenergic, alpha; Recombinant Proteins; Saccharomyces cerevisiae; Transfection; Tumor Cells, Cultured; Yohimbine

1994
Species orthologs of the alpha-2A adrenergic receptor: the pharmacological properties of the bovine and rat receptors differ from the human and porcine receptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:2

    Topics: Animals; Binding Sites; Cattle; Cell Line; Dioxanes; Humans; Idazoxan; Rats; Receptors, Adrenergic, alpha-2; Species Specificity; Swine; Yohimbine

1994
Alpha 2-adrenoceptor antagonist potencies of two hydroxylated metabolites of yohimbine.
    British journal of pharmacology, 1993, Volume: 108, Issue:4

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Blood Platelets; Blood Proteins; Brimonidine Tartrate; Cell Membrane; Dioxanes; Epinephrine; Humans; Hydroxylation; Idazoxan; In Vitro Techniques; Lipolysis; Male; Platelet Aggregation; Protein Binding; Quinoxalines; Yohimbine

1993
Estradiol attenuates alpha 2-adrenoceptor-mediated inhibition of hypothalamic norepinephrine release.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:8

    Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Dioxanes; Estradiol; Female; Hypothalamus; Idazoxan; Norepinephrine; Ovariectomy; Potassium Chloride; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Yohimbine

1993
Motor and cardiovascular effects of selective alpha 2-adrenoceptor antagonists in the decerebrated rabbit.
    European journal of pharmacology, 1993, Jun-24, Volume: 237, Issue:2-3

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Decerebrate State; Dioxanes; Electric Stimulation; Female; Heart Rate; Idazoxan; Injections, Spinal; Male; Motor Neurons; Rabbits; Reflex; Retrospective Studies; Sural Nerve; Yohimbine

1993
Alpha 2A adrenoceptors and non-adrenergic idazoxan binding sites in calf brain and retina are distinct from those in human brain.
    Neurochemistry international, 1993, Volume: 22, Issue:5

    Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cattle; Cell Membrane; Dioxanes; Frontal Lobe; Humans; Idazoxan; Receptors, Adrenergic, alpha; Retina; Species Specificity; Yohimbine

1993
Determination on functional basis of presynaptic alpha 2-adrenoceptor subtypes in guinea-pig duodenum.
    Neuroscience letters, 1996, May-24, Volume: 210, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Cholinergic Fibers; Duodenum; Electric Stimulation; Gastrointestinal Motility; Guinea Pigs; Idazoxan; Imidazoles; Indoles; Isoindoles; Isoquinolines; Male; Medetomidine; Muscle Contraction; Nordefrin; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Receptors, Adrenergic, alpha-2; Synaptic Membranes; Vasoconstrictor Agents; Xylazine; Yohimbine

1996
alpha 2A/D-Adrenoceptor subtype predominates also in the neonatal rat spinal cord.
    Brain research. Developmental brain research, 1996, Jun-14, Volume: 94, Issue:1

    Topics: Adrenergic alpha-Agonists; Age Factors; Animals; Animals, Newborn; Female; Idazoxan; Male; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Spinal Cord; Tritium; Yohimbine

1996
Buffers differentially alter the binding of [3H]rauwolscine and [3H]RX821002 to the alpha-2 adrenergic receptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 278, Issue:3

    Topics: Animals; Buffers; CHO Cells; Cricetinae; Humans; Idazoxan; Kinetics; Opossums; Oxymetazoline; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Species Specificity; Yohimbine

1996
Alpha-adrenoceptors in equine digital veins: evidence for the presence of both alpha1 and alpha2-receptors mediating vasoconstriction.
    Journal of veterinary pharmacology and therapeutics, 1997, Volume: 20, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Binding, Competitive; Brimonidine Tartrate; Dopamine; Horses; Idazoxan; In Vitro Techniques; Isometric Contraction; Methoxamine; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Vasoconstriction; Veins; Yohimbine

1997
Expression of functional alpha2-adrenergic receptor subtypes in human corpus cavernosum and in cultured trabecular smooth muscle cells.
    Receptors & signal transduction, 1997, Volume: 7, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Binding, Competitive; Brimonidine Tartrate; Cells, Cultured; Colforsin; Cyclic AMP; Humans; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Penis; Quinoxalines; Radioisotopes; Receptors, Adrenergic, alpha-2; Ribonucleases; RNA, Messenger; Yohimbine

1997
Different apparent modes of inhibition of alpha2A-adrenoceptor by alpha2-adrenoceptor antagonists.
    European journal of pharmacology, 1997, Sep-17, Volume: 335, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Humans; Idazoxan; Quinolizines; Receptors, Adrenergic, alpha-2; Tritium; Tumor Cells, Cultured; Yohimbine

1997
[3H]RS79948-197 binding to human, rat, guinea pig and pig alpha2A-, alpha2B- and alpha2C-adrenoceptors. Comparison with MK912, RX821002, rauwolscine and yohimbine.
    European journal of pharmacology, 1998, Feb-05, Volume: 343, Issue:1

