Page last updated: 2024-09-02

rx 821002 and wb 4101

rx 821002 has been researched along with wb 4101 in 12 studies

Compound Research Comparison

Studies
(rx 821002)
Trials
(rx 821002)
Recent Studies (post-2010)
(rx 821002)
Studies
(wb 4101)
Trials
(wb 4101)
Recent Studies (post-2010) (wb 4101)
317045477134

Protein Interaction Comparison

ProteinTaxonomyrx 821002 (IC50)wb 4101 (IC50)
Alpha-1A adrenergic receptorHomo sapiens (human)0.001

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (25.00)18.2507
2000's4 (33.33)29.6817
2010's5 (41.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Denis-Pouxviel, C; Devedjian, JC; Esclapez, F; Paris, H1
Neubig, RR; Porter, AC; Uhlén, S1
Caramona, MM; Figueiredo, IV; Guimarães, S; Moura, D; Paiva, MQ1
Antunes-Rodrigues, J; Corrêa, FM; Crippa, GE; Fernandes, KB; Tavares, RF1
Corrêa, FM; Fernandes, KB; Resstel, LB1
Alves, FH; Corrêa, FM; Crestani, CC; Tavares, RF1
Alves, FH; Correa, FM; Crestani, CC; Resstel, LB3
Alves, FH; Correa, FM; Crestani, CC; Resstel, LB; Scopinho, AA1
Côrrea, FM; Crestani, CC; Fabri, DR; Gomes, FV; Hott, SC; Reis, DG; Resstel, LB1
de Aguiar Corrêa, FM; Fortaleza, EA; Scopinho, AA1

Other Studies

12 other study(ies) available for rx 821002 and wb 4101

ArticleYear
Further characterization of human alpha 2-adrenoceptor subtypes: [3H]RX821002 binding and definition of additional selective drugs.
    European journal of pharmacology, 1994, Jan-24, Volume: 252, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Cell Line; Dioxanes; Humans; Idazoxan; Plasmids; Radioligand Assay; Receptors, Adrenergic, alpha; Transfection

1994
The novel alpha-2 adrenergic radioligand [3H]-MK912 is alpha-2C selective among human alpha-2A, alpha-2B and alpha-2C adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; CHO Cells; Cricetinae; Dibenzazepines; Humans; Imidazoles; Indoles; Isoindoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2

1994
Prejunctional alpha2A-autoreceptors in the human gastric and ileocolic arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:2

    Topics: Adrenergic alpha-Antagonists; Aged; Arteries; Autoreceptors; Colon; Dioxanes; Dopamine Antagonists; Dose-Response Relationship, Drug; Electric Stimulation; Female; Gastric Mucosa; Humans; Idazoxan; Ileum; In Vitro Techniques; Male; Middle Aged; Neuromuscular Junction; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha-2; Spiro Compounds; Stomach; Tritium; Yohimbine

1998
Mechanisms involved in the pressor response to noradrenaline injection into the cingulate cortex of unanesthetized rats.
    Neuropharmacology, 2003, Volume: 44, Issue:6

    Topics: Adrenergic alpha-Antagonists; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Blood Pressure; Dioxanes; Dose-Response Relationship, Drug; Ganglionic Blockers; Gyrus Cinguli; Heart Rate; Hypophysectomy; Idazoxan; Male; Mecamylamine; Microinjections; Norepinephrine; Phenoxybenzamine; Rats; Rats, Wistar

2003
alpha-Adrenergic and muscarinic cholinergic receptors are not involved in the modulation of the parasympathetic baroreflex by the medial prefrontal cortex in rats.
    Life sciences, 2005, Aug-12, Volume: 77, Issue:13

    Topics: Animals; Atropine; Baroreflex; Cobalt; Dioxanes; Idazoxan; Male; Parasympathetic Nervous System; Phenylephrine; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic

2005
Role of the bed nucleus of the stria terminalis in the cardiovascular responses to acute restraint stress in rats.
    Stress (Amsterdam, Netherlands), 2009, Volume: 12, Issue:3

    Topics: Animals; Blood Pressure; Cardiovascular System; Cobalt; Dioxanes; Heart Rate; Idazoxan; Male; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Restraint, Physical; Stress, Psychological; Synaptic Transmission; Thalamic Nuclei; Tropanes

2009
Insular cortex alpha1-adrenoceptors modulate the parasympathetic component of the baroreflex in unanesthetized rats.
    Brain research, 2009, Oct-27, Volume: 1295

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Baroreflex; Blood Pressure; Cerebral Cortex; Dioxanes; Heart Rate; Idazoxan; Male; Norepinephrine; Parasympathetic Nervous System; Phenylephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Regression Analysis; Synaptic Transmission

2009
Bed nucleus of the stria terminalis α1- and α2-adrenoceptors differentially modulate the cardiovascular responses to exercise in rats.
    Neuroscience, 2011, Mar-17, Volume: 177

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Dioxanes; Exercise Tolerance; Idazoxan; Male; Physical Conditioning, Animal; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Septal Nuclei; Synaptic Transmission

2011
Lateral septal area α1- and α2-adrenoceptors differently modulate baroreflex activity in unanaesthetized rats.
    Experimental physiology, 2012, Volume: 97, Issue:9

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Baroreflex; Blood Pressure; Dioxanes; Heart Rate; Idazoxan; Male; Norepinephrine; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Septal Nuclei; Synaptic Transmission; Tachycardia

2012
Both α1- and β1-adrenoceptors in the bed nucleus of the stria terminalis are involved in the expression of conditioned contextual fear.
    British journal of pharmacology, 2012, Volume: 167, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Conditioning, Psychological; Dioxanes; Electroshock; Fear; Idazoxan; Imidazoles; Male; Phentolamine; Propanolamines; Propranolol; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-1; Septal Nuclei

2012
α1 and α2-adrenoceptors in the medial amygdaloid nucleus modulate differently the cardiovascular responses to restraint stress in rats.
    Pharmacological research, 2012, Volume: 66, Issue:2

    Topics: Adrenergic alpha-Antagonists; Amygdala; Animals; Blood Pressure; Dioxanes; Heart Rate; Idazoxan; Male; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Restraint, Physical; Stress, Psychological

2012
Both α1- and α2-adrenoceptors in the insular cortex are involved in the cardiovascular responses to acute restraint stress in rats.
    PloS one, 2014, Volume: 9, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular System; Cerebral Cortex; Dioxanes; Heart Rate; Idazoxan; Male; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Restraint, Physical; Stress, Mechanical; Synaptic Transmission

2014