rx 821002 has been researched along with wb 4101 in 12 studies
Studies (rx 821002) | Trials (rx 821002) | Recent Studies (post-2010) (rx 821002) | Studies (wb 4101) | Trials (wb 4101) | Recent Studies (post-2010) (wb 4101) |
---|---|---|---|---|---|
317 | 0 | 45 | 477 | 1 | 34 |
Protein | Taxonomy | rx 821002 (IC50) | wb 4101 (IC50) |
---|---|---|---|
Alpha-1A adrenergic receptor | Homo sapiens (human) | 0.001 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (25.00) | 18.2507 |
2000's | 4 (33.33) | 29.6817 |
2010's | 5 (41.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Denis-Pouxviel, C; Devedjian, JC; Esclapez, F; Paris, H | 1 |
Neubig, RR; Porter, AC; Uhlén, S | 1 |
Caramona, MM; Figueiredo, IV; Guimarães, S; Moura, D; Paiva, MQ | 1 |
Antunes-Rodrigues, J; Corrêa, FM; Crippa, GE; Fernandes, KB; Tavares, RF | 1 |
Corrêa, FM; Fernandes, KB; Resstel, LB | 1 |
Alves, FH; Corrêa, FM; Crestani, CC; Tavares, RF | 1 |
Alves, FH; Correa, FM; Crestani, CC; Resstel, LB | 3 |
Alves, FH; Correa, FM; Crestani, CC; Resstel, LB; Scopinho, AA | 1 |
Côrrea, FM; Crestani, CC; Fabri, DR; Gomes, FV; Hott, SC; Reis, DG; Resstel, LB | 1 |
de Aguiar Corrêa, FM; Fortaleza, EA; Scopinho, AA | 1 |
12 other study(ies) available for rx 821002 and wb 4101
Article | Year |
---|---|
Further characterization of human alpha 2-adrenoceptor subtypes: [3H]RX821002 binding and definition of additional selective drugs.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cell Line; Dioxanes; Humans; Idazoxan; Plasmids; Radioligand Assay; Receptors, Adrenergic, alpha; Transfection | 1994 |
The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Dibenzazepines; Humans; Imidazoles; Indoles; Isoindoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2 | 1994 |
Prejunctional alpha2A-autoreceptors in the human gastric and ileocolic arteries.
Topics: Adrenergic alpha-Antagonists; Aged; Arteries; Autoreceptors; Colon; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gastric Mucosa; Humans; Idazoxan; Ileum; In Vitro Techniques; Male; Middle Aged; Neuromuscular Junction; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha-2; Spiro Compounds; Stomach; Tritium; Yohimbine | 1998 |
Mechanisms involved in the pressor response to noradrenaline injection into the cingulate cortex of unanesthetized rats.
Topics: Adrenergic alpha-Antagonists; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Blood Pressure; Dioxanes; Dose-Response Relationship, Drug; Ganglionic Blockers; Gyrus Cinguli; Heart Rate; Hypophysectomy; Idazoxan; Male; Mecamylamine; Microinjections; Norepinephrine; Phenoxybenzamine; Rats; Rats, Wistar | 2003 |
alpha-Adrenergic and muscarinic cholinergic receptors are not involved in the modulation of the parasympathetic baroreflex by the medial prefrontal cortex in rats.
Topics: Animals; Atropine; Baroreflex; Cobalt; Dioxanes; Idazoxan; Male; Parasympathetic Nervous System; Phenylephrine; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic | 2005 |
Role of the bed nucleus of the stria terminalis in the cardiovascular responses to acute restraint stress in rats.
Topics: Animals; Blood Pressure; Cardiovascular System; Cobalt; Dioxanes; Heart Rate; Idazoxan; Male; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Restraint, Physical; Stress, Psychological; Synaptic Transmission; Thalamic Nuclei; Tropanes | 2009 |
Insular cortex alpha1-adrenoceptors modulate the parasympathetic component of the baroreflex in unanesthetized rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Baroreflex; Blood Pressure; Cerebral Cortex; Dioxanes; Heart Rate; Idazoxan; Male; Norepinephrine; Parasympathetic Nervous System; Phenylephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Regression Analysis; Synaptic Transmission | 2009 |
Bed nucleus of the stria terminalis α1- and α2-adrenoceptors differentially modulate the cardiovascular responses to exercise in rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Dioxanes; Exercise Tolerance; Idazoxan; Male; Physical Conditioning, Animal; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Septal Nuclei; Synaptic Transmission | 2011 |
Lateral septal area α1- and α2-adrenoceptors differently modulate baroreflex activity in unanaesthetized rats.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Baroreflex; Blood Pressure; Dioxanes; Heart Rate; Idazoxan; Male; Norepinephrine; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Septal Nuclei; Synaptic Transmission; Tachycardia | 2012 |
Both α1- and β1-adrenoceptors in the bed nucleus of the stria terminalis are involved in the expression of conditioned contextual fear.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Conditioning, Psychological; Dioxanes; Electroshock; Fear; Idazoxan; Imidazoles; Male; Phentolamine; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Septal Nuclei | 2012 |
α1 and α2-adrenoceptors in the medial amygdaloid nucleus modulate differently the cardiovascular responses to restraint stress in rats.
Topics: Adrenergic alpha-Antagonists; Amygdala; Animals; Blood Pressure; Dioxanes; Heart Rate; Idazoxan; Male; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Restraint, Physical; Stress, Psychological | 2012 |
Both α1- and α2-adrenoceptors in the insular cortex are involved in the cardiovascular responses to acute restraint stress in rats.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Cerebral Cortex; Dioxanes; Heart Rate; Idazoxan; Male; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Restraint, Physical; Stress, Mechanical; Synaptic Transmission | 2014 |