    Topics: Adrenergic Agents; Animals; Guinea Pigs; Humans; Idazoxan; Isoquinolines; Naphthyridines; Quinolizines; Rats; Receptors, Adrenergic, alpha-2; Swine; Yohimbine

1998
Characterization of the allosteric interactions between antagonists and amiloride analogues at the human alpha2A-adrenergic receptor.
    Molecular pharmacology, 1998, Volume: 53, Issue:5

    Topics: Adrenergic alpha-Antagonists; Allosteric Regulation; Amiloride; Animals; CHO Cells; Cricetinae; Humans; Idazoxan; Protein Binding; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

1998
Hypercapnia-induced long-term depression of respiratory activity requires alpha2-adrenergic receptors.
    Journal of applied physiology (Bethesda, Md. : 1985), 1998, Volume: 84, Issue:6

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Carbon Dioxide; Hypercapnia; Hypoglossal Nerve; Idazoxan; Male; Norepinephrine; Phrenic Nerve; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Respiratory Mechanics; Vagotomy; Yohimbine

1998
Effects of alpha2-adrenoceptor antagonists on metabolic processes of swine: II. Nitrogen balance responses.
    Journal of animal science, 1998, Volume: 76, Issue:7

    Topics: Administration, Oral; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animal Feed; Animals; Digestion; Dose-Response Relationship, Drug; Ethanolamines; Idazoxan; Injections, Subcutaneous; Linear Models; Male; Nitrogen; Random Allocation; Swine; Yohimbine

1998
Actions of alpha2 adrenoceptor ligands at alpha2A and 5-HT1A receptors: the antagonist, atipamezole, and the agonist, dexmedetomidine, are highly selective for alpha2A adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brimonidine Tartrate; CHO Cells; Cricetinae; Guanfacine; Humans; Idazoxan; Imidazoles; Ligands; Medetomidine; Quinoxalines; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Yohimbine

1998
Prejunctional alpha2A-autoreceptors in the human gastric and ileocolic arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:2

    Topics: Adrenergic alpha-Antagonists; Aged; Arteries; Autoreceptors; Colon; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gastric Mucosa; Humans; Idazoxan; Ileum; In Vitro Techniques; Male; Middle Aged; Neuromuscular Junction; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha-2; Spiro Compounds; Stomach; Tritium; Yohimbine

1998
Adrenergic alpha2C-receptors reside in rat striatal GABAergic projection neurons: comparison of radioligand binding and immunohistochemistry.
    Neuroscience, 1999, Volume: 93, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Antibodies; Autoradiography; Binding, Competitive; Brain Chemistry; Calbindin 1; Calbindin 2; Calbindins; Corpus Striatum; gamma-Aminobutyric Acid; Idazoxan; Immunohistochemistry; Male; Neurons; Norepinephrine; Parvalbumins; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; S100 Calcium Binding Protein G; Tissue Fixation; Tritium; Yohimbine

1999
Non-adrenergic binding of [3H]atipamezole in rat kidney--regional distribution and comparison to alpha2-adrenoceptors.
    British journal of pharmacology, 1999, Volume: 128, Issue:6

    Topics: Animals; Autoradiography; Binding Sites; Binding, Competitive; Female; Idazoxan; Imidazoles; Kidney; Male; Membranes; Monoamine Oxidase; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

1999
Clozapine reversal of the deficits in coordinated movement induced by D2 receptor blockade does not depend upon antagonism of alpha2 adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:6

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Ataxia; Clozapine; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Haloperidol; Idazoxan; Loxapine; Male; Muscarinic Antagonists; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Scopolamine; Yohimbine

1999
Ligand recognition of serine-cysteine amino acid exchanges in transmembrane domain 5 of alpha2-adrenergic receptors by UK 14,304.
    Journal of neurochemistry, 2000, Volume: 74, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Chlorpromazine; CHO Cells; Cricetinae; Cysteine; Dopamine Antagonists; Humans; Idazoxan; Ligands; Mice; Models, Molecular; Molecular Sequence Data; Oxymetazoline; Protein Structure, Tertiary; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Sequence Homology, Amino Acid; Serine; Transfection; Tritium; Yohimbine

2000
Synthesis and alpha-adrenergic binding ligand affinities of 2-iminoimidazolidine derivatives.
    Chemical & pharmaceutical bulletin, 2000, Volume: 48, Issue:5

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Idazoxan; Imidazoles; In Vitro Techniques; Ligands; Magnetic Resonance Spectroscopy; Prazosin; Rats; Receptors, Adrenergic, alpha-2; Spectrophotometry, Infrared; Yohimbine

2000
Inverse agonism at alpha(2)-adrenoceptors in native tissue.
    European journal of pharmacology, 2000, Jun-16, Volume: 398, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Brain; Dose-Response Relationship, Drug; Guanosine Triphosphate; Idazoxan; Kinetics; Protein Binding; Quinolizines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

2000
Agonist trafficking of G(i/o)-mediated alpha(2A)-adrenoceptor responses in HEL 92.1.7 cells.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Biological Transport; Calcium; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Epinephrine; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Idazoxan; Pertussis Toxin; Propranolol; Receptors, Adrenergic, alpha-2; Tumor Cells, Cultured; Virulence Factors, Bordetella; Yohimbine

2001
The alpha 2 adrenoceptor antagonists RX 821002 and yohimbine delay-dependently impair choice accuracy in a delayed non-matching-to-position task in rats.
    Psychopharmacology, 2001, Volume: 155, Issue:4

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Idazoxan; Male; Muscarinic Antagonists; Psychomotor Performance; Rats; Scopolamine; Yohimbine

2001
Inhibition of pilocarpine-induced salivation in rats by central noradrenaline.
    Archives of oral biology, 2002, Volume: 47, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Idazoxan; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscarinic Agonists; Norepinephrine; Pilocarpine; Prazosin; Rats; Rats, Sprague-Dawley; Saliva; Salivation; Statistics as Topic; Yohimbine

2002
Central alpha(2) adrenergic receptors and cholinergic-induced salivation in rats.
    Brain research bulletin, 2003, Jan-30, Volume: 59, Issue:5

    Topics: Adrenergic alpha-Antagonists; Animals; Brain; Idazoxan; Imidazoles; Injections, Intraperitoneal; Injections, Intraventricular; Male; Muscarinic Agonists; Pilocarpine; Prazosin; Rats; Receptors, Adrenergic, alpha-2; Salivation; Sympatholytics; Yohimbine

2003
Regional distribution of alpha(2C)-adrenoceptors in brain and spinal cord of control mice and transgenic mice overexpressing the alpha(2C)-subtype: an autoradiographic study with [(3)H]RX821002 and [(3)H]rauwolscine.
    Neuroscience, 2003, Volume: 117, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brain; Female; Idazoxan; Mice; Mice, Inbred Strains; Mice, Transgenic; Neurons; Norepinephrine; Radioligand Assay; Receptors, Adrenergic, alpha-2; Spinal Cord; Synaptic Transmission; Tritium; Up-Regulation; Yohimbine

2003
[Ethyl-3H]RS-79948-197 alpha2-adrenoceptor autoradiography validation in alpha2-adrenoceptor knockout mice.
    European journal of pharmacology, 2004, Aug-30, Volume: 497, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Autoradiography; Binding Sites; Binding, Competitive; Cerebral Cortex; Idazoxan; In Vitro Techniques; Isoquinolines; Ligands; Mice; Mice, Knockout; Naphthyridines; Oxymetazoline; Phentolamine; Prazosin; Putamen; Radioligand Assay; Receptors, Adrenergic, alpha-2; Tritium; Yohimbine

2004
Long-lasting effects of yohimbine on the ejaculatory function in male dogs.
    Biomedical research (Tokyo, Japan), 2005, Volume: 26, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dogs; Ejaculation; Idazoxan; Male; Penile Erection; Sexual Behavior, Animal; Time Factors; Yohimbine

2005
Probable involvement of alpha(2C)-adrenoceptor subtype and endogenous opioid peptides in the peripheral antinociceptive effect induced by xylazine.
    European journal of pharmacology, 2009, Apr-17, Volume: 608, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Analgesics; Animals; Dinoprostone; Dose-Response Relationship, Drug; Hyperalgesia; Idazoxan; Imidazoles; Leucine; Male; Naloxone; Opioid Peptides; Pain; Pain Measurement; Rats; Rats, Wistar; Xylazine; Yohimbine

2009
α2-adrenergic drugs modulate the binding of [18F]fallypride to dopamine D2/3 receptors in striatum of living mouse.
    Synapse (New York, N.Y.), 2010, Volume: 64, Issue:8

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzamides; Binding, Competitive; Brain Mapping; Clonidine; Corpus Striatum; Dopamine; Female; Idazoxan; Mice; Mice, Inbred BALB C; Positron-Emission Tomography; Pyrrolidines; Receptors, Adrenergic, alpha-2; Receptors, Dopamine D2; Yohimbine

2010
Inhibition of sodium appetite by lipopolysaccharide: involvement of alpha2-adrenoceptors.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2011, Volume: 301, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Appetite; Blood Pressure; Body Temperature; Dose-Response Relationship, Drug; Gastric Emptying; Heart Rate; Idazoxan; Injections, Intraperitoneal; Lipopolysaccharides; Male; Models, Animal; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Sodium Chloride, Dietary; Yohimbine

2011
Commissural nucleus of the solitary tract regulates the antihypertensive effects elicited by moxonidine.
    Neuroscience, 2013, Oct-10, Volume: 250

    Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Antihypertensive Agents; Blood Pressure; Consciousness; Fourth Ventricle; Heart Rate; Idazoxan; Imidazoles; Injections; Injections, Intraventricular; Male; Neurons; Rats; Rats, Inbred SHR; Rats, Wistar; Solitary Nucleus; Stereotaxic Techniques; Yohimbine

2013